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List of works by Nagavarakishore Pillarsetty

(124)I-iodopyridopyrimidinone for PET of Abl kinase-expressing tumors in vivo.

scientific article published on January 2010

(18)F-Based Pretargeted PET Imaging Based on Bioorthogonal Diels-Alder Click Chemistry.

scientific article published on 19 October 2015

(18)F-labeled-bioorthogonal liposomes for in vivo targeting

scientific article published on 7 November 2013

2-18F-Fluoropropionic acid as a PET imaging agent for prostate cancer.

scientific article published on 16 September 2009

A Chemical Biology Approach to the Chaperome in Cancer-HSP90 and Beyond

scientific article published on 01 April 2020

A One-Pot Radio-synthesis of [18 F]PARPi

scientific article published on 11 May 2020

A rapid bead-based radioligand binding assay for the determination of target-binding fraction and quality control of radiopharmaceuticals

scientific article published on 01 April 2019

An improved strategy for the synthesis of [¹⁸F]-labeled arabinofuranosyl nucleosides.

scientific article published on 18 July 2012

Antilipolytic drug boosts glucose metabolism in prostate cancer.

scientific article published on 28 February 2013

Building Blocks for the Construction of Bioorthogonally Reactive Peptides via Solid-Phase Peptide Synthesis.

scientific article published on 06 April 2014

Characterization of supramolecular (H2O)18 water morphology and water-methanol (H2O)15(CH3OH)3 clusters in a novel phosphorus functionalized trimeric amino acid host.

scientific article

Copper-64 labeled liposomes for imaging bone marrow.

scientific article published on 27 August 2016

Design and Synthesis of a Bombesin Peptide-Conjugated Tripodal Phosphino Dithioether Ligand Topology for the Stabilization of the fac-[M(CO)3]+ Core (M = 99 mTc or Re) ⬇️

scientific article published on May 18, 2011

Design, synthesis, and chemistry of sterically nondemanding primary bisphosphines

scientific article published on 01 January 2005

Efficient (18)F-labeling of large 37-amino-acid pHLIP peptide analogues and their biological evaluation.

scientific article

Erratum to: Repeatability of [68Ga]DKFZ11-PSMA PET Scans for Detecting Prostate-specific Membrane Antigen-positive Prostate Cancer

scientific article

First-in-Human Trial of Epichaperome-Targeted Positron Emission Tomography in Cancer Patients

scientific article published on 04 May 2020

Fluorine-labeled dasatinib nanoformulations as targeted molecular imaging probes in a PDGFB-driven murine glioblastoma model.

scientific article published on December 2012

Imaging Sigma-1 Receptor (S1R) Expression Using Iodine-124-Labeled 1-(4-Iodophenyl)-3-(2-adamantyl)guanidine ([124I]IPAG)

scientific article published on 01 April 2020

Improved radiosynthesis of 123I-MAPi, an Auger theranostic agent

scientific article published on 18 June 2020

Improved synthesis of 2'-deoxy-2'-[18F]-fluoro-1-beta-D-arabinofuranosyl-5-iodouracil ([18F]-FIAU).

scientific article published on 6 March 2010

In vitro and in vivo antitumor properties of tetrakis((trishydroxy- methyl)phosphine)gold(I) chloride.

scientific article published in March 2003

In vivo imaging of Bcr-Abl overexpressing tumors with a radiolabeled imatinib analog as an imaging surrogate for imatinib.

scientific article published on 15 July 2011

Increased KIT inhibition enhances therapeutic efficacy in gastrointestinal stromal tumor

scientific article

Influence of free fatty acids on glucose uptake in prostate cancer cells

scientific article published on 17 December 2013

Leveraging PET to image folate receptor α therapy of an antibody-drug conjugate

scientific article published on 28 August 2018

Monitoring the efficacy of adoptively transferred prostate cancer-targeted human T lymphocytes with PET and bioluminescence imaging.

scientific article published on 13 June 2008

Optimizing tumor targeting of the lipophilic EGFR-binding radiotracer SKI 243 using a liposomal nanoparticle delivery system ⬇️

scientific article published on February 10, 2011

Paradigms for Precision Medicine in Epichaperome Cancer Therapy

scientific article published on 24 October 2019

Pharmacologically controlling protein-protein interactions through epichaperomes for therapeutic vulnerability in cancer

scientific article published on 25 November 2021

Preclinical tolerance and pharmacokinetic assessment of MU-Gold, a novel chemotherapeutic agent, in laboratory dogs.

scientific article published in January 2003

Predicting gemcitabine delivery by 18F-FAC PET in murine models of pancreatic cancer

scientific article published on 09 July 2020

Pretargeting of internalizing trastuzumab and cetuximab with a 18F-tetrazine tracer in xenograft models

scientific article published on 2 December 2017

Radioiodinated PARP1 tracers for glioblastoma imaging

scientific article published on 4 September 2015

Radiosynthesis of the iodine-124 labeled Hsp90 inhibitor PU-H71.

scientific article published on 25 January 2016

Sustained ERK inhibition maximizes responses of BrafV600E thyroid cancers to radioiodine

scientific article published on 26 September 2016

Syntheses, in vitro and in vivo characterization of a 99mTc-(I)-tricarbonyl-benzylamino-dihydroxymethyl phosphine (NP(2)) chelate

scientific article published on 01 May 2003

Synthesis and biological evaluation of a fluorine-18 derivative of dasatinib.

scientific article published on 23 October 2007

Synthesis and characterization of (99m)Tc- and (188)Re-complexes with a diamido-dihydroxymethylenephosphine-based bifunctional chelating agent (N(2)P(2)-BFCA)

scientific article published on 01 January 2002

Synthesis and evaluation of (18)F-labeled ATP competitive inhibitors of topoisomerase II as probes for imaging topoisomerase II expression.

scientific article published on 8 September 2014

Synthesis and evaluation of 18F-labeled benzylguanidine analogs for targeting the human norepinephrine transporter

scientific article published on 31 October 2013

Synthesis and evaluation of [18F] labeled pyrimidine nucleosides for positron emission tomography imaging of herpes simplex virus 1 thymidine kinase gene expression.

scientific article published on August 2006

Synthesis and evaluation of an (18)F-labeled pyrimidine-pyridine amine for targeting CXCR4 receptors in gliomas.

scientific article published on 14 May 2016

Synthesis of novel PET tracer 124I-trametinib for MAPK/ERK kinase distribution and resistance monitoring

scientific article published on 22 May 2020

Target engagement imaging of PARP inhibitors in small-cell lung cancer.

scientific article published on 12 January 2018

Tetrahydroprotoberberine alkaloids with dopamine and σ receptor affinity.

scientific article published on 21 March 2016

The epichaperome is a mediator of toxic hippocampal stress and leads to protein connectivity-based dysfunction

scientific article published on 16 January 2020

The epichaperome is an integrated chaperome network that facilitates tumour survival

scientific article published on 05 October 2016

The synthesis and evaluation of N1-(4-(2-[18F]-fluoroethyl)phenyl)-N8-hydroxyoctanediamide ([18F]-FESAHA), a PET radiotracer designed for the delineation of histone deacetylase expression in cancer.

scientific article

Tumor-specific targeting with modified Sindbis viral vectors: evaluation with optical imaging and positron emission tomography in vivo.

scientific article published on April 2013

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