List of works - Ari Koskinen

3-Heterocycle-phenyl N-alkylcarbamates as FAAH inhibitors: design, synthesis and 3D-QSAR studies.

scientific article published in February 2010

An enantioselective synthesis of the C(33)–C(37) fragment of Amphotericin B ⬇️

scientific article published on September 21, 2003

Asymmetric synthesis of Pachastrissamine (Jaspine B) and its diastereomers via η3-allylpalladium intermediates

scientific article published on 24 January 2011

Binding of CGRP analogs and their effect on adenylate cyclase activity in porcine iris-ciliary body

scientific article published on 01 December 1998

Boron enolate chemistry toward the syntheses of polyketide stereotetrads

scientific article

Calyculins and related marine natural products as serine-threonine protein phosphatase PP1 and PP2A inhibitors and total syntheses of calyculin A, B, and C.

scientific article published on 21 January 2010

Catalytic activity dependency on catalyst components in aerobic copper-TEMPO oxidation.

scientific article published in October 2009

Concise, stereodivergent and highly stereoselective synthesis of cis- and trans-2-substituted 3-hydroxypiperidines - development of a phosphite-driven cyclodehydration.

scientific article published on 11 February 2014

Conformational ensembles of flexible beta-turn mimetics in DMSO-d6.

scientific article published on 11 March 2010

Conversion of carbonyl compounds to alkynes: general overview and recent developments.

scientific article published on 24 March 2010

Design, synthesis, and in vitro evaluation of carbamate derivatives of 2-benzoxazolyl- and 2-benzothiazolyl-(3-hydroxyphenyl)-methanones as novel fatty acid amide hydrolase inhibitors.

scientific article published in August 2007

Diastereoselective intramolecular allyl transfer from allyl carbamate accompanied by 5-endo-trig ring closure.

scientific article published on 22 January 2013

Diastereoselective synthesis of vicinal amino alcohols

scientific article published on 25 April 2012

Editorial to the Special Issue "Total Synthesis of Natural Products: A Themed Issue Dedicated to Professor Dr. Dieter Schinzer for His 65th Birthday"

scientific article published on 10 December 2020

Efficient, stereodivergent access to 3-piperidinols by traceless P(OEt)3 cyclodehydration

scientific article published on 03 October 2013

Garner's aldehyde as a versatile intermediate in the synthesis of enantiopure natural products

scientific article

Highly enantioselective conjugate addition of thiols using mild scandium triflate catalysis

scientific article published on 06 June 2007

Locked conformations for proline pyrrolidine ring: synthesis and conformational analysis of cis- and trans-4-tert-butylprolines.

scientific article published in August 2005

Novel crown ether and salen metal chelation driven molecular pincers

scientific article published on 01 September 2006

Origins of Stereoselectivity in the Corey-Chaykovsky Reaction. Insights from Quantum Chemistry

scientific article published on 01 June 1999

Pharmacological importance of optically active tetrahydro-β-carbolines and synthetic approaches to create the C1 stereocenter

scientific article

Polyketide stereotetrads in natural products.

scientific article

Rapid and practical synthesis of (−)-1-deoxyaltronojirimycin

scientific article published on 24 December 2010

Synthesis of quinolinyl and isoquinolinyl phenyl ketones as novel agonists for the cannabinoid CB2 receptor.

scientific article published on 12 May 2009

Synthesis of the C(26)-C(32) Oxazole Fragment of Calyculin C: A Test Case for Oxazole Syntheses

scientific article published on 01 January 1998

The 9-Phenyl-9-fluorenyl Group for Nitrogen Protection in Enantiospecific Synthesis ⬇️

scientific article published on September 17, 2010

The binding mode of calyculin A to protein phosphatase-1. A novel spiroketal vector model.

scientific article

The synthesis and biological evaluation of para-substituted phenolic N-alkyl carbamates as endocannabinoid hydrolyzing enzyme inhibitors.

scientific article

Total synthesis of amaminol A: establishment of the absolute stereochemistry

scientific article published on 23 October 2007

Towards the total synthesis of calyculin C: preparation of the C(9)-C(25) spiroketal-dipropionate unit.

scientific article published on 4 August 2010

List of works by Ari Koskinen

3-Heterocycle-phenyl N-alkylcarbamates as FAAH inhibitors: design, synthesis and 3D-QSAR studies.

An enantioselective synthesis of the C(33)–C(37) fragment of Amphotericin B ⬇️

Asymmetric synthesis of Pachastrissamine (Jaspine B) and its diastereomers via η3-allylpalladium intermediates

Binding of CGRP analogs and their effect on adenylate cyclase activity in porcine iris-ciliary body

Boron enolate chemistry toward the syntheses of polyketide stereotetrads

Calyculins and related marine natural products as serine-threonine protein phosphatase PP1 and PP2A inhibitors and total syntheses of calyculin A, B, and C.

Catalytic activity dependency on catalyst components in aerobic copper-TEMPO oxidation.

Concise, stereodivergent and highly stereoselective synthesis of cis- and trans-2-substituted 3-hydroxypiperidines - development of a phosphite-driven cyclodehydration.

Conformational ensembles of flexible beta-turn mimetics in DMSO-d6.

Conversion of carbonyl compounds to alkynes: general overview and recent developments.

Design, synthesis, and in vitro evaluation of carbamate derivatives of 2-benzoxazolyl- and 2-benzothiazolyl-(3-hydroxyphenyl)-methanones as novel fatty acid amide hydrolase inhibitors.

Diastereoselective intramolecular allyl transfer from allyl carbamate accompanied by 5-endo-trig ring closure.

Diastereoselective synthesis of vicinal amino alcohols

Editorial to the Special Issue "Total Synthesis of Natural Products: A Themed Issue Dedicated to Professor Dr. Dieter Schinzer for His 65th Birthday"

Efficient, stereodivergent access to 3-piperidinols by traceless P(OEt)3 cyclodehydration

Garner's aldehyde as a versatile intermediate in the synthesis of enantiopure natural products

Highly enantioselective conjugate addition of thiols using mild scandium triflate catalysis

Locked conformations for proline pyrrolidine ring: synthesis and conformational analysis of cis- and trans-4-tert-butylprolines.

Novel crown ether and salen metal chelation driven molecular pincers

Origins of Stereoselectivity in the Corey-Chaykovsky Reaction. Insights from Quantum Chemistry

Pharmacological importance of optically active tetrahydro-β-carbolines and synthetic approaches to create the C1 stereocenter

Polyketide stereotetrads in natural products.

Rapid and practical synthesis of (−)-1-deoxyaltronojirimycin

Synthesis of quinolinyl and isoquinolinyl phenyl ketones as novel agonists for the cannabinoid CB2 receptor.

Synthesis of the C(26)-C(32) Oxazole Fragment of Calyculin C: A Test Case for Oxazole Syntheses

The 9-Phenyl-9-fluorenyl Group for Nitrogen Protection in Enantiospecific Synthesis ⬇️

The binding mode of calyculin A to protein phosphatase-1. A novel spiroketal vector model.

The synthesis and biological evaluation of para-substituted phenolic N-alkyl carbamates as endocannabinoid hydrolyzing enzyme inhibitors.

Total synthesis of amaminol A: establishment of the absolute stereochemistry

Towards the total synthesis of calyculin C: preparation of the C(9)-C(25) spiroketal-dipropionate unit.