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List of works by Dale O Kiesewetter

(18)F-alfatide II and (18)F-FDG dual-tracer dynamic PET for parametric, early prediction of tumor response to therapy

scientific article

18F-Labeled Single-Stranded DNA Aptamer for PET Imaging of Protein Tyrosine Kinase-7 Expression

scientific article

18F-radiolabeled analogs of exendin-4 for PET imaging of GLP-1 in insulinoma

scientific article published on December 15, 2011

64Cu-AMD3100--a novel imaging agent for targeting chemokine receptor CXCR4.

scientific article published on 15 January 2009

68Ga-NOTA-Exendin-4 PET/CT in Localization of an Occult Insulinoma and Appearance of Coexisting Esophageal Carcinoma

scientific article published on 4 December 2015

68Ga-NOTA-exendin-4 PET/CT in detection of occult insulinoma and evaluation of physiological uptake

scientific article

76BrBMK‐152, a nonpeptide analogue, with high affinity and low nonspecific binding for the corticotropin‐releasing factor type 1 receptor

scientific article published on April 11, 2011

<sup>177</sup>Lu-DOTA-EB-TATE, A Radiolabeled Analog of Somatostatin Receptor Type 2, for the Imaging and Treatment of Thyroid Cancer

scientific article published on 22 December 2020

A Logic-Gated Modular Nanovesicle Enables Programmable Drug Release for On-Demand Chemotherapy

A cyclic HSV1-TK reporter for real-time PET imaging of apoptosis

scientific article published on 20 March 2014

A paclitaxel prodrug with bifunctional folate and albumin binding moieties for both passive and active targeted cancer therapy.

scientific article

A photothermally responsive nanoprobe for bioimaging based on Edman degradation

scientific article published on 5 May 2016

A potential cholinergic mechanism of procaine's limbic activation

scientific article published in July 2004

A symmetrical fluorous dendron-cyanine dye-conjugated bimodal nanoprobe for quantitative 19F MRI and NIR fluorescence bioimaging

scientific article

Al[18F]NOTA-T140 Peptide for Noninvasive Visualization of CXCR4 Expression

scientific article published on July 2015

Albumin-Binding Evans Blue Derivatives for Diagnostic Imaging and Production of Long-Acting Therapeutics

scientific article published on 28 September 2016

Albumin-chaperoned cyanine dye yields superbright NIR-II fluorophore with enhanced pharmacokinetics

scientific article published on 13 September 2019

An automated one-step one-pot [(18)F]FCWAY synthesis: development and minimization of chemical impurities

scientific article

Antiretroviral tissue kinetics: in vivo imaging using positron emission tomography

scientific article published on 10 August 2009

Application of LC-MS to the analysis of new radiopharmaceuticals

scientific article

Application of highly sensitive UPLC-MS to determine biodistribution at tracer doses: validation with the 5-HT1A ligand [(18)F]FPWAY.

scientific article published on 26 March 2009

Applications of LC-MS in PET radioligand development and metabolic elucidation

scientific article published on July 2010

Automated radiochemical synthesis of [18F]FBEM: a thiol reactive synthon for radiofluorination of peptides and proteins

scientific article

Bioinspired nanocomplex for spatiotemporal imaging of sequential mRNA expression in differentiating neural stem cells

scientific article

Boramino acid as a marker for amino acid transporters

scientific article published on 11 September 2015

Changes in HER2 expression in breast cancer xenografts after therapy can be quantified using PET and (18)F-labeled affibody molecules

scientific article published on 12 June 2009

Chelator-free (64)Cu-integrated gold nanomaterials for positron emission tomography imaging guided photothermal cancer therapy

scientific article

Chemical Conjugation of Evans Blue Derivative: A Strategy to Develop Long-Acting Therapeutics through Albumin Binding

scientific article published on January 2016

Comparison Study of [18F]FAl-NOTA-PRGD2, [18F]FPPRGD2, and [68Ga]Ga-NOTA-PRGD2 for PET Imaging of U87MG Tumors in Mice

scientific article published on November 3, 2011

Comparison of (18)F-labeled CXCR4 antagonist peptides for PET imaging of CXCR4 expression

scientific article published on December 2013

Comparison of three dimeric 18F-AlF-NOTA-RGD tracers

scientific article published on April 2014

Correction to "Novel 19F Activatable Probe for the Detection of Matrix Metalloprotease-2 Activity by MRI/MRS".

