List of works - Kevin Burgess

3- and 5-Functionalized BODIPYs via the Liebeskind-Srogl reaction.

scientific article

4,4-Difluoro-4-bora-3a,4a-diaza-s-indacene (BODIPY) dyes modified for extended conjugation and restricted bond rotations

scientific article published on 01 May 2000

A Linker Scaffold to Present Dimers of Pharmacophores Prepared by Solid-Phase Syntheses

scientific article published on 01 December 2000

A Near-IR Fluorescent Dasatinib Derivative That Localizes in Cancer Cells

scientific article published on 01 April 2019

A Near-Infrared Fluorescence Chemosensor Based on Isothiocyanate-Aza-BODIPY for Cyanide Detection at the Parts per Billion Level: Applications in Buffer Media and Living Cell Imaging

scientific article published on 05 February 2019

A blue-to-red energy-transfer thymidine analogue that functions in DNA.

scientific article published in May 2004

A cheap, catalytic, scalable, and environmentally benign method for alkene epoxidations.

scientific article published in March 2001

A chemoselective route to β-enamino esters and thioesters

scientific article

A combinatorial approach for targeted delivery using small molecules and reversible masking to bypass nonspecific uptake in vivo

scientific article

A combinatorial method for solution-phase synthesis of labeled bivalent beta-turn mimics.

scientific article

A comparison between oxazoline-imidazolinylidene, -imidazolylidine, -benzimidazolylidene hydrogenation catalysts.

scientific article published on 19 September 2013

A diversity oriented synthesis of 3'-O-modified nucleoside triphosphates for DNA 'sequencing by synthesis'

scientific article published on 06 June 2006

A labeled guanidine ligand for studying sweet taste

scientific article published on 01 April 1998

A peptidomimetic of NT-3 acts as a TrkC antagonist

scientific article

A zwitterionic near-infrared dye linked TrkC targeting agent for imaging metastatic breast cancer

scientific article published on 03 August 2018

Aldol-type chirons from asymmetric hydrogenations of trisubstituted alkenes.

scientific article

Alpha,omega-functionalized 2,4-dimethylpentane dyads and 2,4,6-trimethylheptane triads through asymmetric hydrogenation.

scientific article

An agent for optical imaging of TrkC-expressing, breast cancer

scientific article published on 14 September 2017

An asymmetric hydrogenation route to (-)-spongidepsin

scientific article published on 01 October 2010

An iterative route to "decorated" ethylene glycol-based linkers

scientific article published on 07 March 2006

Anthranilic acid-containing cyclic tetrapeptides: at the crossroads of conformational rigidity and synthetic accessibility

scientific article

Asymmetric hydrogenation approaches to valuable, acyclic 1,3-hydroxymethyl chirons

scientific article published on 19 June 2008

Asymmetric hydrogenation routes to deoxypolyketide chirons

scientific article published on 01 January 2007

Asymmetric syntheses of α-methyl γ-amino acid derivatives

scientific article published on 18 August 2011

Aza-BODIPY dyes with enhanced hydrophilicity

scientific article published on June 2015

BODIPY dyes and their derivatives: syntheses and spectroscopic properties.

scientific article

BODIPY dyes in photodynamic therapy.

scientific article

Base dependence in copper-catalyzed Huisgen reactions: efficient formation of bistriazoles

scientific article published on 01 January 2007

Blocking Coronavirus 19 Infection via the SARS-CoV-2 Spike Protein: Initial Steps

scientific article published on 18 May 2020

Catalytic homogeneous asymmetric hydrogenations of largely unfunctionalized alkenes.

scientific article

Chiral imidazolylidine ligands for asymmetric hydrogenation of aryl alkenes

scientific article published on 01 September 2001

Chitosan-Coated Poly(lactic-co-glycolic acid)-Diiodinated boron-Dipyrromethene Nanoparticles Improve Tumor Selectivity and Stealth Properties in Photodynamic Cancer Therapy

scientific article published in July 2016

Click-Addressable Cassette for Photoaffinity Labeling.

