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List of works by Morten P. Meldal

'One bead two compound libraries' for detecting chemical and biochemical conversions

scientific article

2’-Deoxypuromycin: Synthesis and Antiviral Evaluation

6 Properties of solid supports

scientific article published on January 1, 1997

A comparative study of the physicochemical properties of iron isomaltoside 1000 (Monofer), a new intravenous iron preparation and its clinical implications

scientific article

A general approach to the synthesis of O- and N-linked glycopeptides.

scientific article published on April 1994

A single-vector EYFP reporter gene assay for G protein-coupled receptors

scientific article published on 11 February 2015

A solid-phase approach to mouse melanocortin receptor agonists derived from a novel thioether cyclized peptidomimetic scaffold

scientific article published on September 2002

Alpha-azido acids for direct use in solid-phase peptide synthesis

scientific article published on 01 December 2000

Alpha-keto amide peptides: a synthetic strategy to resin-bound peptide isosteres for protease inhibitor screening on solid support

scientific article published in March 2004

Amino acid derived 1,4-dialkyl substituted imidazolones

scientific article published in January 2010

Analysis of organic reactions by thin layer chromatography combined with matrix-assisted laser desorption/ionization time-of-flight mass spectrometry ⬇️

scientific article published on January 1, 1998

Anthranilamide and nitrotyrosine as a donor-acceptor pair in internally quenched fluorescent substrates for endopeptidases: multicolumn peptide synthesis of enzyme substrates for subtilisin Carlsberg and pepsin

scientific article published on 01 May 1991

Attachment of cyclodextrin acids to PEGA resin and study of binding with fluorescence microscopy

scientific article published in July 2021

Attachment of oligosaccharides to peptide antigen profoundly affects binding to major histocompatibility complex class II molecules and peptide immunogenicity

scientific article published on May 1994

Azotides as Modular Peptide-Based Ligands for Asymmetric Lewis Acid Catalysis

scientific article published on 13 May 2019

C-Terminal lactamization of peptides

scientific article published on 24 December 2020

C-Terminally modified peptides via cleavage of the HMBA linker by O-, N- or S-nucleophiles.

scientific article published on 29 February 2016

Carbohydrate and peptide specificity of MHC class II-restricted T cell hybridomas raised against an O-glycosylated self peptide

scientific article published on 01 April 1997

Characterization of T cell hybridomas raised against a glycopeptide containing the tumor-associated T antigen, (betaGal (1-3) alphaGalNAc-O/Ser).

scientific article published in January 2002

Characterization of the substrate specificity of the major cysteine protease (cruzipain) from Trypanosoma cruzi using a portion-mixing combinatorial library and fluorogenic peptides.

scientific article published on April 1997

Click Chemistry Mediated Functionalization of Vertical Nanowires for Biological Applications

scientific article published on 25 November 2015

Click-Chemistry-Mediated Synthesis of Selective Melanocortin Receptor 4 Agonists.

scientific article

Combinatorial library of peptide isosters based on Diels-Alder reactions: identification of novel inhibitors against a recombinant cysteine protease from Leishmania mexicana

scientific article

Combinatorial library of peptidotriazoles: identification of [1,2,3]-triazole inhibitors against a recombinant Leishmania mexicana cysteine protease

scientific article published in May 2004

Comparative studies of adhesion peptides based on l- or d-amino acids.

scientific article published in September 2016

Complex of sialoadhesin with a glycopeptide ligand.

scientific article published in November 2004

Computational Evolution of Threonine-Rich β-Hairpin Peptides Mimicking Specificity and Affinity of Antibodies

scientific article published on 28 January 2019

Constrained glycopeptide ligands for MPRs. Limitations of unprotected phosphorylated building blocks

scientific article published on 01 January 1997

Controlled peptide solvation in portion-mixing libraries of FRET peptides: improved specificity determination for Dengue 2 virus NS2B-NS3 protease and human cathepsin S.

