List of works - Richard Neubig

International Union of Pharmacology. XLVI. G protein-coupled receptor list.

scientific article

Regulators of G-protein signalling as new central nervous system drug targets.

scientific article

International Union of Pharmacology Committee on Receptor Nomenclature and Drug Classification. XXXVIII. Update on terms and symbols in quantitative pharmacology

scientific article (publication date: December 2003)

Phagocyte-derived catecholamines enhance acute inflammatory injury

scientific article published in Nature

Membrane organization in G-protein mechanisms.

scientific article published on September 1994

The highly conserved DRY motif of class A G protein-coupled receptors: beyond the ground state.

scientific article published on 27 December 2006

The Concise Guide to PHARMACOLOGY 2013/14: overview

scientific article

Acetylcholine and local anesthetic binding to Torpedo nicotinic postsynaptic membranes after removal of nonreceptor peptides

scientific article published on February 1, 1979

International Union of Basic and Clinical Pharmacology. LXVII. Recommendations for the recognition and nomenclature of G protein-coupled receptor heteromultimers.

scientific article published on March 2007

Structure of Galphaq-p63RhoGEF-RhoA complex reveals a pathway for the activation of RhoA by GPCRs

scientific article

IUPHAR-DB: the IUPHAR database of G protein-coupled receptors and ion channels

scientific article

CCG-1423: a small-molecule inhibitor of RhoA transcriptional signaling.

scientific article published on August 2007

International Union of Basic and Clinical Pharmacology. LXXXVIII. G protein-coupled receptor list: recommendations for new pairings with cognate ligands

scientific article

A point mutation in Galphao and Galphai1 blocks interaction with regulator of G protein signaling proteins

scientific article published on 01 May 1998

Equilibrium binding of [3H]tubocurarine and [3H]acetylcholine by torpedo postsynaptic membranes: stoichiometry and ligand interactions

scientific article published on November 27, 1979

International Union of Pharmacology. LVI. Ghrelin receptor nomenclature, distribution, and function

scientific article

Identification of small-molecule inhibitors of RGS4 using a high-throughput flow cytometry protein interaction assay

scientific article

A spatial focusing model for G protein signals. Regulator of G protein signaling (RGS) protien-mediated kinetic scaffolding.

scientific article

Small molecule protein-protein interaction inhibitors as CNS therapeutic agents: current progress and future hurdles.

scientific article published on 17 September 2008

Novel Rho/MRTF/SRF inhibitors block matrix-stiffness and TGF-β-induced fibrogenesis in human colonic myofibroblasts

scientific article published on January 2014

Redox modification of nuclear actin by MICAL-2 regulates SRF signaling

scientific article

Inhibition of myocardin-related transcription factor/serum response factor signaling decreases lung fibrosis and promotes mesenchymal cell apoptosis.

scientific article

N-terminal residues control proteasomal degradation of RGS2, RGS4, and RGS5 in human embryonic kidney 293 cells

scientific article

AT1 receptor mutant lacking heterotrimeric G protein coupling activates the Src-Ras-ERK pathway without nuclear translocation of ERKs.

scientific article published on 3 January 2002

M4 Muscarinic Receptor Signaling Ameliorates Striatal Plasticity Deficits in Models of L-DOPA-Induced Dyskinesia

scientific article published on November 2015

Receptor-selective effects of endogenous RGS3 and RGS5 to regulate mitogen-activated protein kinase activation in rat vascular smooth muscle cells

scientific journal article

International Union of Basic and Clinical Pharmacology. XC. multisite pharmacology: recommendations for the nomenclature of receptor allosterism and allosteric ligands.

scientific article

Targeting the myofibroblast genetic switch: inhibitors of myocardin-related transcription factor/serum response factor-regulated gene transcription prevent fibrosis in a murine model of skin injury

scientific article

Immunofluorescence localization at the mammalian neuromuscular junction of the Mr 43,000 protein of Torpedo postsynaptic membranes.

scientific article

Endogenous RGS proteins and Galpha subtypes differentially control muscarinic and adenosine-mediated chronotropic effects.

