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List of works by Andrew B Tobin

6-Phenylpyrimidin-4-ones as Positive Allosteric Modulators at the M1 mAChR: The Determinants of Allosteric Activity

scientific article published on 28 December 2018

Artemisinin-resistant K13 mutations rewire Plasmodium falciparum's intra-erythrocytic metabolic program to enhance survival

scientific article published on 22 January 2021

Assessment of the molecular mechanisms of action of novel 4-phenylpyridine-2-one and 6-phenylpyrimidin-4-one allosteric modulators at the M1 muscarinic acetylcholine receptors

scientific article published on 24 April 2018

Author Correction: Combinatorial expression of GPCR isoforms affects signalling and drug responses

scientific article published on 25 November 2020

Biased M1-muscarinic-receptor-mutant mice inform the design of next-generation drugs

scientific article published on 20 February 2020

Bitopic Binding Mode of an M1 Muscarinic Acetylcholine Receptor Agonist Associated with Adverse Clinical Trial Outcomes.

scientific article published on 25 April 2018

Chemogenetics defines receptor-mediated functions of short chain free fatty acids

scientific article published on 15 April 2019

Combinatorial expression of GPCR isoforms affects signalling and drug responses

scientific article published on 04 November 2020

Crystal structure of the M5 muscarinic acetylcholine receptor

scientific article published on 26 November 2019

Development of Potent PfCLK3 Inhibitors Based on TCMDC-135051 as a New Class of Antimalarials

scientific article published on 11 August 2020

M1 muscarinic allosteric modulators slow prion neurodegeneration and restore memory loss

scientific article

Pathophysiological regulation of lung function by the free fatty acid receptor FFA4

scientific article published on 01 August 2020

Restoring Agonist Function at a Chemogenetically Modified M1 Muscarinic Acetylcholine Receptor

scientific article published on 16 November 2020

Stimulus bias provides evidence for conformational constraints in the structure of a G protein-coupled receptor

scientific article

Structure-Activity Relationship Studies of Tetrahydroquinolone Free Fatty Acid Receptor 3 Modulators

scientific article published on 19 March 2020

The M<sub>1</sub> muscarinic receptor is present in situ as a ligand-regulated mixture of monomers and oligomeric complexes

scientific article published on 07 June 2022

Validation of the protein kinase PfCLK3 as a multistage cross-species malarial drug target

scientific article

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