scientific article

Controlled reduction of acarbose: conformational analysis of acarbose and the resulting saturated products

scientific article published in December 1991

Covalent and stable CuAAC modification of silicon surfaces for control of cell adhesion

scientific article published on 03 March 2015

Cu-catalyzed azide-alkyne cycloaddition

scientific article

Design and Combinatorial Development of Shield-1 Peptide Mimetics Binding to Destabilized FKBP12

scientific article published on 23 February 2020

Differences in substrate specificities between cysteine protease CPB isoforms of Leishmania mexicana are mediated by a few amino acid changes

scientific article published on September 2004

Diffusion of reagents in macrobeads

scientific article

Dihydroquinazolinones via A3-Type Reactions of N-Carbamoyliminium Ions

scientific article published on 13 August 2020

Divergent pathway for the solid-phase conversion of aromatic acetylenes to carboxylic acids, alpha-ketocarboxylic acids, and methyl ketones

scientific article published on 28 June 2008

Diversity-Oriented Syntheses by Combining CuAAC and Stereoselective INCIC Reactions with Peptides

scientific article

Efficient solid-phase synthesis of peptide-based phosphine ligands: towards combinatorial libraries of selective transition metal catalysts

scientific article

Expression and characterization of a recombinant cysteine proteinase of Leishmania mexicana.

scientific article published on April 2000

Expression and substrate specificity of a recombinant cysteine proteinase B of Leishmania braziliensis.

scientific article

Extensive comparison of the substrate preferences of two subtilisins as determined with peptide substrates which are based on the principle of intramolecular quenching

scientific article published on 01 July 1992

Fluorescence-quenched solid phase combinatorial libraries in the characterization of cysteine protease substrate specificity

scientific article

Glycopeptide and Oligosaccharide Libraries

scientific article

Glycopeptide mimics of mammalian Man9GlcNAc2. Ligand binding to mannan-binding proteins (MBPs).

scientific article published on November 1996

Glycopeptides as oligosaccharide mimics: high affinity sialopeptide ligands for sialoadhesin from combinatorial libraries.

scientific article

Gram-scale synthesis of alpha,alpha-trehalose 6-monophosphate and alpha,alpha-trehalose 6,6'-diphosphate

scientific article published on 01 July 1994

Graphical Abstract

scientific article published on 01 October 2001

Heterologous expression of peptidyl-Lys metallopeptidase of Armillaria mellea and mutagenic analysis of the recombinant peptidase.

scientific article published on 15 November 2015

Highly efficient solid-phase oxidative cleavage of olefins by OsO4-NalO4 in the intramolecular N-acyliminium Pictet-Spengler reaction.

scientific article published in June 2005

Hydrodynamic Control of Alzheimer Aβ Fibrillation with Glucosaminic Acid Containing Click-Cyclized β-Bodies

scientific article published on 21 December 2023

Hydrolysis by cathepsin B of fluorescent peptides derived from human prorenin

scientific article published on 01 June 2000

Identification of peptides inhibitory to recombinant cysteine proteinase, CPB, of Leishmania mexicana

scientific article

Imidazolones in diastereoselective cyclization reactions and Cu(II)-catalysed cross-coupling reactions.

scientific article published in July 2009

In vivo imaging of matrix metalloproteinase 12 and matrix metalloproteinase 13 activities in the mouse model of collagen-induced arthritis

scientific article

Inhibition of cruzipain visualized in a fluorescence quenched solid-phase inhibitor library assay.D-Amino Acid Inhibitors for cruzipain, cathepsin B and cathepsin L ⬇️

scientific article published on April 1, 1998

Internally quenched fluorescent peptide substrates disclose the subsite preferences of human caspases 1, 3, 6, 7 and 8

scientific article

In vivo imaging of MMP-13 activity in the murine destabilised medial meniscus surgical model of osteoarthritis

scientific article published on 18 April 2014

Isomerization of D-glucose with glucose-isomerase. A mechanistic study

scientific article published on 01 January 1983

K88 fimbrial antigens: identification of antigenic determinants by the use of synthetic peptides.

scientific article

Kinetic Analysis of the Mechanism and Specificity of Protein-disulfide Isomerase Using Fluorescence-quenched Peptides ⬇️

scientific article published on September 25, 1998

Lectin domains of polypeptide GalNAc transferases exhibit glycopeptide binding specificity

scientific article (publication date: 16 September 2011)

