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List of works by David Vandervelde

18Oxygen incorporation into inorganic phosphate in the reaction catalyzed by N5,10-methenyltetrahydrofolate synthetase

scientific article published on 01 May 1995

A 19F NMR study of lomefloxacin in human erythrocytes and its interaction with hemoglobin

scientific article published on 01 September 1995

A one-step synthesis of a deuterated paclitaxel analogue: 10-deacetoxy-(10alpha-2H)paclitaxel

scientific article published on 01 December 1999

A tandem Prins/Schmidt reaction approach to marine alkaloids: formal and total syntheses of lepadiformines A and C

scientific article

Alternate substrates of human glutaryl-CoA dehydrogenase: structure and reactivity of substrates, and identification of a novel 2-enoyl-CoA product.

scientific article published in January 2002

An Initial Event in the Insect Innate Immune Response: Structural and Biological Studies of Interactions between β-1,3-Glucan and the N-Terminal Domain of β-1,3-Glucan Recognition Protein

scientific article

Biofilm-specific extracellular matrix proteins of nontypeable Haemophilus influenzae

scientific article

CO Coupling Chemistry of a Terminal Mo Carbide: Sequential Addition of Proton, Hydride, and CO Releases Ethenone

scientific article published on 19 September 2019

Characterization and dynamics of substituted ruthenacyclobutanes relevant to the olefin cross-metathesis reaction

scientific article published on 31 March 2011

Characterization of the complexation of fluoroquinolone antimicrobials with metal ions by nuclear magnetic resonance spectroscopy

scientific article published on 01 January 1993

Comparative effects of (SBE)7m-beta-CD and HP-beta-CD on the stability of two anti-neoplastic agents, melphalan and carmustine

scientific article published on 01 February 2000

Comprehensive study of sansalvamide A derivatives and their structure-activity relationships against drug-resistant colon cancer cell lines.

scientific article published on 11 January 2008

Conformation of ATP and ADP bound to N10-formyltetrahydrofolate synthetase determined by TRNOE NMR spectroscopy.

scientific article published in January 1994

Conformational analysis of the beta-amyloid peptide fragment, beta(12-28)

scientific article published on 01 October 1995

Conformational studies on resiniferatoxin (RTX), an ultrapotent vanilloid agonist

scientific article published on 01 February 1998

Conformationally restricted paclitaxel analogues: macrocyclic mimics of the "hydrophobic collapse" conformation

scientific article published on 01 October 1999

Cyclodextrin-catalyzed deacetylation of spironolactone is pH and cyclodextrin dependent

scientific article published on 01 February 2000

Deamidation of model beta-turn cyclic peptides in the solid state

scientific article published on 01 December 2005

Diastereomeric phosphonate ester adducts of chymotrypsin: 31P-NMR measurements

scientific article published on 01 January 1993

Effect of buffer species on the thermally induced aggregation of interferon-tau

scientific article published on 01 June 2006

Effect of conformation on the rate of deamidation of vancomycin in aqueous solutions

scientific article published on 01 June 2000

Effect of progressive benzyl substitution on the conformations of aminocaproic acid-cyclized dipeptides.

scientific article published in April 2001

Effect of restricted conformational flexibility on the permeation of model hexapeptides across Caco-2 cell monolayers

scientific article published on 01 February 1997

Effect of stereochemistry on the transport of Aca-linked β-turn peptidomimetics across a human intestinal cell line

scientific article published on September 1, 1997

Effect of zinc binding on the structure and stability of fibrolase, a fibrinolytic protein from snake venom

scientific article published on 01 July 1992

Effects of amino acid chirality and the chemical linker on the cell permeation characteristics of cyclic prodrugs of opioid peptides.

scientific article published in February 2006

Evaluation of NMR diffusion measurements for the conformational analysis of flexible peptides.

scientific article

Experimental and theoretical investigations into the unusual regioselectivity of 4,5-, 5,6-, and 6,7-indole aryne cycloadditions

scientific article

Fibrolase. A fibrinolytic protein from snake venom.

scientific article published on January 1993

Fluoride-facilitated deuterium exchange from DMSO-d6 to polyamide-based cryptands.

scientific article published in October 2004

Get5 Carboxyl-terminal Domain Is a Novel Dimerization Motif That Tethers an Extended Get4/Get5 Complex

scientific article

Highly regioirregular polypropylene from asymmetric group 4 anilide(pyridine)phenoxide complexes.

scientific article published on 25 May 2012

Hydrocotylosides I-VII, new oleanane saponins from hydrocotylesibthorpioides.

scientific article published in March 2004

Hydrolysis of the prodrug, 2',3',5'-triacetyl-6-azauridine.