scientific article published on 2 February 2006

Endogenous RGS protein action modulates mu-opioid signaling through Galphao. Effects on adenylyl cyclase, extracellular signal-regulated kinases, and intracellular calcium pathways

scientific article published on 10 January 2003

Regulators of G protein signaling & drugs of abuse.

scientific article

A juxtamembrane mutation in the N terminus of the dopamine transporter induces preference for an inward-facing conformation.

scientific article

Regulators of G protein signaling proteins as targets for drug discovery.

scientific article published on January 2010

Permeability control by cholinergic receptors in Torpedo postsynaptic membranes: agonist dose-response relations measured at second and millisecond times

scientific article published on 01 June 1980

Pleiotropic phenotype of a genomic knock-in of an RGS-insensitive G184S Gnai2 allele

scientific article

Conformations of Torpedo acetylcholine receptor associated with ion transport and desensitization

scientific article published on 01 July 1982

Reversible, allosteric small-molecule inhibitors of regulator of G protein signaling proteins

scientific article

Thrombin and lysophosphatidic acid receptors utilize distinct rhoGEFs in prostate cancer cells

scientific article

Rapid kinetics of regulator of G-protein signaling (RGS)-mediated Galphai and Galphao deactivation. Galpha specificity of RGS4 AND RGS7

scientific article published on 01 October 2000

Thinking outside of the "RGS box": new approaches to therapeutic targeting of regulators of G protein signaling.

scientific article

A nanomolar-potency small molecule inhibitor of regulator of G-protein signaling proteins

scientific article

Inverse agonist activity of agouti and agouti-related protein.

scientific article

Design, synthesis and prostate cancer cell-based studies of analogs of the Rho/MKL1 transcriptional pathway inhibitor, CCG-1423.

scientific article

Stimulation of cellular signaling and G protein subunit dissociation by G protein betagamma subunit-binding peptides.

scientific article published on 20 March 2003

Walker A lysine mutations of TAP1 and TAP2 interfere with peptide translocation but not peptide binding.

scientific article

RGS inhibition at G(alpha)i2 selectively potentiates 5-HT1A-mediated antidepressant effects.

scientific article

Guanine nucleotide effects on catecholamine secretion from digitonin-permeabilized adrenal chromaffin cells

scientific article published on 01 August 1986

RGS/Gi2alpha interactions modulate platelet accumulation and thrombus formation at sites of vascular injury

scientific article

Assembly of high order G alpha q-effector complexes with RGS proteins

scientific article published on 20 October 2008

List of works by Richard Neubig

International Union of Pharmacology. XLVI. G protein-coupled receptor list.

Regulators of G-protein signalling as new central nervous system drug targets.

International Union of Pharmacology Committee on Receptor Nomenclature and Drug Classification. XXXVIII. Update on terms and symbols in quantitative pharmacology

Phagocyte-derived catecholamines enhance acute inflammatory injury

Membrane organization in G-protein mechanisms.

The highly conserved DRY motif of class A G protein-coupled receptors: beyond the ground state.

The Concise Guide to PHARMACOLOGY 2013/14: overview

Acetylcholine and local anesthetic binding to Torpedo nicotinic postsynaptic membranes after removal of nonreceptor peptides

International Union of Basic and Clinical Pharmacology. LXVII. Recommendations for the recognition and nomenclature of G protein-coupled receptor heteromultimers.

Structure of Galphaq-p63RhoGEF-RhoA complex reveals a pathway for the activation of RhoA by GPCRs

IUPHAR-DB: the IUPHAR database of G protein-coupled receptors and ion channels

CCG-1423: a small-molecule inhibitor of RhoA transcriptional signaling.