MC4R Agonists: Structural Overview on Antiobesity Therapeutics

scientific article published on 22 February 2018

MHC molecules protect T cell epitopes against proteolytic destruction ⬇️

scientific article published on September 15, 1992

MUC1-derived glycopeptide libraries with improved MHC anchors are strong antigens and prime mouse T cells for proliferative responses to lysates of human breast cancer tissue

scientific article

Maintaining biological activity by using triazoles as disulfide bond mimetics

scientific article published on 29 March 2011

Mechanism and Scope of Base-Controlled Catalyst-Free N-Arylation of Amines with Unactivated Fluorobenzenes

scientific article

Mercury iodide as a catalyst in oligosaccharide synthesis.

scientific article published on January 1983

Metabolically stable cellular adhesion to inert surfaces.

scientific article published on 16 September 2011

Metallo-Organozymes with Specific Proteolytic Activity

scientific article published on 30 October 2018

Methods for the preparation of chlorophyllide a: an intermediate of the chlorophyll biosynthetic pathway

scientific article published on 23 August 2011

Microparticle matrix encoding of beads

scientific article published on 01 May 2010

Molecular recognition of a Salmonella trisaccharide epitope by monoclonal antibody Se155-4.

scientific article published on May 1994

Multiple Column Synthesis of a Library of T‐Cell Stimulating Tn‐Antigenic Glycopeptide Analogues for the Molecular Characterization of T‐Cell–Glycan Specificity ⬇️

scientific article published on July 1, 1996

Mutational replacements of the amino acid residues forming the hydrophobic S4 binding pocket of subtilisin 309 from Bacillus lentus

scientific article published on 01 September 1993

N-Terminal peptide aldehydes as electrophiles in combinatorial solid phase synthesis of novel peptide isosteres.

scientific article

N-acyliminium intermediates in solid-phase synthesis

scientific article published on January 2010

Novel Application of Peptidyl-Lys Metallopeptidase as a C-Terminal Processing Protease

scientific article published on 01 January 2016

Novel Type of Rigid C-Linked Glycosylacetylene−Phenylalanine Building Blocks for Combinatorial Synthesis of C-linked Glycopeptides

Oligosaccharide Mimetics Obtained by Novel, Rapid Screening of Carboxylic Acid Encoded Glycopeptide Libraries

article published in 1998

Optimizing delays in the MBOB, broadband HMBC, and broadband XLOC NMR pulse sequences

scientific article published on 01 June 2002

Palladium on carbon encapsulated in POEPOP(1500): a resin-supported catalyst for hydrogenation reactions

scientific article published on 01 January 2002

Peptidotriazoles on solid phase: [1,2,3]-triazoles by regiospecific copper(i)-catalyzed 1,3-dipolar cycloadditions of terminal alkynes to azides

scientific article

Physical properties of poly(ethylene glycol) (PEG)-based resins for combinatorial solid phase organic chemistry: a comparison of PEG-cross-linked and PEG-grafted resins

scientific article published on 01 March 2000

Polymer "Clicking" by CuAAC Reactions

scientific article from 2008

Processing of glycans on glycoprotein and glycopeptide antigens in antigen-presenting cells

scientific article

Radically altered T cell receptor signaling in glycopeptide-specific T cell hybridoma induced by antigen with minimal differences in the glycan group

scientific article

Ralph F. Hirschmann award address 2009: Merger of organic chemistry with peptide diversity.

scientific article published on January 2010

Rational Tuning of Fluorobenzene Probes for Cysteine-Selective Protein Modification

scientific article published on 14 April 2018

Recent advances in covalent, site-specific protein immobilization

scientific article

Reversible dimerization of acid-denatured ACBP controlled by helix A4.

