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List of works by Benoit Joseph

3-Aryl-2-quinolone derivatives: synthesis and characterization of in vitro and in vivo antitumor effects with emphasis on a new therapeutical target connected with cell migration

scientific article published in June 2002

Correction: Characterization of Transglutaminase 2 activity inhibitors in monocytes in vitro and their effect in a mouse model for multiple sclerosis

scientific article published in PLoS ONE

Cytotoxic nucleoside analogues: different strategies to improve their clinical efficacy.

scientific article published on January 2008

Impact of meriolins, a new class of cyclin-dependent kinase inhibitors, on malignant glioma proliferation and neo-angiogenesis.

scientific article

Indolobenzazepin-7-ones and 6-, 8-, and 9-membered ring derivatives as tubulin polymerization inhibitors: synthesis and structure--activity relationship studies

scientific article

Inhibition of hepatitis C virus NS5B polymerase by S-trityl-L-cysteine derivatives.

scientific article published on 12 January 2012

Meriolins (3-(pyrimidin-4-yl)-7-azaindoles): synthesis, kinase inhibitory activity, cellular effects, and structure of a CDK2/cyclin A/meriolin complex.

scientific article published on 31 January 2008

Meriolins, a new class of cell death inducing kinase inhibitors with enhanced selectivity for cyclin-dependent kinases

scientific article

N-&-N, a new class of cell death-inducing kinase inhibitors derived from the purine roscovitine

scientific article

New 1-arylindoles based serotonin 5-HT7 antagonists. Synthesis and binding evaluation studies

scientific article published on 28 January 2014

New insights into homopiperazine-based 5-HT1A/5-HT7R ligands: synthesis and biological evaluation

scientific article published in June 2010

Room-Temperature and Transition-Metal-Free Intramolecular α-Arylation of Ketones: A Mild Access to Tetracyclic Indoles and 7-Azaindoles

scientific article published on 21 December 2018

Structure-activity relationship and multidrug resistance study of new S-trityl-L-cysteine derivatives as inhibitors of Eg5

scientific article

Structure-activity relationship of S-trityl-L-cysteine analogues as inhibitors of the human mitotic kinesin Eg5.

scientific article published on 12 February 2008

Synthesis and antiproliferative activity of clausine E, mukonine, and koenoline bioisosteres

scientific article published on 18 May 2007

Synthesis and antiproliferative evaluation of pyrazolo[1,5-a]-1,3,5-triazine myoseverin derivatives.

scientific article published on 10 March 2009

Synthesis and biological evaluation in rat and cat of [18F]12ST05 as a potential 5-HT6 PET radioligand

scientific article published on 21 September 2007

Synthesis and in vitro cytotoxic evaluation of N-substituted benzo[5,6]cycloheptal[b]indoles

scientific article published on 01 December 2000

Synthesis, cytotoxicity, DNA interaction and topoisomerase II inhibition properties of tetrahydropyrrolo[3,4-a]carbazole-1,3-dione and tetrahydropyrido-[3,2-b]pyrrolo[3,4-g]indole-1,3-dione derivatives.

scientific article published in June 2001

Targeting RNA structure in SMN2 reverses spinal muscular atrophy molecular phenotypes.

scientific article

Targeting low molecular weight cyclin E (LMW-E) in breast cancer.

scientific article published on 22 June 2011

Unexpected matrix interactions in liquid secondary ion mass spectrometry of two pyranosyl mercaptans

scientific article published on 01 May 2011

Use of ATP analogs to inhibit HIV-1 transcription

scientific article