List of works - Daniela Gündisch

3D QSAR analyses-guided rational design of novel ligands for the (alpha4)2(beta2)3 nicotinic acetylcholine receptor

scientific article published in May 2003

6H,13H-Pyrazino[1,2-a;4,5-a']diindole analogs: probing the pharmacophore for allosteric ligands of muscarinic M2 receptors

scientific article published on 4 January 2006

A hydrazide linker strategy for heterobivalent compounds as ortho- and allosteric ligands of acetylcholine-binding proteins

scientific article

Bispidine as a Privileged Scaffold

scientific article published on 15 September 2015

Carbazole Scaffold in Medicinal Chemistry and Natural Products: A Review from 2010-2015.

scientific article published on 15 September 2015

Cytisine-based nicotinic partial agonists as novel antidepressant compounds

scientific article published on 22 January 2009

Development of a 5-Hydroxytryptamine2A Receptor Binding Assay for High Throughput Screening Using 96-Well Microfilter Plates

scholarly article by Antje Harms et al published 1 August 2000 in Journal of Biomolecular Screening

Effects of Abeta1-42 fibrils and of the tetrapeptide Pr-IIGL on the phosphorylation state of the tau-protein and on the alpha7 nicotinic acetylcholine receptor in vitro

scientific article published in February 2005

Feasibility of 2-deoxy-2-[18F]fluoro-D-glucose- A85380-PET for imaging of human cardiac nicotinic acetylcholine receptors in vivo.

scientific article

Feasibility of [18F]-2-Fluoro-A85380-PET imaging of human vascular nicotinic acetylcholine receptors in vivo

scientific article published on May 2012

Halogenated and isosteric cytisine derivatives with increased affinity and functional activity at nicotinic acetylcholine receptors

scientific article

Heliotropiumides A and B, new phenolamides with N-carbamoyl putrescine moiety from Heliotropium foertherianum collected in Hawaii and their biological activities

scientific article published on 9 September 2017

In vitro characterization of 6-[18F]fluoro-A-85380, a high-affinity ligand for alpha4beta2* nicotinic acetylcholine receptors

scientific article published in February 2005

In vitro evaluation of nicotinic acetylcholine receptors with 2-[18F]F-A85380 in Parkinson's disease

scientific article

Nicotine decreases food intake through activation of POMC neurons

scientific article

Nicotinic acetylcholine receptor ligands, a patent review (2006 – 2011) ⬇️

scientific article published on December 1, 2011

Prenylated indole alkaloids from Flustra foliacea with subtype specific binding on NAChRs

scientific article

Semisynthetic analogues of toxiferine I and their pharmacological properties at α7 nAChRs, muscle-type nAChRs, and the allosteric binding site of muscarinic M2 receptors

scientific article

Smoking upregulates alpha4beta2* nicotinic acetylcholine receptors in the human brain

scientific article

Syntheses and evaluation of pyridazine and pyrimidine containing bioisosteres of (+/-)-pyrido[3.4-b]homotropane and pyrido-[3.4-b]tropane as novel nAChR ligands

scientific article published in January 2002

Synthesis and evaluation of phenylcarbamate derivatives as ligands for nicotinic acetylcholine receptors

scientific article published in September 2004

Synthesis and nicotinic binding studies on enantiopure diazine analogues of the novel (2-chloro-5-pyridyl)-9-azabicyclo[4.2.1]non-2-ene UB-165.

scientific article

Synthetic approaches and bio-distribution studies of [11C]methyl-phenidate.

scientific article published in January 2007

The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor (nAChR) ligands. Part 1: the influence of different hydrogen bond acceptor systems on alkyl and (hetero)aryl substituents

scientific article

The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor ligands. Part 2: carboxamide derivatives with different spacer motifs

scientific article

The twin drug approach for novel nicotinic acetylcholine receptor ligands

scientific article published on 20 June 2015

[Nuclides and tracers--mechanisms and application. Radiodiagnosis for peripheral organ diseases].

scientific article published in January 2005

List of works by Daniela Gündisch

3D QSAR analyses-guided rational design of novel ligands for the (alpha4)2(beta2)3 nicotinic acetylcholine receptor

6H,13H-Pyrazino[1,2-a;4,5-a']diindole analogs: probing the pharmacophore for allosteric ligands of muscarinic M2 receptors

A hydrazide linker strategy for heterobivalent compounds as ortho- and allosteric ligands of acetylcholine-binding proteins

Bispidine as a Privileged Scaffold

Carbazole Scaffold in Medicinal Chemistry and Natural Products: A Review from 2010-2015.

Cytisine-based nicotinic partial agonists as novel antidepressant compounds

Development of a 5-Hydroxytryptamine2A Receptor Binding Assay for High Throughput Screening Using 96-Well Microfilter Plates

Effects of Abeta1-42 fibrils and of the tetrapeptide Pr-IIGL on the phosphorylation state of the tau-protein and on the alpha7 nicotinic acetylcholine receptor in vitro

Feasibility of 2-deoxy-2-[18F]fluoro-D-glucose- A85380-PET for imaging of human cardiac nicotinic acetylcholine receptors in vivo.

Feasibility of [18F]-2-Fluoro-A85380-PET imaging of human vascular nicotinic acetylcholine receptors in vivo

Halogenated and isosteric cytisine derivatives with increased affinity and functional activity at nicotinic acetylcholine receptors

Heliotropiumides A and B, new phenolamides with N-carbamoyl putrescine moiety from Heliotropium foertherianum collected in Hawaii and their biological activities

In vitro characterization of 6-[18F]fluoro-A-85380, a high-affinity ligand for alpha4beta2* nicotinic acetylcholine receptors

In vitro evaluation of nicotinic acetylcholine receptors with 2-[18F]F-A85380 in Parkinson's disease

Nicotine decreases food intake through activation of POMC neurons

Nicotinic acetylcholine receptor ligands, a patent review (2006 – 2011) ⬇️

Prenylated indole alkaloids from Flustra foliacea with subtype specific binding on NAChRs

Semisynthetic analogues of toxiferine I and their pharmacological properties at α7 nAChRs, muscle-type nAChRs, and the allosteric binding site of muscarinic M2 receptors

Smoking upregulates alpha4beta2* nicotinic acetylcholine receptors in the human brain

Syntheses and evaluation of pyridazine and pyrimidine containing bioisosteres of (+/-)-pyrido[3.4-b]homotropane and pyrido-[3.4-b]tropane as novel nAChR ligands

Synthesis and evaluation of phenylcarbamate derivatives as ligands for nicotinic acetylcholine receptors

Synthesis and nicotinic binding studies on enantiopure diazine analogues of the novel (2-chloro-5-pyridyl)-9-azabicyclo[4.2.1]non-2-ene UB-165.

Synthetic approaches and bio-distribution studies of [11C]methyl-phenidate.

The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor (nAChR) ligands. Part 1: the influence of different hydrogen bond acceptor systems on alkyl and (hetero)aryl substituents

The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor ligands. Part 2: carboxamide derivatives with different spacer motifs

The twin drug approach for novel nicotinic acetylcholine receptor ligands

[Nuclides and tracers--mechanisms and application. Radiodiagnosis for peripheral organ diseases].