List of works - Hartmut H. Glossmann

(?)-3H-desmethoxyverapamil labelling of putative calcium channels in brain: autoradiographic distribution and allosteric coupling to 1,4-dihydropyridine and diltiazem binding sites ⬇️

scientific article published on September 1, 1984

125I-iodipine, a new high affinity ligand for the putative calcium channel.

scientific article

7-Dehydrocholesterol-dependent proteolysis of HMG-CoA reductase suppresses sterol biosynthesis in a mouse model of Smith-Lemli-Opitz/RSH syndrome

scientific article

?-Adrenergic receptors in guinea-pig myocardial tissue ⬇️

scientific article published on December 1, 1976

A marriage of two "Methusalem" drugs for the treatment of psoriasis?: Arguments for a pilot trial with metformin as add-on for methotrexate.

scientific article published on April 2013

A novel 1,4-dihydropyridine-binding site on mitochondrial membranes from guinea-pig heart, liver and kidney.

scientific article published on July 1988

A rapid procedure for the purification of cardiac 1,4-dihydropyridine receptors from porcine heart

scientific article published on 01 May 1991

Adrenal cortex adenylate cyclase. Specific binding sites for 5'-guanylyl-imidodiphosphate in partially purified plasma membranes from bovine adrenal cortex

scientific article published on 01 January 1975

Alpha 2 adrenoceptors in rat brain: the divalent cation site

scientific article published on 01 November 1980

Alpha adrenoceptors in rat brain: Direct identification with prazosin ⬇️

scientific article published on September 1, 1979

Analysis of membrane protein self-association in lipid systems by fluorescence particle counting: application to the dihydropyridine receptor

scientific article published on 01 April 1997

Association of calcium channel α 1S and β 1a subunits is required for the targeting of β 1a but not of α 1S into skeletal muscle triads ⬇️

scientific article published on April 28, 1998

Association of the src-gene product of Rous sarcoma virus with a pyruvate-kinase inactivation factor.

scientific article published in July 1981

Benzothiazepine binding domain of purified L-type calcium channels: direct labeling using a novel fluorescent diltiazem analogue.

scientific article published on March 1995

Bovine adrenal cortex adenylate cyclase: Properties of the particulate enzyme and effects of guanyl nucleotides ⬇️

scientific article published on January 1, 1975

Calcium channels from Cyprinus carpio skeletal muscle.

scientific article published on February 1991

Calcium channels: the beta-subunit increases the affinity of dihydropyridine and Ca2+ binding sites of the alpha 1-subunit.

scientific article published on September 1994

Calcium- and potassium-channel blockers interact with alpha-adrenoceptors.

scientific article published in September 1980

Cation sensitivity of [125I]heat binding to alpha 1-adrenoceptors in rat cerebral cortex membranes

scientific article published on 01 October 1981

Commentary: Lactate-Induced Glucose Output Is Unchanged by Metformin at a Therapeutic Concentration-A Mass Spectrometry Imaging Study of the Perfused Rat Liver

scientific article published on 19 February 2019

Complex molecular mechanism for dihydropyridine binding to L-type Ca(2+)-channels as revealed by fluorescence resonance energy transfer

scientific article published on 01 October 1994

Conserved Ca2+-antagonist-binding properties and putative folding structure of a recombinant high-affinity dihydropyridine-binding domain.

scientific article

Coordination of Ca2+ by the pore region glutamates is essential for high-affinity dihydropyridine binding to the cardiac Ca2+ channel alpha 1 subunit.

scientific article

Correlation between the negative inotropic potency and binding parameters of 1,4-dihydropyridine and phenylalkylamine calcium channel blockers in cat heart

scientific article published on 01 November 1986

Differential effects of Ca2+ channel beta1a and beta2a subunits on complex formation with alpha1S and on current expression in tsA201 cells.

scientific article published on April 1998

Differential labelling of putative skeletal muscle calcium channels by [3H]-nifedipine, [3H]-nitrendipine, [3H]-nimodipine and [3H]-PN 200 110

scientific article published on 01 July 1983

Does rosuvastatin increase serum levels of 25-hydroxy-vitamin D?

