List of works - Antonio Garofalo

A critical study on the application of the zero-crossing derivative spectrophotometry to the photodegradation monitoring of lacidipine

scientific article published on 06 January 2006

An approach to the stereo-controlled synthesis of polycyclic derivatives of l-4-thiazolidinecarboxylic acid active against HIV-1 integrase

scientific article published on 15 June 2006

An update on small molecules targeting CXCR4 as starting points for the development of anti-cancer therapeutics

scientific article published on 12 August 2017

Antiproliferative action of pyrrolobenzoxazepine derivatives in cultured cells: Absence of correlation with binding to the peripheral-type benzodiazepine binding site ⬇️

scientific article published on February 15, 1998

Cytotoxic potential of novel 6,7-dimethoxyquinazolines ⬇️

scientific article published on December 21, 2011

Design and Synthesis of 3‐Carbamoylbenzoic Acid Derivatives as Inhibitors of Human Apurinic/Apyrimidinic Endonuclease 1 (APE1) ⬇️

scientific article published on September 5, 2012

Design and monitoring of photostability systems for amlodipine dosage forms.

scientific article published in October 2003

Discovery of a Novel Orally Active Small-Molecule gp130 Inhibitor for the Treatment of Ovarian Cancer ⬇️

scientific article published on March 27, 2013

Dual inhibition of survivin and MAOA synergistically impairs growth of PTEN-negative prostate cancer.

scientific article

Efficient and simple synthesis of 6-aryl-1,4-dimethyl-9H-carbazoles.

scientific article

Identification of two benzopyrroloxazines acting as selective GPER antagonists in breast cancer cells and cancer-associated fibroblasts

scientific article

New antipsychotic agents with serotonin and dopamine antagonist properties based on a pyrrolo[2,1-b][1,3]benzothiazepine structure.

scientific article published in September 1998

Photodegradation monitoring of amlodipine by derivative spectrophotometry.

scientific article published in January 2002

Pyrrolo[2,1-c][1,4]benzothiazines: synthesis, structure-activity relationships, molecular modeling studies, and cardiovascular activity.

scientific article published in October 1995

Pyrrolobenzothiazepinones and pyrrolobenzoxazepinones: novel and specific non-nucleoside HIV-1 reverse transcriptase inhibitors with antiviral activity.

scientific article published on July 1996

Quinoxalinylethylpyridylthioureas (QXPTs) as potent non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors. Further SAR studies and identification of a novel orally bioavailable hydrazine-based antiviral agent.

scientific article

Small molecule inhibitors of CXCR4.

scientific article

Stabilization of MDA-7/IL-24 for colon cancer therapy ⬇️

scientific article published on March 7, 2013

Synthesis and antitumor activities of a series of novel quinoxalinhydrazides.

scientific article published on 5 October 2006

Synthesis of esters of androgens with unsaturated fatty acids for androgen requiring therapy.

scientific article published on 22 October 2012

Synthesis of novel thiazolothiazepine based HIV-1 integrase inhibitors.

scientific article

Synthesis, biological activity, and SARs of pyrrolobenzoxazepine derivatives, a new class of specific "peripheral-type" benzodiazepine receptor ligands.

scientific article published on August 1996

List of works by Antonio Garofalo

A critical study on the application of the zero-crossing derivative spectrophotometry to the photodegradation monitoring of lacidipine

An approach to the stereo-controlled synthesis of polycyclic derivatives of l-4-thiazolidinecarboxylic acid active against HIV-1 integrase

An update on small molecules targeting CXCR4 as starting points for the development of anti-cancer therapeutics

Antiproliferative action of pyrrolobenzoxazepine derivatives in cultured cells: Absence of correlation with binding to the peripheral-type benzodiazepine binding site ⬇️

Cytotoxic potential of novel 6,7-dimethoxyquinazolines ⬇️

Design and Synthesis of 3‐Carbamoylbenzoic Acid Derivatives as Inhibitors of Human Apurinic/Apyrimidinic Endonuclease 1 (APE1) ⬇️

Design and monitoring of photostability systems for amlodipine dosage forms.

Discovery of a Novel Orally Active Small-Molecule gp130 Inhibitor for the Treatment of Ovarian Cancer ⬇️

Dual inhibition of survivin and MAOA synergistically impairs growth of PTEN-negative prostate cancer.

Efficient and simple synthesis of 6-aryl-1,4-dimethyl-9H-carbazoles.

Identification of two benzopyrroloxazines acting as selective GPER antagonists in breast cancer cells and cancer-associated fibroblasts

New antipsychotic agents with serotonin and dopamine antagonist properties based on a pyrrolo[2,1-b][1,3]benzothiazepine structure.

Photodegradation monitoring of amlodipine by derivative spectrophotometry.

Pyrrolo[2,1-c][1,4]benzothiazines: synthesis, structure-activity relationships, molecular modeling studies, and cardiovascular activity.

Pyrrolobenzothiazepinones and pyrrolobenzoxazepinones: novel and specific non-nucleoside HIV-1 reverse transcriptase inhibitors with antiviral activity.

Quinoxalinylethylpyridylthioureas (QXPTs) as potent non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors. Further SAR studies and identification of a novel orally bioavailable hydrazine-based antiviral agent.

Small molecule inhibitors of CXCR4.

Stabilization of MDA-7/IL-24 for colon cancer therapy ⬇️

Synthesis and antitumor activities of a series of novel quinoxalinhydrazides.

Synthesis of esters of androgens with unsaturated fatty acids for androgen requiring therapy.

Synthesis of novel thiazolothiazepine based HIV-1 integrase inhibitors.

Synthesis, biological activity, and SARs of pyrrolobenzoxazepine derivatives, a new class of specific "peripheral-type" benzodiazepine receptor ligands.