scientific article published on 24 January 2018

Combinatorial assembly of small molecules into bivalent antagonists of TrkC or TrkA receptors

scientific article

Combinatorial technologies involving reiterative division/coupling/recombination: statistical considerations.

scientific article published in September 1994

Comparison Of Asymmetric Hydrogenations Of Unsaturated- Carboxylic Acids And -Esters.

scientific article published on February 2013

Comparisons of the conformational biases imposed by trans-2,3-methanomethionine and alpha-methylmethionine

scientific article published on 01 October 1997

Conjugation of Dasatinib with MHI-148 Has a Significant Advantageous Effect in Viability Assays for Glioblastoma Cells

scientific article published on 07 August 2019

Correction to A Near-IR Fluorescent Dasatinib Derivative That Localizes in Cancer Cells

scientific article published on 03 June 2019

Correlations between secondary structure- and protein-protein interface-mimicry: the interface mimicry hypothesis

scientific article published on 01 March 2019

Cyanine-Gemcitabine Conjugates as Targeted Theranostic Agents for Glioblastoma Tumor Cells

scientific article published on 11 October 2019

Cyclic semipeptoids: peptoid-organic hybrid macrocycles

scientific article published on 01 March 2006

Design criteria for minimalist mimics of protein-protein interface segments

scientific article published on 01 January 2019

DiSSiMiL: Diverse Small Size Mini-Libraries applied to simple and rapid epitope mapping of a monoclonal antibody.

scientific article

Double-targeting using a TrkC ligand conjugated to dipyrrometheneboron difluoride (BODIPY) based photodynamic therapy (PDT) agent.

scientific article published on 24 September 2013

Electronic effects steer the mechanism of asymmetric hydrogenations of unfunctionalized aryl-substituted alkenes.

scientific article published in December 2004

Elimination of residual natural nucleotides from 3'-O-modified-dNTP syntheses by enzymatic mop-up

scientific article published on 01 November 1998

Enantioselective hydrogenations of arylalkenes mediated by [Ir(cod) (JM-Phos) ]+ complexes.

scientific article

Energy transfer cassettes in silica nanoparticles target intracellular organelles.

scientific article published on 31 March 2011

Energy transfer dyads based on Nile Red.

scientific article published on November 2009

Enhanced antiopiate activity and enzyme resistance in a peptidomimetic of FMRFamide containing E-2,3-methanomethionine and E-2,3-methanophenylalanine

scientific article published on 01 January 1996

Enhanced antiopiate activity in peptidomimetics of FMRFamide containing Z-2,3-methanomethionine

scientific article published on 01 January 1993

Evaluating minimalist mimics by exploring key orientations on secondary structures (EKOS)

scientific article published on 14 October 2013

Expanding the scope of oligo-pyrrolinone-pyrrolidines as protein-protein interface mimics.

scientific article

Extended piperidine-piperidinone protein interface mimics

scientific article published on 13 April 2015

Facile macrocyclizations to beta-turn mimics with diverse structural, physical, and conformational properties.

scientific article

Filling gaps in asymmetric hydrogenation methods for acyclic stereocontrol: application to chirons for polyketide-derived natural products

scientific article published on 05 October 2012

Fluorescent amino- and thiopyronin dyes

scientific article published on 09 April 2008

Fluorescent indicators for intracellular pH.

scientific article published on May 2010

Functionalization of the 4,4-difluoro-4-bora-3a,4a-diaza-s-indacene (BODIPY) core

scientific article published on November 2007

Heterogeneous Phase Transfer Catalysis in Solid Phase Syntheses of Anth-Cyclic Tetrapeptides

scientific article

Heterovalent selectivity and the combinatorial advantage.

scientific article

Homo-Roche ester derivatives by asymmetric hydrogenation and organocatalysis.

scientific article

In vitro and in vivo photocytotoxicity of boron dipyrromethene derivatives for photodynamic therapy.