scientific article

Effect of oc-adrenoceptor agonists on cell membrane potential in renal epitheloid Madin Darby canine kidney cells ⬇️

scientific article published on April 3, 1991

Effects of ion channel toxins and specific neurotoxins on the cyclic nucleotide content of cerebellar slices, primary brain cultures and neural cell lines ⬇️

scientific article published on June 1, 1979

ErratumGenetic Defects in Postsqualene Cholesterol Biosynthesis

scientific article published on 01 May 2000

Evidence for an external location of the dihydropyridine agonist receptor site on smooth muscle and skeletal muscle calcium channels ⬇️

scientific article published on April 1, 1993

Evidence of multiple receptor sites within the putative calcium channel.

scientific article published in October 1982

Functional Consequences of P/Q-type Ca2+Channel Cav2.1 Missense Mutations Associated with Episodic Ataxia Type 2 and Progressive Ataxia ⬇️

scientific article published on December 12, 2001

Genetic defects in postsqualene cholesterol biosynthesis.

scientific article

Human red-blood-cell Ca2+-antagonist binding sites. Evidence for an unusual receptor coupled to the nucleoside transporter

scientific article published on 01 July 1985

Hydrophobic calcium channel ligands: methodical problems and their solution.

scientific article published in November 1989

Identification of 1,4-dihydropyridine binding regions within the alpha 1 subunit of skeletal muscle Ca2+ channels by photoaffinity labeling with diazipine

scientific article published on October 1991

Identification of PK-A phosphorylation sites in the carboxyl terminus of L-type calcium channel alpha 1 subunits.

scientific article

Identification of Voltage Operated Calcium Channels by Binding Studies: Differentiation of Subclasses of Calcium Antagonist Drugs with3H-Nimodipine Radioligand Binding ⬇️

scientific article published on January 1, 1983

Identification of putative calcium channels in skeletal muscle microsomes.

scientific article

Images in cardiovascular medicine. Generalized large vessel arteritis visualized by 18fluorodeoxyglucose-positron emission tomography.

scientific article published on February 2003

Improved micro-perfusion chamber for multiple and rapid solution exchange in adherent single cells.

scientific article published on January 1995

Inhibition of cardiac L-type calcium channels by quaternary amlodipine: implications for pharmacokinetics and access to dihydropyridine binding site.

scientific article published in January 1995

Investigations on the mechanism of cyclic guanosine monophosphate increase due to depolarizing agents as studied with sea anemone toxin II in mouse cerebellar slices ⬇️

scientific article published on June 1, 1979

Ionic modulation of alpha-adrenoceptors.

scientific article published in January 1982

L-type calcium channels: binding domains for dihydropyridines and benzothiazepines are located in close proximity to each other

scientific article published on 01 March 1997

Mammalian β-adrenoceptors: concomitant biospecific elution with protein kinase activity from sepharose-alprenolol ⬇️

scientific article published on November 5, 1981

Mechanism of dihydropyridine interaction with critical binding residues of L-type Ca2+ channel alpha 1 subunits.

scientific article

Molecular basis of drug interaction with L-type Ca2+ channels

scientific article published on 01 August 1998

Molecular cloning and expression of the human delta7-sterol reductase

scientific article

Molecular structure of rat brain apamin receptor: differential photoaffinity labeling of putative K+ channel subunits and target size analysis.

scientific article published in July 1986

Mutations in the gene encoding 3 beta-hydroxysteroid-delta 8, delta 7-isomerase cause X-linked dominant Conradi-Hünermann syndrome

scientific article

Mutations in the Δ7-sterol reductase gene in patients with the Smith–Lemli–Opitz syndrome ⬇️

scientific article published on July 7, 1998

Novel 1,4-dihydropyridine (Bay K 8644) facilitates calcium-dependent [3H]noradrenaline release from PC 12 cells

scientific article published on 01 April 1984

Novel pharmacological chaperones that correct phenylketonuria in mice.

scientific article

Novel sites for phenylalkylamines: characterisation of a sodium-sensitive drug receptor with (−)-[3H]emopamil ⬇️

scientific article published on October 14, 1991

Oral supplementation with calcitriol, calcidiol, vitamin D3 or moderate sun exposure?

scientific article published on 2 May 2013

Pharmacological Analysis of Sterol Δ8-Δ7 Isomerase Proteins with [3H]Ifenprodil ⬇️

scientific article published on September 1, 1998

Pharmacology and structure of high conductance calcium-activated potassium channels.

scientific article

Phenylalkylamine Ca2+ antagonist binding protein. Molecular cloning, tissue distribution, and heterologous expression

scientific article

Photoaffinity labelling of Ca2+ channels with [3H]azidopine.

