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List of works by Marianne Sadar

14-3-3 sigma increases the transcriptional activity of the androgen receptor in the absence of androgens.

scientific article published on 12 April 2007

Activation of the androgen receptor N-terminal domain by interleukin-6 via MAPK and STAT3 signal transduction pathways

scientific article (publication date: March 2002)

Advances in small molecule inhibitors of androgen receptor for the treatment of advanced prostate cancer.

scientific article

Amino-terminus domain of the androgen receptor as a molecular target to prevent the hormonal progression of prostate cancer.

scientific article

An androgen receptor N-terminal domain antagonist for treating prostate cancer.

scientific article published on 03 June 2013

An imaging agent to detect androgen receptor and its active splice variants in prostate cancer

scientific article published on July 2016

An orthotopic metastatic prostate cancer model in SCID mice via grafting of a transplantable human prostate tumor line.

scientific article published on November 2005

Analysis of the prostate cancer cell line LNCaP transcriptome using a sequencing-by-synthesis approach.

scientific article

Androgen Receptor Splice Variant 7 Drives the Growth of Castration Resistant Prostate Cancer without Being Involved in the Efficacy of Taxane Chemotherapy

scientific article published on 16 November 2018

Androgen receptor and its splice variants in prostate cancer

scientific article

Androgen receptor decoy molecules block the growth of prostate cancer

scholarly article

Androgen receptor targeted therapies in castration-resistant prostate cancer: Bench to clinic.

scientific article published on 14 June 2016

Androgen-independent induction of prostate-specific antigen gene expression via cross-talk between the androgen receptor and protein kinase A signal transduction pathways

scientific article published on 01 March 1999

Androgenic Induction of Prostate-specific Antigen Gene Is Repressed by Protein-Protein Interaction between the Androgen Receptor and AP-1/c-Jun in the Human Prostate Cancer Cell Line LNCaP ⬇️

scientific article (publication date: 11 July 1997)

Androgens and androgen receptor in prostate and ovarian malignancies.

scientific article

Butyrate analogue, isobutyramide, inhibits tumor growth and time to androgen-independent progression in the human prostate LNCaP tumor model

scientific article published on 01 June 1998

Characterization of niphatenones that inhibit androgen receptor N-terminal domain

scientific article

Combination therapy with androgen receptor N-terminal domain antagonist EPI-7170 and enzalutamide yields synergistic activity in AR-V7-positive prostate cancer

scientific article published on 30 July 2020

Connective tissue-activating peptide III: a novel blood biomarker for early lung cancer detection.

scientific article published on 04 May 2009

Cotargeting Androgen Receptor Splice Variants and mTOR Signaling Pathway for the Treatment of Castration-Resistant Prostate Cancer

scientific article published on 28 December 2015

Development of metastatic and non-metastatic tumor lines from a patient's prostate cancer specimen-identification of a small subpopulation with metastatic potential in the primary tumor.

scientific article published on November 2010

Directing abiraterone metabolism: balancing the scales between clinical relevance and experimental observation

scientific article published on 01 September 2016

Discovery of drugs that directly target the intrinsically disordered region of the androgen receptor

scientific article published on 26 February 2020

Does increased expression of glucocorticoid receptor support application of antagonists to this receptor for the treatment of castration resistant prostate cancer?

scientific article published on 13 June 2018

Enzalutamide and blocking androgen receptor in advanced prostate cancer: lessons learnt from the history of drug development of antiandrogens

scientific article published on 16 February 2018

FUS/TLS is a co-activator of androgen receptor in prostate cancer cells

scientific article

Incarnatapeptins A and B, Nonribosomal Peptides Discovered Using Genome Mining and 1H/15N HSQC-TOCSY

scientific article published on 13 April 2020

Induction of CYP1A1 by GABA receptor ligands

scientific article published on 01 December 1996

Induction of neuronal apoptosis inhibitory protein expression in response to androgen deprivation in prostate cancer

scientific article

Isolation and characterization of castration-resistant prostate cancer LNCaP95 clones

scientific article published on 20 September 2020

LNCaP Atlas: gene expression associated with in vivo progression to castration-recurrent prostate cancer

scientific article

Large scale phosphoproteome analysis of LNCaP human prostate cancer cells

scientific article

N-terminal targeting of androgen receptor variant enhances response of castration resistant prostate cancer to taxane chemotherapy

scientific article published on 15 November 2014

Niphatenones, glycerol ethers from the sponge Niphates digitalis block androgen receptor transcriptional activity in prostate cancer cells: structure elucidation, synthesis, and biological activity.

scientific article

Non-Genomic Actions of the Androgen Receptor in Prostate Cancer

scientific article published on 17 January 2017

Order within a Disordered Structure.

scientific article published in January 2018

Osteoblast-derived factors induce an expression signature that identifies prostate cancer metastasis and hormonal progression.

scientific article published on 7 April 2009

Osteoblast-derived factors induce androgen-independent proliferation and expression of prostate-specific antigen in human prostate cancer cells.

scientific article published on March 2004

Phenobarbital induction of CYP1A1 gene expression in a primary culture of rainbow trout hepatocytes.

scientific article published on July 1996

Phenobarbital induction of cytochrome P4501A1 is regulated by cAMP-dependent protein kinase-mediated signaling pathways in rainbow trout hepatocytes

scientific article published on 01 August 1996

Picrotoxin is a CYP1A1 inducer in rainbow trout hepatocytes

scientific article published on 01 September 1995

Prostate cancer: molecular biology of early progression to androgen independence.

scientific article

Ralaniten Sensitizes Enzalutamide-Resistant Prostate Cancer to Ionizing Radiation in Prostate Cancer Cells that Express Androgen Receptor Splice Variants

scientific article published on 21 July 2020

Regression of castrate-recurrent prostate cancer by a small-molecule inhibitor of the amino-terminus domain of the androgen receptor

scientific article

Sintokamide A Is a Novel Antagonist of Androgen Receptor That Uniquely Binds Activation Function-1 in Its Amino-terminal Domain.

scientific article published on 30 August 2016

Sintokamides A to E, chlorinated peptides from the sponge Dysidea sp. that inhibit transactivation of the N-terminus of the androgen receptor in prostate cancer cells.

scientific article

Small molecule inhibitors targeting the "achilles' heel" of androgen receptor activity

scientific article

Spongian diterpenoids inhibit androgen receptor activity

scientific article published on 26 February 2013

Structure-Activity Relationships for the Marine Natural Product Sintokamides: Androgen Receptor N-Terminus Antagonists of Interest for Treatment of Metastatic Castration-Resistant Prostate Cancer

scientific article published on 30 October 2020

Targeting Androgen Receptor Activation Function-1 with EPI to Overcome Resistance Mechanisms in Castration-Resistant Prostate Cancer

scientific article published on 2 May 2016

Targeting the N-Terminal Domain of the Androgen Receptor: A New Approach for the Treatment of Advanced Prostate Cancer.

scientific article published on 14 September 2016

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