scientific article published in February 2005

SPOCC-194, a new high functional group density PEG-based resin for solid-phase organic synthesis

scientific article published in September 2002

Scaffold diversity through intramolecular cascade reactions of solid-supported cyclic N-acyliminium intermediates

scientific article published on 12 November 2007

Semisynthesis of an Active Enzyme by Quantitative Click Ligation

scientific article published on 28 March 2019

Shared structural motifs in TCR of glycopeptide-recognizing T cell hybridomas

scientific article published on September 1999

Silyl protection in the solid-phase synthesis of N-linked glycopeptides. Preparation of glycosylated fluorogenic substrates for subtilisins

scientific article published on 01 November 1994

Simultaneous "one pot" expressed protein ligation and CuI-catalyzed azide/alkyne cycloaddition for protein immobilization

scientific article published on 8 September 2011

Single-bead structure elucidation. Requirements for analysis of combinatorial solid-phase libraries by Nanoprobe MAS-NMR spectroscopy

scientific article published in 2000

Small-molecule affinity ligands for protein purification: combined computational enrichment and automated in-line screening of an optically encoded library

scientific article

Solid-phase combinatorial library of norstatine-type isosters by the nitroaldol reaction

scientific article published in March 2003

Solid-phase glycosylation of peptide templates and on-bead MAS-NMR analysis: perspectives for glycopeptide libraries

scientific article

Solid-phase intramolecular N-acyliminium Pictet-Spengler reactions as crossroads to scaffold diversity

scientific article

Solid-phase library synthesis, screening, and selection of tight-binding reduced peptide bond inhibitors of a recombinant Leishmania mexicana cysteine protease B.

scientific article

Solid-phase synthesis and biological activity of a thioether analogue of conotoxin G1.

scientific article

Solid-phase synthesis of a peptide-based P,S-ligand system designed for generation of combinatorial catalyst libraries

scientific article

Solid-phase synthesis of aryl-substituted thienoindolizines: sequential Pictet-Spengler, bromination and Suzuki cross-coupling reactions of thiophenes

scientific article published on 4 April 2008

Solid-phase synthesis of bicyclic dipeptide mimetics by intramolecular cyclization of alcohols, thiols, amines, and amides with N-acyliminium intermediates

scientific article published on 01 August 2005

Solid-phase synthesis of carboxylic and oxamic acids via OsO4/NaIO4/HMTA-mediated oxidative cleavage of acetylenic peptides.

scientific article

Solid-phase synthesis of chemotactic peptides using alpha-azido acids

scientific article published on 01 July 2000

Solid-phase synthesis of complex and pharmacologically interesting heterocycles.

scientific article

Solid-phase synthesis of pyrroloisoquinolines via the intramolecular N-acyliminium Pictet-Spengler reaction

scientific article published in July 2005

Solid-phase synthesis of tetrahydro-beta-carbolines and tetrahydroisoquinolines by stereoselective intramolecular N-carbamyliminium Pictet-Spengler reactions

scientific article published on 01 October 2006

Specific Electrostatic Molecular Recognition in Water.

scientific article

Specificity of O-glycosylation by bovine colostrum UDP-GalNAc: polypeptide alpha-N-acetylgalactosaminyltransferase using synthetic glycopeptide substrates

scientific article published on 01 October 1996

Spectroscopic and protein chemical analyses demonstrate the presence of C-mannosylated tryptophan in intact human RNase 2 and its isoforms

scientific article published on 01 September 1996

Studies of binding sites in the subtilisin from Bacillus lentus by means of site directed mutagenesis and kinetic investigations

scientific article published on 01 January 1996

Substrate Specificity Profiling of Peptidyl-Lys Metallopeptidase of Armillaria mellea by FRET Based Peptide Library

scientific article published on January 2015

Substrate preferences of glutamic-acid-specific endopeptidases assessed by synthetic peptide substrates based on intramolecular fluorescence quenching

scientific article

Substrate specificity of recombinant cysteine proteinase, CPB, of Leishmania mexicana

scientific article published in August 2001

Surfactant Mediated Cationic and Anionic Suspension Polymerization of PEG-Based Resins in Silicon Oil: Beaded SPOCC 1500 and POEPOP 1500.

scientific article

Susceptibility of glycans to beta-elimination in Fmoc-based O-glycopeptide synthesis.

