List of works - Václav Bazgier

2,6,9-Trisubstituted purines as CRK3 kinase inhibitors with antileishmanial activity in vitro

scientific article published on 16 April 2015

A novel series of highly potent 2,6,9-trisubstituted purine cyclin-dependent kinase inhibitors

scientific article published on 24 July 2013

Acetylated deoxycholic (DCA) and cholic (CA) acids are potent ligands of pregnane X (PXR) receptor

scientific article

Antiallergic effects of pigments isolated from green sea urchin (Strongylocentrotus droebachiensis) shells

scientific article

Biological activities of new monohydroxylated brassinosteroid analogues with a carboxylic group in the side chain

scientific article published on 21 April 2014

Characterization of a Pyrazolo[4,3-d]pyrimidine Inhibitor of Cyclin-Dependent Kinases 2 and 5 and Aurora A With Pro-Apoptotic and Anti-Angiogenic Activity In Vitro

scientific article published on 22 July 2015

Discovery of N2-(4-Amino-cyclohexyl)-9-cyclopentyl- N6-(4-morpholin-4-ylmethyl-phenyl)- 9H-purine-2,6-diamine as a Potent FLT3 Kinase Inhibitor for Acute Myeloid Leukemia with FLT3 Mutations.

scientific article published on 19 April 2018

Exponential repulsion improves structural predictability of molecular docking

scientific article published on 13 September 2016

Fluorone dyes have binding sites on both cytoplasmic and extracellular domains of Na,K-ATPase

scientific article published on 8 November 2012

MOLEonline: a web-based tool for analyzing channels, tunnels and pores (2018 update).

scientific article published in July 2018

Membrane-attached mammalian cytochromes P450: An overview of the membrane's effects on structure, drug binding, and interactions with redox partners.

scientific article published on 5 March 2018

MolMeDB: Molecules on Membranes Database

scientific article published on 19 November 2018

Mole 2.5 - Tool for Detection and Analysis of Macromolecular Pores and Channels

scholarly article by Karel Berka et al published February 2017 in Biophysical Journal

Novel N-substituted indole Schiff bases as dual inhibitors of cyclooxygenase-2 and 5-lipoxygenase enzymes: Synthesis, biological activities in vitro and docking study

scientific article published on 10 August 2016

Novel thidiazuron-derived inhibitors of cytokinin oxidase/dehydrogenase

scientific article

RH421 binds into the ATP-binding site on the Na+/K+-ATPase

scientific article published on 31 July 2017

Synthesis and kinase inhibitory activity of new sulfonamide derivatives of pyrazolo[4,3-e][1,2,4]triazines

scientific article published on 18 March 2014

Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors

scientific article published on 19 December 2015

List of works by Václav Bazgier

2,6,9-Trisubstituted purines as CRK3 kinase inhibitors with antileishmanial activity in vitro

A novel series of highly potent 2,6,9-trisubstituted purine cyclin-dependent kinase inhibitors

Acetylated deoxycholic (DCA) and cholic (CA) acids are potent ligands of pregnane X (PXR) receptor

Antiallergic effects of pigments isolated from green sea urchin (Strongylocentrotus droebachiensis) shells

Biological activities of new monohydroxylated brassinosteroid analogues with a carboxylic group in the side chain

Characterization of a Pyrazolo[4,3-d]pyrimidine Inhibitor of Cyclin-Dependent Kinases 2 and 5 and Aurora A With Pro-Apoptotic and Anti-Angiogenic Activity In Vitro

Discovery of N2-(4-Amino-cyclohexyl)-9-cyclopentyl- N6-(4-morpholin-4-ylmethyl-phenyl)- 9H-purine-2,6-diamine as a Potent FLT3 Kinase Inhibitor for Acute Myeloid Leukemia with FLT3 Mutations.

Exponential repulsion improves structural predictability of molecular docking

Fluorone dyes have binding sites on both cytoplasmic and extracellular domains of Na,K-ATPase

MOLEonline: a web-based tool for analyzing channels, tunnels and pores (2018 update).

Membrane-attached mammalian cytochromes P450: An overview of the membrane's effects on structure, drug binding, and interactions with redox partners.

MolMeDB: Molecules on Membranes Database

Mole 2.5 - Tool for Detection and Analysis of Macromolecular Pores and Channels

Novel N-substituted indole Schiff bases as dual inhibitors of cyclooxygenase-2 and 5-lipoxygenase enzymes: Synthesis, biological activities in vitro and docking study

Novel thidiazuron-derived inhibitors of cytokinin oxidase/dehydrogenase

RH421 binds into the ATP-binding site on the Na+/K+-ATPase

Synthesis and kinase inhibitory activity of new sulfonamide derivatives of pyrazolo[4,3-e][1,2,4]triazines

Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors