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List of works by Lorena A Kallal

A High-Content Imaging Screen for Cellular Regulators of β-Catenin Protein Abundance

scientific article published on 9 December 2015

A High-Throughput Dose-Response Cellular Thermal Shift Assay for Rapid Screening of Drug Target Engagement in Living Cells, Exemplified Using SMYD3 and IDO1

scientific article published on 28 September 2017

A novel approach applying a chemical biology strategy in phenotypic screening reveals pathway-selective regulators of histone 3 K27 tri-methylation

scientific article

An orally active TRPV4 channel blocker prevents and resolves pulmonary edema induced by heart failure

scientific article

Benzofuran-substituted urea derivatives as novel P2Y(1) receptor antagonists

scientific article published on 9 June 2010

Development of a high-throughput cell-based assay for superoxide production in HL-60 cells

scientific article published on 12 March 2010

Development of a yeast bioassay to characterize G protein-coupled receptor kinases. Identification of an NH2-terminal region essential for receptor phosphorylation

scientific article published on 24 September 2003

Development of phenotypic screening assays for γ-globin induction using primary human bone marrow day 7 erythroid progenitor cells

scientific article published on 25 October 2013

Discovery of novel and long acting muscarinic acetylcholine receptor antagonists

scientific article

Evidence for allosteric interactions of antagonist binding to the smoothened receptor

scientific article

Fluorescence microscopy techniques for the study of G protein-coupled receptor trafficking

scientific article published on 01 January 2002

High-Throughput Cellular Thermal Shift Assays in Research and Drug Discovery

scientific article published on 30 September 2019

Identification of benzimidazole diamides as selective inhibitors of the nucleotide-binding oligomerization domain 2 (NOD2) signaling pathway

scientific article (publication date: 2013)

Identification of selective small molecule inhibitors of the nucleotide-binding oligomerization domain 1 (NOD1) signaling pathway

scientific article

Identification via a Parallel Hit Progression Strategy of Improved Small Molecule Inhibitors of the Malaria Purine Uptake Transporter that Inhibit Plasmodium falciparum Parasite Proliferation

scientific article published on 14 August 2019

M3 muscarinic acetylcholine receptor antagonists: SAR and optimization of bi-aryl amines

scientific article published on 4 February 2009

Next-Generation Compound Delivery Platforms to Support Miniaturized Biology

scientific article published on 06 February 2019

Tetrahydro-4-quinolinamines identified as novel P2Y(1) receptor antagonists

scientific article published on 2 October 2008

The development of a high-content screening binding assay for the smoothened receptor.

scientific article published on 29 May 2012