scientific article published on September 1995

Improved preparation and structural conformation of the fluorescence labelling reagents 1,2-diamino-4,5-dimethoxybenzene and 3,4-dihydro-6,7-dimethoxy-4-methyl-3-oxo-quinoxaline-2-carbonyl chloride

scientific article published on 01 January 1990

Indole-derived arynes and their Diels-Alder reactivity with furans

scientific article published on 19 September 2007

Isolation and characterization by NMR spectroscopy of three monosubstituted 4-sulfobutyl ether derivatives of cyclomaltoheptaose (beta-cyclodextrin)

scientific article published on 01 April 1997

Isolation of endogenous modulators for the GABAA and taurine receptors

scientific article published on 01 November 1993

Kinetics and products of the acid-catalyzed ring-opening of atmospherically relevant butyl epoxy alcohols.

scientific article

Lewis Acid Enhancement of Proton Induced CO2 Cleavage: Bond Weakening and Ligand Residence Time Effects

scientific article published on 01 August 2018

Lewis acid promoted titanium alkylidene formation: off-cycle intermediates relevant to olefin trimerization catalysis

scientific article published on 18 July 2014

Modulating the Folding Landscape of Superoxide Dismutase 1 with Targeted Molecular Binders.

scientific article published on 25 April 2018

New polyamide cryptand for anion binding.

scientific article published in August 2003

Nitrogen Insertion into a Corrole Ring: Iridium Monoazaporphyrins

scientific article published on August 30, 2011

Novel d-seco paclitaxel analogues: synthesis, biological evaluation, and model testing.

scientific article

Nucleoside triphosphate specificity of tubulin

scientific article published on 01 August 2000

Optimum doses of deuterium oxide and sodium bromide for the determination of total body water and extracellular fluid

scientific article published on January 1, 1991

Paclitaxel Analogues fromTaxus×mediacv. Hicksii

scientific article published on 01 February 1999

Poly(L-lysine) as a model drug macromolecule with which to investigate secondary structure and microporous membrane transport, part 2: diffusion studies

scientific article published on 01 November 2002

Preparation and physicochemical characterization of a novel water-soluble prodrug of carbamazepine.

scientific article

Protonation of crotonyl-CoA dienolate by human glutaryl-CoA dehydrogenase occurs by solvent-derived protons.

scientific article

Reactivity of Metabolic Intermediates and Cofactor Stability under Model Early Earth Conditions

scientific article published on 25 January 2020

Reactivity toward deamidation of asparagine residues in beta-turn structures.

scientific article published on September 2000

Redox and pH gradients drive amino acid synthesis in iron oxyhydroxide mineral systems

scientific article published on 25 February 2019

Regioselective Diels-Alder cycloadditions and other reactions of 4,5-, 5,6-, and 6,7-indole arynes.

scientific article

Secondary structure of a dynamic type I'beta-hairpin peptide.

scientific article published in April 2004

Site-specifically traced drug release and biodistribution of a paclitaxel-antibody conjugate toward improvement of the linker structure.

scientific article

Solution behavior of a novel type 1 interferon, interferon-tau.

scientific article published in December 2005

Stability of the thrombolytic protein fibrolase: effect of temperature and pH on activity and conformation

scientific article published on 01 September 1991

Structure-activity studies of antitumor taxanes: synthesis of novel C-13 side chain homologated taxol and taxotere analogs

scientific article published on 01 September 1994

Synthesis and conformation of Gly-Gly dipeptides constrained with phenylalanine-like aminocaproic acid linkers

scientific article published on 01 June 2000

Synthesis and conformational analysis of a coumarinic acid-based cyclic prodrug of an opioid peptide with modified sensitivity to esterase-catalyzed bioconversion.

scientific article published in April 2002

The dormancy-specific regulator, SutA, is intrinsically disordered and modulates transcription initiation in Pseudomonas aeruginosa

scientific article published on 10 July 2019

The effect of beta-turn structure on the passive diffusion of peptides across Caco-2 cell monolayers

scientific article published on 01 October 1997

The effect of conformation on membrane permeability of an acyloxyalkoxy-linked cyclic prodrug of a model hexapeptide

scientific article published on 01 November 1996

The effect of conformation on the membrane permeation of coumarinic acid- and phenylpropionic acid-based cyclic prodrugs of opioid peptides.

scientific article published in April 1999

The effect of the aromatic rings of taxol on biological activity and solution conformation: synthesis and evaluation of saturated taxol and taxotere analogues

scientific article published on 01 September 1994

The oxetane conformational lock of paclitaxel: structural analysis of D-secopaclitaxel.

scientific article

Total Synthesis and Characterization of 7-Hypoquinuclidonium Tetrafluoroborate and 7-Hypoquinuclidone BF3 Complex

scientific article (publication date: 27 January 2016)

Total synthesis and evaluation of C25-benzyloxyepothilone C for tubulin assembly and cytotoxicity against MCF-7 breast cancer cells.

scientific article

Total synthesis and evaluation of C26-hydroxyepothilone D derivatives for photoaffinity labeling of beta-tubulin.

scientific article

Transport characteristics of peptides and peptidomimetics: II. Hydroxyethylamine bioisostere-containing peptidomimetics as substrates for the oligopeptide transporter and P-glycoprotein in the intestinal mucosa.

scientific article

Two-, three-, and four-dimensional nuclear magnetic resonance spectroscopy of protein pharmaceuticals.

scientific article published on January 1995