scientific article

Photoaffinity labelling of the phenylalkylamine receptor of the skeletal muscle transverse-tubule calcium channel.

scientific article published in February 1987

Prospective virtual screening in a sparse data scenario: design of small-molecule TLR2 antagonists.

scientific article

Purification and reconstitution of calcium channel drug-receptor sites.

scientific article published in January 1988

Purification of the putative calcium channel from skeletal muscle with the aid of [3H]-nimodipine binding.

scientific article

Purified calcium channels have three allosterically coupled drug receptors

scientific article published on 01 March 1986

Purified skeletal muscle 1,4-dihydropyridine receptor forms phosphorylation-dependent oligomeric calcium channels in planar bilayers.

scientific article

Putative calcium channel molecular weight determination by target size analysis.

scientific article

Quercetin inhibits tyrosine phosphorylation by the cyclic nucleotide-independent, transforming protein kinase, pp60src

scientific article published on 01 August 1981

Radiation inactivation of alpha 1-adrenoceptors

scientific article published on 01 June 1983

Reversible labeling of a chemosensitizer binding domain of p-glycoprotein with a novel 1,4-dihydropyridine drug transport inhibitor.

scientific article published on February 1996

Sequence Differences between α1Cand α1SCa2+Channel Subunits Reveal Structural Determinants of a Guarded and Modulated Benzothiazepine Receptor

scientific article published in Journal of Biological Chemistry

Solid phase radioimmunoassay for cyclic AMP using staphylococcal protein A-antibody adsorbent ⬇️

scientific article published on May 1, 1977

Solubilization and partial purification of putative calcium channels labelled with [3H]-nimodipine ⬇️

scientific article published on August 1, 1983

Solubilization of a mammalian ?-adrenergic receptor ⬇️

scientific article published on December 1, 1978

Soluble bovine adrenal cortex guanylate cyclase: Effect of sodium nitroprusside, nitrosamines, and hydrophobic ligands on activity, substrate specificity and cation requirement ⬇️

scientific article published on August 1, 1978

Structural basis of drug binding to L Ca2+ channels

scientific article published in March 1998

Target size analysis and molecular properties of Ca2+ channels labelled with [3H]verapamil.

scientific article published in May 1984

Target size analysis of skeletal muscle Ca2+ channels. Positive allosteric heterotropic regulation by d-cis-diltiazem is associated with apparent channel oligomer dissociation.

scientific article published in June 1983

Temperature‐dependent regulation of d‐cis‐[3H]diltiazem binding to Ca2+ channels by 1,4‐dihydropyridine channel agonists and antagonists ⬇️

scientific article published on August 22, 1983

The identification of cytoplasmic membrane calcium-entry channels by ligand-binding studies

scientific article published on 01 December 1984

The increase in hormone-stimulated adenylate cyclase activity following Rous sarcoma virus transformation.

scientific article published in June 1982

The mysteries of sigma receptors: new family members reveal a role in cholesterol synthesis

scientific article (publication date: March 1997)

The preparation of brush border membranes from rat kidney using an aqueous two-phase polymer system

scientific article published on 01 January 1974

Torpor: The Rise and Fall of 3-Monoiodothyronamine from Brain to Gut-From Gut to Brain?

scientific article

Transfer of 1,4-dihydropyridine sensitivity from L-type to class A (BI) calcium channels

scientific article published on 01 January 1996

Uneventful self poisoning with a very high dose of captopril

scientific article published on 01 December 1990

Very high affinity interaction of DPI 201-106 and BDF 8784 enantiomers with the phenylalkylamine-sensitive Ca2(+)-channel in Drosophila head membranes.

scientific article published on February 1991

Visualization of the domain structure of an L-type Ca2+ channel using electron cryo-microscopy.

scientific article published on September 2003

Vitamin D, UV, and skin cancer in the elderly: to expose or not to expose?

scientific article published on 22 December 2010

[125I]-HEAT, a selective, high-affinity, high specific activity ligand for alpha 1-adrenoceptors

scientific article published on 01 December 1981

[125I]-HEAT:fifty percent of the ligand can bind to the alpha1-adrenoceptors with extremely high affinity.

scientific article published in October 1982

alpha-Adrenoceptors in rat brain: sodium changes the affinity of agonists for prazosin sites

scientific article published on 01 February 1980

List of works by Hartmut H. Glossmann

(?)-3H-desmethoxyverapamil labelling of putative calcium channels in brain: autoradiographic distribution and allosteric coupling to 1,4-dihydropyridine and diltiazem binding sites ⬇️

125I-iodipine, a new high affinity ligand for the putative calcium channel.