International Union of Basic and Clinical Pharmacology. LXXXVIII. G protein-coupled receptor list: recommendations for new pairings with cognate ligands

A point mutation in Galphao and Galphai1 blocks interaction with regulator of G protein signaling proteins

Equilibrium binding of [3H]tubocurarine and [3H]acetylcholine by torpedo postsynaptic membranes: stoichiometry and ligand interactions

International Union of Pharmacology. LVI. Ghrelin receptor nomenclature, distribution, and function

Identification of small-molecule inhibitors of RGS4 using a high-throughput flow cytometry protein interaction assay

A spatial focusing model for G protein signals. Regulator of G protein signaling (RGS) protien-mediated kinetic scaffolding.

Small molecule protein-protein interaction inhibitors as CNS therapeutic agents: current progress and future hurdles.

Novel Rho/MRTF/SRF inhibitors block matrix-stiffness and TGF-β-induced fibrogenesis in human colonic myofibroblasts

Redox modification of nuclear actin by MICAL-2 regulates SRF signaling

Inhibition of myocardin-related transcription factor/serum response factor signaling decreases lung fibrosis and promotes mesenchymal cell apoptosis.

N-terminal residues control proteasomal degradation of RGS2, RGS4, and RGS5 in human embryonic kidney 293 cells

AT1 receptor mutant lacking heterotrimeric G protein coupling activates the Src-Ras-ERK pathway without nuclear translocation of ERKs.

M4 Muscarinic Receptor Signaling Ameliorates Striatal Plasticity Deficits in Models of L-DOPA-Induced Dyskinesia

Receptor-selective effects of endogenous RGS3 and RGS5 to regulate mitogen-activated protein kinase activation in rat vascular smooth muscle cells

International Union of Basic and Clinical Pharmacology. XC. multisite pharmacology: recommendations for the nomenclature of receptor allosterism and allosteric ligands.

Targeting the myofibroblast genetic switch: inhibitors of myocardin-related transcription factor/serum response factor-regulated gene transcription prevent fibrosis in a murine model of skin injury

Immunofluorescence localization at the mammalian neuromuscular junction of the Mr 43,000 protein of Torpedo postsynaptic membranes.

Endogenous RGS proteins and Galpha subtypes differentially control muscarinic and adenosine-mediated chronotropic effects.

Endogenous RGS protein action modulates mu-opioid signaling through Galphao. Effects on adenylyl cyclase, extracellular signal-regulated kinases, and intracellular calcium pathways

Regulators of G protein signaling & drugs of abuse.

A juxtamembrane mutation in the N terminus of the dopamine transporter induces preference for an inward-facing conformation.

Regulators of G protein signaling proteins as targets for drug discovery.

Permeability control by cholinergic receptors in Torpedo postsynaptic membranes: agonist dose-response relations measured at second and millisecond times

Pleiotropic phenotype of a genomic knock-in of an RGS-insensitive G184S Gnai2 allele

Conformations of Torpedo acetylcholine receptor associated with ion transport and desensitization

Reversible, allosteric small-molecule inhibitors of regulator of G protein signaling proteins

Thrombin and lysophosphatidic acid receptors utilize distinct rhoGEFs in prostate cancer cells

Rapid kinetics of regulator of G-protein signaling (RGS)-mediated Galphai and Galphao deactivation. Galpha specificity of RGS4 AND RGS7

Thinking outside of the "RGS box": new approaches to therapeutic targeting of regulators of G protein signaling.

A nanomolar-potency small molecule inhibitor of regulator of G-protein signaling proteins

Inverse agonist activity of agouti and agouti-related protein.

Design, synthesis and prostate cancer cell-based studies of analogs of the Rho/MKL1 transcriptional pathway inhibitor, CCG-1423.

Stimulation of cellular signaling and G protein subunit dissociation by G protein betagamma subunit-binding peptides.

Walker A lysine mutations of TAP1 and TAP2 interfere with peptide translocation but not peptide binding.

RGS inhibition at G(alpha)i2 selectively potentiates 5-HT1A-mediated antidepressant effects.

Guanine nucleotide effects on catecholamine secretion from digitonin-permeabilized adrenal chromaffin cells

RGS/Gi2alpha interactions modulate platelet accumulation and thrombus formation at sites of vascular injury

Assembly of high order G alpha q-effector complexes with RGS proteins