scientific article published on 9 March 2017

Design of a functional cyclic HSV1-TK reporter and its application to PET imaging of apoptosis

scientific article published on 30 April 2015

Determination of [18F]FCWAY, [18F]FP-TZTP, and their metabolites in plasma using rapid and efficient liquid-liquid and solid phase extractions

scientific article published on April 1, 2003

Development of 5-HT1A receptor radioligands to determine receptor density and changes in endogenous 5-HT.

scientific article published in May 2006

Development of a new thiol site-specific prosthetic group and its conjugation with [Cys(40)]-exendin-4 for in vivo targeting of insulinomas

scientific article published on 28 June 2013

Drug Delivery: NIR-Responsive On-Demand Release of CO from Metal Carbonyl-Caged Graphene Oxide Nanomedicine (Adv. Mater. 42/2015)

scientific article published in November 2015

Dual-factor triggered fluorogenic nanoprobe for ultrahigh contrast and subdiffraction fluorescence imaging.

scientific article

Enantiomeric radiochemical synthesis of R and S (1-(6-amino-9H-purin-9-yl)-3-fluoropropan-2-yloxy)methylphosphonic acid (FPMPA)

scientific article published on March 2008

Engineered Zn(II)-Dipicolylamine-Gold Nanorod Provides Effective Prostate Cancer Treatment by Combining siRNA Delivery and Photothermal Therapy

scientific article published on 26 September 2017

Estimation of paclitaxel biodistribution and uptake in human-derived xenografts in vivo with (18)F-fluoropaclitaxel.

scientific article published on November 2005

Evaluation of [18F]fluoroxanomeline {5-{4-[(6-[18F]fluorohexyl)oxy]-1,2,5-thiadiazol-3-yl}-1-methyl-1,2,3,6-tetrahydropyridine} in muscarinic knockout mice

scientific article published on 17 January 2007

Evaluation of an [18F]AlF-NOTA Analog of Exendin-4 for Imaging of GLP-1 Receptor in Insulinoma

scientific article published on October 17, 2012

Evaluation of fluorine-labeled gastrin-releasing peptide receptor (GRPR) agonists and antagonists by LC/MS

scientific article published on February 22, 2012

Evans Blue Attachment Enhances Somatostatin Receptor Subtype-2 Imaging and Radiotherapy

scientific article published in January 2018

Fluorine-18 radiochemistry, labeling strategies and synthetic routes

scientific article

Fluoro-, bromo-, and iodopaclitaxel derivatives: synthesis and biological evaluation

scientific article

Glucagon-Like Peptide-1 Receptor PET/CT with 68Ga-NOTA-Exendin-4 for Detecting Localized Insulinoma: A Prospective Cohort Study

scientific article published on 21 January 2016

Higher in vivo muscarinic-2 receptor distribution volumes in aging subjects with an apolipoprotein E-epsilon4 allele

scientific article published in September 2003

Identification of metabolites of fluorine-18-labeled M2 muscarinic receptor agonist, 3-(3-[(3-fluoropropyl)thio]-1,2,5-thiadiazol-4-yl)-1,2,5,6-tetrahydro-1-methylpyridine, produced by human and rat hepatocytes

scientific article published in January 2002

Imaging of the muscarinic acetylcholine neuroreceptor in rats with the M2 selective agonist [18F]FP-TZTP

scientific article published on August 9, 2011

Improvement of CXCR4 tracer specificity for PET imaging

scientific article published on September 22, 2011

In Vivo Labeling of Serum Albumin for PET.

scientific article

In vivo albumin labeling and lymphatic imaging

scientific article

In vivo muscarinic 2 receptor imaging in cognitively normal young and older volunteers

scientific article

Increased uptake of [¹²³I]meta-iodobenzylguanidine, [¹⁸F]fluorodopamine, and [³H]norepinephrine in mouse pheochromocytoma cells and tumors after treatment with the histone deacetylase inhibitors

scientific article

Inhibition of [18F]FP-TZTP binding by loading doses of muscarinic agonists P-TZTP or FP-TZTP in vivo is not due to agonist-induced reduction in cerebral blood flow

scientific article

Intrinsically radioactive [64Cu]CuInS/ZnS quantum dots for PET and optical imaging: improved radiochemical stability and controllable Cerenkov luminescence

