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List of works by Jakub Staroń

-Skatyltryptamines-Dual 5-HTR/DR Ligands with Antipsychotic and Procognitive Potential

scientific article published on 29 July 2021

2-Aminoimidazole-based antagonists of the 5-HT6 receptor - A new concept in aminergic GPCR ligand design

scientific article published on 05 June 2019

5-HT1A receptor ligands and their therapeutic applications: review of new patents

scientific article published on 07 September 2018

Bioisosteric matrices for ligands of serotonin receptors

scientific article published on 13 March 2015

Encapsulation of curcumin in polyelectrolyte nanocapsules and their neuroprotective activity.

scientific article published on 25 July 2016

Factors controlling the reactivity of divalent metal ions towards pheophytin a

scientific article

Fluorinated indole-imidazole conjugates: Selective orally bioavailable 5-HT7 receptor low-basicity agonists, potential neuropathic painkillers

scientific article published on 11 March 2019

Halogen bonding enhances activity in a series of dual 5-HT6/D2 ligands designed in a hybrid bioisostere generation/virtual screening protocol

scholarly article in RSC Advances, vol. 6 no. 60, 2016

In Search of Effective Anticancer Agents-Novel Sugar Esters Based on Polyhydroxyalkanoate Monomers

scientific article published on 5 July 2021

Lactose esters: synthesis and biotechnological applications.

scientific article published on 06 June 2017

Lessons from chlorophylls: modifications of porphyrinoids towards optimized solar energy conversion

scientific article published on 03 October 2014

Low-basicity 5-HT7 Receptor Agonists Synthesized Using the van Leusen Multicomponent Protocol

scientific article

Prenatal Exposure to Benzophenone-3 Impairs Autophagy, Disrupts RXRs/PPARγ Signaling, and Alters Epigenetic and Post-Translational Statuses in Brain Neurons

scientific article published on 06 November 2018

Pyrano[2,3,4-cd]indole as a Scaffold for Selective Nonbasic 5-HT6R Ligands

scientific article

Rational design of 5-HT 6 R ligands using a bioisosteric strategy: synthesis, biological evaluation and molecular modelling

scientific article published in 2015

Rationally designed N-phenylsulfonylindoles as a tool for the analysis of the non-basic 5-HT<sub>6</sub>R ligands binding mode

scientific article published on 09 October 2020

Reaction mechanism of sterol hydroxylation by steroid C25 dehydrogenase - Homology model, reactivity and isoenzymatic diversity

scientific article published on 27 April 2017

Recent Progress in Chemical Modifications of Chlorophylls and Bacteriochlorophylls for the Applications in Photodynamic Therapy

scientific article published on 17 August 2015

Regioselective hydroxylation of cholecalciferol, cholesterol and other sterol derivatives by steroid C25 dehydrogenase

scientific article

Serotonin type 5A receptor antagonists inhibit D-lysergic acid diethylamide discriminatory cue in rats

scientific article published on 27 August 2019

The effect of the intramolecular C-H⋯O interactions on the conformational preferences of bis-arylsulfones - 5-HT receptor antagonists and beyond

scientific article published on 17 May 2018

Virtual screening-driven discovery of dual 5-HT6/5-HT2A receptor ligands with pro-cognitive properties

scientific article published on 07 November 2019

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