scientific article

In vivo studies of nanostructure-based photosensitizers for photodynamic cancer therapy

scientific article

Interplay Of Stereochemistry, Conformational Rigidity, And Ease Of Synthesis For 13-Membered Cyclic Peptidomimetics Containing APC Residues.

scientific article published on 31 May 2017

Intracellular imaging of organelles with new water-soluble benzophenoxazine dyes.

scientific article published on 3 March 2010

Iridium-mediated asymmetric hydrogenation of 2,3-diphenylbutadiene: a revealing kinetic study.

scientific article published in November 2003

Lipid diffusion from single molecules of a labeled protein undergoing dynamic association with giant unilamellar vesicles and supported bilayers.

scientific article published on 9 January 2008

Long-lasting rescue of age-associated deficits in cognition and the CNS cholinergic phenotype by a partial agonist peptidomimetic ligand of TrkA.

scientific article

Manganese-catalyzed epoxidations of alkenes in bicarbonate solutions.

scientific article published in October 2002

Mechanistic insights into iridium-catalyzed asymmetric hydrogenation of dienes.

scientific article

Metal-catalyzed epoxidations of alkenes with hydrogen peroxide

scientific article published on 01 July 2003

Microwave-assisted syntheses of regioisomerically pure bromorhodamine derivatives

scientific article published on 01 October 2003

Minimalist and universal peptidomimetics.

scientific article

Molecular basis of neurotrophin-receptor interactions.

scientific article published on December 2003

Near-infrared aza-BODIPY fluorescent probe for selective Cu2+ detection and its potential in living cell imaging

scientific article

New templates for syntheses of ring-fused, C(10) beta-turn peptidomimetics leading to the first reported small-molecule mimic of neurotrophin-3.

scientific article

New, optically active phosphine oxazoline (JM-Phos) ligands: syntheses and applications in allylation reactions.

scientific article

Nicotine abstinence syndrome precipitated by an analog of neuropeptide FF

scientific article published on 01 July 1996

Non-covalent delivery of proteins into mammalian cells

scientific article published on 30 October 2008

Novel Small Molecule Probes for Metastatic Melanoma.

scientific article

Oligoethylene glycol-substituted aza-BODIPY dyes as red emitting ER-probes

scientific article published in July 2015

Oligonucleotides with strongly fluorescent groups pi-conjugated to a nucleobase: syntheses, melting temperatures, and conformation

scientific article published on 01 August 2003

Omegatides: constrained analogs of peptide primary sequence

scientific article published on 19 December 2011

On the Mechanisms of Uptake of Tumor-Seeking Cyanine Dyes

scientific article published on 24 October 2018

On the stability of furanopyrimidin-2-one bases in oligonucleotides

scientific article published on 07 May 2004

Organelle-selective energy transfer: a fluorescent indicator of intracellular environment

scientific article

Oxidative induction of beta-turn conformations in cyclic peptidomimetics: conformational analyses as indicators of configuration.

scientific article published in August 2002

PROTAC Compatibilities, Degrading Cell-Surface Receptors, and the Sticky Problem of Finding a Molecular Glue

scientific article published on 28 October 2020

PROTACs suppression of CDK4/6, crucial kinases for cell cycle regulation in cancer

scientific article published on 01 February 2019

Peptidomimetics via copper-catalyzed azide-alkyne cycloadditions.

scientific article published on 12 June 2007

Photophysics and stability of cyano-substituted boradiazaindacene dyes.

scientific article published on 12 May 2009

Productive Manipulation of Cyanine Dye π-Networks

scientific article published on 24 May 2019

Protein labelling and albumin binding characteristics of the near-IR Cy7 fluorophore, QuatCy

scientific article published on 18 July 2019

Protein-protein interface mimicry by an oxazoline piperidine-2,4-dione

scientific article published on 27 January 2015

Pyrrolinone-pyrrolidine oligomers as universal peptidomimetics

scientific article

QuatCy: A Heptamethine Cyanine Modification With Improved Characteristics.