7-Dehydrocholesterol-dependent proteolysis of HMG-CoA reductase suppresses sterol biosynthesis in a mouse model of Smith-Lemli-Opitz/RSH syndrome

?-Adrenergic receptors in guinea-pig myocardial tissue ⬇️

A marriage of two "Methusalem" drugs for the treatment of psoriasis?: Arguments for a pilot trial with metformin as add-on for methotrexate.

A novel 1,4-dihydropyridine-binding site on mitochondrial membranes from guinea-pig heart, liver and kidney.

A rapid procedure for the purification of cardiac 1,4-dihydropyridine receptors from porcine heart

Adrenal cortex adenylate cyclase. Specific binding sites for 5'-guanylyl-imidodiphosphate in partially purified plasma membranes from bovine adrenal cortex

Alpha 2 adrenoceptors in rat brain: the divalent cation site

Alpha adrenoceptors in rat brain: Direct identification with prazosin ⬇️

Analysis of membrane protein self-association in lipid systems by fluorescence particle counting: application to the dihydropyridine receptor

Association of calcium channel α 1S and β 1a subunits is required for the targeting of β 1a but not of α 1S into skeletal muscle triads ⬇️

Association of the src-gene product of Rous sarcoma virus with a pyruvate-kinase inactivation factor.

Benzothiazepine binding domain of purified L-type calcium channels: direct labeling using a novel fluorescent diltiazem analogue.

Bovine adrenal cortex adenylate cyclase: Properties of the particulate enzyme and effects of guanyl nucleotides ⬇️

Calcium channels from Cyprinus carpio skeletal muscle.

Calcium channels: the beta-subunit increases the affinity of dihydropyridine and Ca2+ binding sites of the alpha 1-subunit.

Calcium- and potassium-channel blockers interact with alpha-adrenoceptors.

Cation sensitivity of [125I]heat binding to alpha 1-adrenoceptors in rat cerebral cortex membranes

Commentary: Lactate-Induced Glucose Output Is Unchanged by Metformin at a Therapeutic Concentration-A Mass Spectrometry Imaging Study of the Perfused Rat Liver

Complex molecular mechanism for dihydropyridine binding to L-type Ca(2+)-channels as revealed by fluorescence resonance energy transfer

Conserved Ca2+-antagonist-binding properties and putative folding structure of a recombinant high-affinity dihydropyridine-binding domain.

Coordination of Ca2+ by the pore region glutamates is essential for high-affinity dihydropyridine binding to the cardiac Ca2+ channel alpha 1 subunit.

Correlation between the negative inotropic potency and binding parameters of 1,4-dihydropyridine and phenylalkylamine calcium channel blockers in cat heart

Differential effects of Ca2+ channel beta1a and beta2a subunits on complex formation with alpha1S and on current expression in tsA201 cells.

Differential labelling of putative skeletal muscle calcium channels by [3H]-nifedipine, [3H]-nitrendipine, [3H]-nimodipine and [3H]-PN 200 110

Does rosuvastatin increase serum levels of 25-hydroxy-vitamin D?

Effect of oc-adrenoceptor agonists on cell membrane potential in renal epitheloid Madin Darby canine kidney cells ⬇️

Effects of ion channel toxins and specific neurotoxins on the cyclic nucleotide content of cerebellar slices, primary brain cultures and neural cell lines ⬇️

ErratumGenetic Defects in Postsqualene Cholesterol Biosynthesis

Evidence for an external location of the dihydropyridine agonist receptor site on smooth muscle and skeletal muscle calcium channels ⬇️

Evidence of multiple receptor sites within the putative calcium channel.

Functional Consequences of P/Q-type Ca2+Channel Cav2.1 Missense Mutations Associated with Episodic Ataxia Type 2 and Progressive Ataxia ⬇️

Genetic defects in postsqualene cholesterol biosynthesis.

Human red-blood-cell Ca2+-antagonist binding sites. Evidence for an unusual receptor coupled to the nucleoside transporter

Hydrophobic calcium channel ligands: methodical problems and their solution.

Identification of 1,4-dihydropyridine binding regions within the alpha 1 subunit of skeletal muscle Ca2+ channels by photoaffinity labeling with diazipine

Identification of PK-A phosphorylation sites in the carboxyl terminus of L-type calcium channel alpha 1 subunits.