scientific article published on June 1994

Sustainable Flow Synthesis of Encoded Beads for Combinatorial Chemistry and Chemical Biology

scientific article published on 18 July 2018

Synthesis and application of sialic acid-containing building blocks for glycopeptide libraries. Establishing glycosylation conditions

scientific article published in 2000

Synthesis and characterisation of highly glycosylated glycopeptides with Tn-antigenic structures corresponding to human glycophorin AN

scientific article published on 01 March 1997

Synthesis of Shld Derivatives, Their Binding to the Destabilizing Domain, and Influence on Protein Accumulation in Transgenic Plants

scientific article published on 14 May 2019

Synthesis of aldehyde building blocks protected as acid labile N-Boc N,O-acetals: toward combinatorial solid phase synthesis of novel peptide isosteres

scientific article

Synthesis of the glycosyl amino acids N alpha-Fmoc-Ser[Ac4-beta-D-Galp-(1-->3)-Ac2-alpha-D-GalN3p]-OPfp and N alpha-Fmoc-Thr[Ac4-beta-D-Galp-(1-->3)-Ac2-alpha-D-GalN3p]-OPfp and the application in the solid-phase peptide synthesis of multiply glycos

scientific article published on 01 March 1995

Synthesis of tumor associated sialyl-T-glycopeptides and their immunogenicity.

scientific article

Synthesis, characterization and biocompatibility of PEGA resins ⬇️

scientific article published on January 1, 1995

Synthetic hFSH peptide constructs in the evaluation of previous studies on the hFSH receptor interaction

scientific article published on 01 November 1997

Synthetic methods of glycopeptide assembly, and biological analysis of glycopeptide products ⬇️

scientific article published on December 1, 1997

T cell recognition of Tn-glycosylated peptide antigens

scientific article published in June 1996

T-Helper-Cell Determinants in Protein Antigens are Preferentially Located in Cysteine-Rich Antigen Segments Resistant to Proteolytic Cleavage by Cathepsin B, L, and D ⬇️

scientific article published on October 1, 1991

T-cell recognition of tumor-associated carbohydrates: the nature of the glycan moiety plays a decisive role in determining glycopeptide immunogenicity ⬇️

scientific article published on 01 August 1997

The Pictet-Spengler reaction in solid-phase combinatorial chemistry.

scientific article

The T-lymphocyte proliferative response to synthetic peptide antigens of defined secondary structure

scientific article published on 01 December 1989

The active ester N-fmoc-3-O-[Ac4-α-D-Manp-(1→2)-Ac3-α-D-Manp-1-]=thre-O-Pfp as a building block in solid-phase synthesis of an o-linked dimannosyl glycopeptide

The conformation of Salmonella O-antigenic oligosaccharides of serogroups A, B, and D1 inferred from 1H- and 13C-nuclear magnetic resonance spectroscopy

scientific article published in July 1984

The conformation of Salmonella O-antigenic polysaccharide chains of serogroups A, B, and D1 predicted by semi-empirical, Hard-Sphere (HSEA) calculations

scientific article published in July 1984

The extracellular polysaccharide of Pichia (Hansenula) holstii NRRL Y-2448: the phosphorylated side chains

scientific article

The extracellular polysaccharide of Pichia (Hansenula) holstii NRRL Y-2448: the structure of the phosphomannan backbone

scientific article published on 01 October 1996

The one-bead two-compound assay for solid phase screening of combinatorial libraries

scientific article

The substrate specificity of a recombinant cysteine protease from Leishmania mexicana: application of a combinatorial peptide library approach

scientific article

UDPgalactose:glycoprotein-N-acetyl-D-galactosamine 3-beta-D-galactosyltransferase activity synthesizing O-glycan core 1 is controlled by the amino acid sequence and glycosylation of glycopeptide substrates

scientific article published on 01 May 1994

ULTRAMINE: a high-capacity polyethylene-imine-based polymer and its application as a scavenger resin

scientific article published in September 2004

Unichemo Protection: A Concept for Chemical Synthesis This work was supported by the Danish National Research Foundation

scientific article published in October 2001

Versatile solid-phase synthesis of peptide-derived 2-oxazolines. Application in the synthesis of ligands for asymmetric catalysis

scientific article published on 01 February 2005

alpha-Ketocarbonyl peptides: a general approach to reactive resin-bound intermediates in the synthesis of peptide isosteres for protease inhibitor screening on solid support

scientific article published in March 2001

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