scientific article

LC/MS evaluation of metabolism and membrane transport of bombesin peptides

scientific article

Liquid chromatography-tandem mass spectrometry identification of metabolites of three phenylcarboxyl derivatives of the 5-HT(1A) antagonist, N-(2-(4-(2-methoxyphenyl)-1-piperazinyl)ethyl)-N-(2-pyridyl) trans-4-fluorocyclohexanecarboxamide (FCWAY), p

scientific article published in November 2002

Long-term multimodal imaging of tumor draining sentinel lymph nodes using mesoporous silica-based nanoprobes

scientific article published on 16 March 2012

Longitudinal PET Imaging of Doxorubicin-Induced Cell Death with 18F-Annexin V

scientific article published on December 1, 2012

Longitudinal PET imaging of muscular inflammation using 18F-DPA-714 and 18F-Alfatide II and differentiation with tumors

scientific article published on 26 February 2014

MicroPET Imaging of Integrin αvβ3 Expressing Tumors Using 89Zr-RGD Peptides

scientific article published on December 1, 2011

Monitoring Tumor Hypoxia Using (18)F-FMISO PET and Pharmacokinetics Modeling after Photodynamic Therapy

scientific article published on 22 August 2016

N-Succinimidyl 4-[18F]-fluoromethylbenzoate-labeled dimeric RGD peptide for imaging tumor integrin expression

scientific article published on December 31, 2011

NIR-Responsive On-Demand Release of CO from Metal Carbonyl-Caged Graphene Oxide Nanomedicine

scientific article published on 24 September 2015

New Methods for Labeling RGD Peptides with Bromine-76

scientific article published on August 22, 2011

Novel "Add-On" Molecule Based on Evans Blue Confers Superior Pharmacokinetics and Transforms Drugs to Theranostic Agents

scientific article published on 22 November 2016

Novel 19F activatable probe for the detection of matrix metalloprotease-2 activity by MRI/MRS.

scientific article

Novel Method for Radiolabeling and Dimerizing Thiolated Peptides Using (18)F-Hexafluorobenzene

scientific article (publication date: 21 October 2015)

One-pot two-step radiosynthesis of a new (18)F-labeled thiol reactive prosthetic group and its conjugate for insulinoma imaging

scientific article

One-step (18)F labeling of biomolecules using organotrifluoroborates

scientific article (publication date: September 2015)

PET imaging of CXCR4 using copper-64 labeled peptide antagonist

scientific article

PET imaging of EGF receptors using [18F]FBEM-EGF in a head and neck squamous cell carcinoma model

scientific article published on 23 November 2011

PET imaging of angiogenesis after myocardial infarction/reperfusion using a one-step labeled integrin-targeted tracer 18F-AlF-NOTA-PRGD2

scientific article published on January 25, 2012

PET imaging of early response to the tyrosine kinase inhibitor ZD4190

scientific article published on March 1, 2011

PET imaging of neuroinflammation in a rat traumatic brain injury model with radiolabeled TSPO ligand DPA-714.

scientific article

PET imaging of tenascin-C with a radiolabeled single-stranded DNA aptamer

scientific article published on 19 February 2015

PET of Glucagonlike Peptide Receptor Upregulation After Myocardial Ischemia or Reperfusion Injury

scientific article published on November 8, 2012

PET of HER2-positive pulmonary metastases with 18F-ZHER2:342 affibody in a murine model of breast cancer: comparison with 18F-FDG.

scientific article published on 11 May 2012

PET of Insulinoma Using 18F-FBEM-EM3106B, a New GLP-1 Analogue

scientific article published on August 19, 2011

PET of Tumor CXCR4 Expression with 4-18F-T140

scientific article published on October 18, 2010

PET-guided evaluation and optimization of internalized antibody-drug conjugates targeting erythropoietin producing hepatoma A2 receptor.