scientific article published on 13 April 2019

Resin effects in solid phase S(n)Ar and S(n)2 macrocyclizations

scientific article published on 01 January 2000

Rigid, conjugated, fluoresceinated thymidine triphosphates: syntheses and polymerase mediated incorporation into DNA analogues.

scientific article published in October 2003

Ring closure to beta-turn mimics via copper-catalyzed azide/alkyne cycloadditions

scientific article published on 01 November 2005

Role of Albumin in Accumulation and Persistence of Tumor-Seeking Cyanine Dyes

scientific article published on 07 January 2020

Rosamines targeting the cancer oxidative phosphorylation pathway.

scientific article

Selective formation of homo- and heterobivalent peptidomimetics

scientific article published on 01 August 2003

Site-Specific Labeling of Proteins with Near-IR Heptamethine Cyanine Dyes

scientific article published on 07 November 2018

Small Molecule Inhibitors Of The PCSK9•LDLR Interaction.

scientific article published on 29 January 2018

Small Molecule Ligands For Active Targeting Of TrkC-expressing Tumor Cells

scientific article published on 9 October 2012

Small Molecule Probes That Perturb A Protein-protein Interface In Antithrombin

scientific article

Small Molecules for Active Targeting in Cancer

scientific article published on 15 March 2016

Solid-phase SN2 macrocyclization reactions to form beta-turn mimics.

scientific article

Solid-phase syntheses of beta-turn analogues to mimic or disrupt protein-protein interactions.

scientific article

Solution- and solid-phase syntheses of substituted guanidinocarboxylic acids.

scientific article

Spectral dispersion and water solubilization of BODIPY dyes via palladium-catalyzed C-H functionalization

scientific article published on 25 April 2007

Stereoselective hydrogenations of aryl-substituted dienes

scientific article published on 06 January 2005

Subcutaneous injection of an analog of neuropeptide FF precipitates morphine abstinence syndrome

scientific article published on 01 January 1993

Syntheses and properties of water-soluble Nile Red derivatives.

scientific article published in September 2006

Syntheses of highly fluorescent GFP-chromophore analogues.

scientific article published on 6 March 2008

Syntheses of regioisomerically pure 5- or 6-halogenated fluoresceins.

scientific article published in October 2003

Syntheses, photophysical properties, and application of through-bond energy-transfer cassettes for biotechnology

scientific article published on 01 October 2006

Synthesis and solution conformation of cyclo[RGDRGD]: a cyclic peptide with selectivity for the alpha V beta 3 receptor

scientific article published on 01 October 1996

Synthesis and spectroscopic properties of rosamines with cyclic amine substituents

scientific article published on 18 October 2008

Synthesis of a new water-soluble rhodamine derivative and application to protein labeling and intracellular imaging

scientific article published on 01 September 2006

Synthesis of fluorescent, photolabile 3'-O-protected nucleoside triphosphates for the base addition sequencing scheme

scientific article published on 01 February 1999

Targeted Maytansinoid Conjugate Improves Therapeutic Index for Metastatic Breast Cancer Cells

scientific article published on 13 August 2018

Targeted PDT agent eradicates TrkC expressing tumors via photodynamic therapy (PDT)

scientific article

Termination of DNA synthesis by novel 3'-modified-deoxyribonucleoside 5'-triphosphates.

scientific article published on October 1994

Test of the potential of a dATP surrogate for sequencing via MALDI-MS.

scientific article published in December 1997

Total Syntheses of Vancomycin

scientific article published on 01 March 1999

TrkC-Targeted Kinase Inhibitors And PROTACs

scientific article published on 12 September 2019

Tropomyosin Receptor Kinase C Targeted Delivery of a Peptidomimetic Ligand-Photosensitizer Conjugate Induces Antitumor Immune Responses Following Photodynamic Therapy

scientific article published on 17 November 2016

Universal peptidomimetics.

scientific article

Water-soluble through-bond energy transfer cassettes for intracellular imaging

scientific article published on 01 August 2006

List of works by Kevin Burgess

3- and 5-Functionalized BODIPYs via the Liebeskind-Srogl reaction.