Identification of Voltage Operated Calcium Channels by Binding Studies: Differentiation of Subclasses of Calcium Antagonist Drugs with3H-Nimodipine Radioligand Binding ⬇️

Identification of putative calcium channels in skeletal muscle microsomes.

Images in cardiovascular medicine. Generalized large vessel arteritis visualized by 18fluorodeoxyglucose-positron emission tomography.

Improved micro-perfusion chamber for multiple and rapid solution exchange in adherent single cells.

Inhibition of cardiac L-type calcium channels by quaternary amlodipine: implications for pharmacokinetics and access to dihydropyridine binding site.

Investigations on the mechanism of cyclic guanosine monophosphate increase due to depolarizing agents as studied with sea anemone toxin II in mouse cerebellar slices ⬇️

Ionic modulation of alpha-adrenoceptors.

L-type calcium channels: binding domains for dihydropyridines and benzothiazepines are located in close proximity to each other

Mammalian β-adrenoceptors: concomitant biospecific elution with protein kinase activity from sepharose-alprenolol ⬇️

Mechanism of dihydropyridine interaction with critical binding residues of L-type Ca2+ channel alpha 1 subunits.

Molecular basis of drug interaction with L-type Ca2+ channels

Molecular cloning and expression of the human delta7-sterol reductase

Molecular structure of rat brain apamin receptor: differential photoaffinity labeling of putative K+ channel subunits and target size analysis.

Mutations in the gene encoding 3 beta-hydroxysteroid-delta 8, delta 7-isomerase cause X-linked dominant Conradi-Hünermann syndrome

Mutations in the Δ7-sterol reductase gene in patients with the Smith–Lemli–Opitz syndrome ⬇️

Novel 1,4-dihydropyridine (Bay K 8644) facilitates calcium-dependent [3H]noradrenaline release from PC 12 cells

Novel pharmacological chaperones that correct phenylketonuria in mice.

Novel sites for phenylalkylamines: characterisation of a sodium-sensitive drug receptor with (−)-[3H]emopamil ⬇️

Oral supplementation with calcitriol, calcidiol, vitamin D3 or moderate sun exposure?

Pharmacological Analysis of Sterol Δ8-Δ7 Isomerase Proteins with [3H]Ifenprodil ⬇️

Pharmacology and structure of high conductance calcium-activated potassium channels.

Phenylalkylamine Ca2+ antagonist binding protein. Molecular cloning, tissue distribution, and heterologous expression

Photoaffinity labelling of Ca2+ channels with [3H]azidopine.

Photoaffinity labelling of the phenylalkylamine receptor of the skeletal muscle transverse-tubule calcium channel.

Prospective virtual screening in a sparse data scenario: design of small-molecule TLR2 antagonists.

Purification and reconstitution of calcium channel drug-receptor sites.

Purification of the putative calcium channel from skeletal muscle with the aid of [3H]-nimodipine binding.

Purified calcium channels have three allosterically coupled drug receptors

Purified skeletal muscle 1,4-dihydropyridine receptor forms phosphorylation-dependent oligomeric calcium channels in planar bilayers.

Putative calcium channel molecular weight determination by target size analysis.

Quercetin inhibits tyrosine phosphorylation by the cyclic nucleotide-independent, transforming protein kinase, pp60src

Radiation inactivation of alpha 1-adrenoceptors

Reversible labeling of a chemosensitizer binding domain of p-glycoprotein with a novel 1,4-dihydropyridine drug transport inhibitor.

Sequence Differences between α1Cand α1SCa2+Channel Subunits Reveal Structural Determinants of a Guarded and Modulated Benzothiazepine Receptor

Solid phase radioimmunoassay for cyclic AMP using staphylococcal protein A-antibody adsorbent ⬇️

Solubilization and partial purification of putative calcium channels labelled with [3H]-nimodipine ⬇️

Solubilization of a mammalian ?-adrenergic receptor ⬇️

Soluble bovine adrenal cortex guanylate cyclase: Effect of sodium nitroprusside, nitrosamines, and hydrophobic ligands on activity, substrate specificity and cation requirement ⬇️

Structural basis of drug binding to L Ca2+ channels

Target size analysis and molecular properties of Ca2+ channels labelled with [3H]verapamil.

Target size analysis of skeletal muscle Ca2+ channels. Positive allosteric heterotropic regulation by d-cis-diltiazem is associated with apparent channel oligomer dissociation.