scientific article

Photosensitizer loaded nano-graphene for multimodality imaging guided tumor photodynamic therapy

scientific article published on 15 January 2014

Positron Emission Tomography Imaging of Tumors Expressing the Human Chemokine Receptor CXCR4 in Mice with the Use of 64Cu-AMD3100

scientific article published on February 1, 2012

Potential of PET to Predict the Response to Trastuzumab Treatment in an ErbB2-Positive Human Xenograft Tumor Model

scientific article published on March 12, 2012

Prokineticin receptor 1 antagonist PC-10 as a biomarker for imaging inflammatory pain

scientific article published on 18 March 2011

Purification of the precursor for the automated radiosynthesis of [18F]FCWAY by counter-current chromatography

scientific article published in April 2004

Quantification of Tumor Vascular Permeability and Blood Volume by Positron Emission Tomography

scientific article published on 14 June 2017

Quantifying conversion of linoleic to arachidonic and other n-6 polyunsaturated fatty acids in unanesthetized rats

scientific article

Quantitative Analysis and Comparison Study of [18F]AlF-NOTA-PRGD2, [18F]FPPRGD2 and [68Ga]Ga-NOTA-PRGD2 Using a Reference Tissue Model

scientific article (publication date: 2012)

Quantitative Analysis and Parametric Imaging of 18F-Labeled Monomeric and Dimeric RGD Peptides Using Compartment Model

scientific article published on December 1, 2012

Quantitative Evaluation of Tumor Early Response to a Vascular-Disrupting Agent with Dynamic PET.

scientific article published on 21 April 2015

RETRACTED ARTICLE: Aging decreases rate of docosahexaenoic acid synthesis-secretion from circulating unesterified α-linolenic acid by rat liver

scientific article published on March 3, 2012

RETRACTED: Liver conversion of docosahexaenoic and arachidonic acids from their 18-carbon precursors in rats on a DHA-free but α-LNA-containing n−3 PUFA adequate diet

scientific article published on May 30, 2011

Radiolabeling of HER2 specific Affibody(R) molecule with F-18.

scientific article published on September 2008

Rapid and Simple One-Step F-18 Labeling of Peptides

scientific article published on February 21, 2011

Rational design of matrix metalloproteinase-13 activatable probes for enhanced specificity

scientific article

Reduced muscarinic type 2 receptor binding in subjects with bipolar disorder

scientific article published in July 2006

Routine quality control of recycled target [18O]water by capillary electrophoresis and gas chromatography

scientific article published on October 1, 2003

Self-illuminating 64Cu-doped CdSe/ZnS nanocrystals for in vivo tumor imaging

scientific article published on 17 January 2014

Site-Specific Labeling of scVEGF with Fluorine-18 for Positron Emission Tomography Imaging

scientific article

Size Dependent Kinetics of Gold Nanorods in EPR Mediated Tumor Delivery

scientific article

Species differences in metabolites of PET ligands: serotonergic 5-HT1A receptor antagonists 3-trans-FCWAY and 3-cis-FCWAY.

scientific article published in November 2006

Stability analysis of glutamic acid linked peptides coupled to NOTA through different chemical linkages

scientific article

Stable Evans Blue Derived Exendin-4 Peptide for Type 2 Diabetes Treatment

scientific article published on 07 December 2015

Sticky nanoparticles: a platform for siRNA delivery by a bis(zinc(II) dipicolylamine)-functionalized, self-assembled nanoconjugate

scientific article published on 23 November 2011

Striatal adenosine A2A receptor-mediated positron emission tomographic imaging in 6-hydroxydopamine-lesioned rats using [18F]-MRS5425

scientific article published on March 30, 2011

Synthesis and characterization of [76Br]-labeled high-affinity A3 adenosine receptor ligands for positron emission tomography

scientific article published on January 2009

The Synthesis and In Vivo Pharmacokinetics of Fluorinated Arachidonic Acid: Implications for Imaging Neuroinflammation

scientific article published on July 31, 2012

The automated radiosynthesis of [18F]FP-TZTP.

scientific article published in January 2003

Usefulness of [18F]-DA and [18F]-DOPA for PET imaging in a mouse model of pheochromocytoma

scientific article published on September 29, 2011

Whole-body synthesis secretion of docosahexaenoic acid from circulating eicosapentaenoic acid in unanesthetized rats

scientific article published on July 2009

Whole-body synthesis-secretion rates of long-chain n-3 PUFAs from circulating unesterified alpha-linolenic acid in unanesthetized rats

scientific article published on 11 December 2008

[(18)F]DPA-714 PET imaging of AMD3100 treatment in a mouse model of stroke

scientific article

[18F]FBEM-Z(HER2:342)-Affibody molecule-a new molecular tracer for in vivo monitoring of HER2 expression by positron emission tomography

scientific article published on 22 December 2007

pH-Sensitive Fluorescent Dyes: Are They Really pH-Sensitive in Cells?

scientific article published on March 25, 2013