4,4-Difluoro-4-bora-3a,4a-diaza-s-indacene (BODIPY) dyes modified for extended conjugation and restricted bond rotations

A Linker Scaffold to Present Dimers of Pharmacophores Prepared by Solid-Phase Syntheses

A Near-IR Fluorescent Dasatinib Derivative That Localizes in Cancer Cells

A Near-Infrared Fluorescence Chemosensor Based on Isothiocyanate-Aza-BODIPY for Cyanide Detection at the Parts per Billion Level: Applications in Buffer Media and Living Cell Imaging

A blue-to-red energy-transfer thymidine analogue that functions in DNA.

A cheap, catalytic, scalable, and environmentally benign method for alkene epoxidations.

A chemoselective route to β-enamino esters and thioesters

A combinatorial approach for targeted delivery using small molecules and reversible masking to bypass nonspecific uptake in vivo

A combinatorial method for solution-phase synthesis of labeled bivalent beta-turn mimics.

A comparison between oxazoline-imidazolinylidene, -imidazolylidine, -benzimidazolylidene hydrogenation catalysts.

A diversity oriented synthesis of 3'-O-modified nucleoside triphosphates for DNA 'sequencing by synthesis'

A labeled guanidine ligand for studying sweet taste

A peptidomimetic of NT-3 acts as a TrkC antagonist

A zwitterionic near-infrared dye linked TrkC targeting agent for imaging metastatic breast cancer

Aldol-type chirons from asymmetric hydrogenations of trisubstituted alkenes.

Alpha,omega-functionalized 2,4-dimethylpentane dyads and 2,4,6-trimethylheptane triads through asymmetric hydrogenation.

An agent for optical imaging of TrkC-expressing, breast cancer

An asymmetric hydrogenation route to (-)-spongidepsin

An iterative route to "decorated" ethylene glycol-based linkers

Anthranilic acid-containing cyclic tetrapeptides: at the crossroads of conformational rigidity and synthetic accessibility

Asymmetric hydrogenation approaches to valuable, acyclic 1,3-hydroxymethyl chirons

Asymmetric hydrogenation routes to deoxypolyketide chirons

Asymmetric syntheses of α-methyl γ-amino acid derivatives

Aza-BODIPY dyes with enhanced hydrophilicity

BODIPY dyes and their derivatives: syntheses and spectroscopic properties.

BODIPY dyes in photodynamic therapy.

Base dependence in copper-catalyzed Huisgen reactions: efficient formation of bistriazoles

Blocking Coronavirus 19 Infection via the SARS-CoV-2 Spike Protein: Initial Steps

Catalytic homogeneous asymmetric hydrogenations of largely unfunctionalized alkenes.

Chiral imidazolylidine ligands for asymmetric hydrogenation of aryl alkenes

Chitosan-Coated Poly(lactic-co-glycolic acid)-Diiodinated boron-Dipyrromethene Nanoparticles Improve Tumor Selectivity and Stealth Properties in Photodynamic Cancer Therapy

Click-Addressable Cassette for Photoaffinity Labeling.

Combinatorial assembly of small molecules into bivalent antagonists of TrkC or TrkA receptors

Combinatorial technologies involving reiterative division/coupling/recombination: statistical considerations.

Comparison Of Asymmetric Hydrogenations Of Unsaturated- Carboxylic Acids And -Esters.

