List of works - Garth Rapeport

Antifungal synergy of a topical triazole, PC945, with a systemic triazole against respiratory Aspergillus fumigatus infection

scientific article published on 01 July 2019

Current approaches to the discovery of novel inhaled medicines

scientific article published on 20 May 2018

Discovery of Narrow Spectrum Kinase Inhibitors: New Therapeutic Agents for the Treatment of COPD and Steroid-Resistant Asthma.

scientific article published on 22 January 2016

Discovery of novel benzothienoazepine derivatives as potent inhibitors of respiratory syncytial virus

scientific article published on 23 March 2017

Effects of intranasally dosed posaconazole on fungal load and biomarkers in Aspergillus fumigatus infected immunocompromised mice.

scientific article published on 11 July 2017

In Vitro and In Vivo Antifungal Profile of a Novel and Long-Acting Inhaled Azole, PC945, on Aspergillus fumigatus Infection

scientific article

In Vitro and In Vivo Efficacy of a Novel and Long Acting Fungicidal Azole, PC1244 on Aspergillus fumigatus Infection.

scientific article published on 12 February 2018

In Vivo Biomarker Analysis of the Effects of Intranasally Dosed PC945, a Novel Antifungal Triazole, on Aspergillus fumigatus Infection in Immunocompromised Mice

scientific article published on 19 June 2017

In vitro antifungal activity of a novel topical triazole PC945 against emerging yeast Candida auris

scientific article published on 01 October 2019

Late therapeutic intervention with a respiratory syncytial virus L-protein polymerase inhibitor, PC786, on respiratory syncytial virus infection in human airway epithelium.

scientific article

Nasosorption as a Minimally Invasive Sampling Procedure: Mucosal Viral Load and Inflammation in Primary RSV Bronchiolitis.

scientific article

Neuropharmacology of emesis induced by anti-cancer therapy.

scientific article published on September 1988

Pharmacokinetics and anti-emetic efficacy of BRL43694, a new selective 5HT-3 antagonist.

scientific article

Plasma protein-binding and CSF concentrations of valproic acid in man following acute oral dosing.

scientific article

Preclinical Characterization of PC786, an Inhaled Small-Molecule Respiratory Syncytial Virus L Protein Polymerase Inhibitor

scientific article published on 26 June 2017

Reduced Nasal Viral Load and IFN Responses in Infants with Respiratory Syncytial Virus Bronchiolitis and Respiratory Failure.

scientific article

Safety, tolerability and viral kinetics during SARS-CoV-2 human challenge in young adults

scientific article published on 31 March 2022

The effects of serum, lithium, ethacrynic acid, and a low external concentration of potassium on specific [3H]-ouabain binding to human lymphocytes after incubation for 3 days.

scientific article

The influence of diet upon liver function tests and serum lipids in healthy male volunteers resident in a Phase I unit.

scientific article published on February 2004

The role of antifungals in the management of patients with severe asthma

scientific article published on 06 November 2020

Variability of phenytoin protein binding in epilepsy

scientific article published on 01 April 1984

List of works by Garth Rapeport

Antifungal synergy of a topical triazole, PC945, with a systemic triazole against respiratory Aspergillus fumigatus infection

Current approaches to the discovery of novel inhaled medicines

Discovery of Narrow Spectrum Kinase Inhibitors: New Therapeutic Agents for the Treatment of COPD and Steroid-Resistant Asthma.

Discovery of novel benzothienoazepine derivatives as potent inhibitors of respiratory syncytial virus

Effects of intranasally dosed posaconazole on fungal load and biomarkers in Aspergillus fumigatus infected immunocompromised mice.

In Vitro and In Vivo Antifungal Profile of a Novel and Long-Acting Inhaled Azole, PC945, on Aspergillus fumigatus Infection

In Vitro and In Vivo Efficacy of a Novel and Long Acting Fungicidal Azole, PC1244 on Aspergillus fumigatus Infection.

In Vivo Biomarker Analysis of the Effects of Intranasally Dosed PC945, a Novel Antifungal Triazole, on Aspergillus fumigatus Infection in Immunocompromised Mice

In vitro antifungal activity of a novel topical triazole PC945 against emerging yeast Candida auris

Late therapeutic intervention with a respiratory syncytial virus L-protein polymerase inhibitor, PC786, on respiratory syncytial virus infection in human airway epithelium.

Nasosorption as a Minimally Invasive Sampling Procedure: Mucosal Viral Load and Inflammation in Primary RSV Bronchiolitis.

Neuropharmacology of emesis induced by anti-cancer therapy.

Pharmacokinetics and anti-emetic efficacy of BRL43694, a new selective 5HT-3 antagonist.

Plasma protein-binding and CSF concentrations of valproic acid in man following acute oral dosing.

Preclinical Characterization of PC786, an Inhaled Small-Molecule Respiratory Syncytial Virus L Protein Polymerase Inhibitor

Reduced Nasal Viral Load and IFN Responses in Infants with Respiratory Syncytial Virus Bronchiolitis and Respiratory Failure.

Safety, tolerability and viral kinetics during SARS-CoV-2 human challenge in young adults

The effects of serum, lithium, ethacrynic acid, and a low external concentration of potassium on specific [3H]-ouabain binding to human lymphocytes after incubation for 3 days.

The influence of diet upon liver function tests and serum lipids in healthy male volunteers resident in a Phase I unit.

The role of antifungals in the management of patients with severe asthma

Variability of phenytoin protein binding in epilepsy