Comparisons of the conformational biases imposed by trans-2,3-methanomethionine and alpha-methylmethionine

Conjugation of Dasatinib with MHI-148 Has a Significant Advantageous Effect in Viability Assays for Glioblastoma Cells

Correction to A Near-IR Fluorescent Dasatinib Derivative That Localizes in Cancer Cells

Correlations between secondary structure- and protein-protein interface-mimicry: the interface mimicry hypothesis

Cyanine-Gemcitabine Conjugates as Targeted Theranostic Agents for Glioblastoma Tumor Cells

Cyclic semipeptoids: peptoid-organic hybrid macrocycles

Design criteria for minimalist mimics of protein-protein interface segments

DiSSiMiL: Diverse Small Size Mini-Libraries applied to simple and rapid epitope mapping of a monoclonal antibody.

Double-targeting using a TrkC ligand conjugated to dipyrrometheneboron difluoride (BODIPY) based photodynamic therapy (PDT) agent.

Electronic effects steer the mechanism of asymmetric hydrogenations of unfunctionalized aryl-substituted alkenes.

Elimination of residual natural nucleotides from 3'-O-modified-dNTP syntheses by enzymatic mop-up

Enantioselective hydrogenations of arylalkenes mediated by [Ir(cod) (JM-Phos) ]+ complexes.

Energy transfer cassettes in silica nanoparticles target intracellular organelles.

Energy transfer dyads based on Nile Red.

Enhanced antiopiate activity and enzyme resistance in a peptidomimetic of FMRFamide containing E-2,3-methanomethionine and E-2,3-methanophenylalanine

Enhanced antiopiate activity in peptidomimetics of FMRFamide containing Z-2,3-methanomethionine

Evaluating minimalist mimics by exploring key orientations on secondary structures (EKOS)

Expanding the scope of oligo-pyrrolinone-pyrrolidines as protein-protein interface mimics.

Extended piperidine-piperidinone protein interface mimics

Facile macrocyclizations to beta-turn mimics with diverse structural, physical, and conformational properties.

Filling gaps in asymmetric hydrogenation methods for acyclic stereocontrol: application to chirons for polyketide-derived natural products

Fluorescent amino- and thiopyronin dyes

Fluorescent indicators for intracellular pH.

Functionalization of the 4,4-difluoro-4-bora-3a,4a-diaza-s-indacene (BODIPY) core

Heterogeneous Phase Transfer Catalysis in Solid Phase Syntheses of Anth-Cyclic Tetrapeptides

Heterovalent selectivity and the combinatorial advantage.

Homo-Roche ester derivatives by asymmetric hydrogenation and organocatalysis.

In vitro and in vivo photocytotoxicity of boron dipyrromethene derivatives for photodynamic therapy.

In vivo studies of nanostructure-based photosensitizers for photodynamic cancer therapy

Interplay Of Stereochemistry, Conformational Rigidity, And Ease Of Synthesis For 13-Membered Cyclic Peptidomimetics Containing APC Residues.

Intracellular imaging of organelles with new water-soluble benzophenoxazine dyes.

Iridium-mediated asymmetric hydrogenation of 2,3-diphenylbutadiene: a revealing kinetic study.

Lipid diffusion from single molecules of a labeled protein undergoing dynamic association with giant unilamellar vesicles and supported bilayers.

Long-lasting rescue of age-associated deficits in cognition and the CNS cholinergic phenotype by a partial agonist peptidomimetic ligand of TrkA.

Manganese-catalyzed epoxidations of alkenes in bicarbonate solutions.

Mechanistic insights into iridium-catalyzed asymmetric hydrogenation of dienes.

Metal-catalyzed epoxidations of alkenes with hydrogen peroxide

Microwave-assisted syntheses of regioisomerically pure bromorhodamine derivatives

Minimalist and universal peptidomimetics.

Molecular basis of neurotrophin-receptor interactions.

Near-infrared aza-BODIPY fluorescent probe for selective Cu2+ detection and its potential in living cell imaging

New templates for syntheses of ring-fused, C(10) beta-turn peptidomimetics leading to the first reported small-molecule mimic of neurotrophin-3.

New, optically active phosphine oxazoline (JM-Phos) ligands: syntheses and applications in allylation reactions.