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List of works by Peter J. H. Scott

(-)-[(18) F]Flubatine: evaluation in rhesus monkeys and a report of the first fully automated radiosynthesis validated for clinical use.

scientific article published on 16 July 2013

A Kinome-Wide Selective Radiolabeled TrkB/C Inhibitor for in Vitro and in Vivo Neuroimaging: Synthesis, Preclinical Evaluation, and First-in-Human

scientific article published on 11 July 2017

A fully-automated one-pot synthesis of [18F]fluoromethylcholine with reduced dimethylaminoethanol contamination via [18F]fluoromethyl tosylate.

scientific article published on 24 April 2013

A spot test for determination of residual TBA levels in 18F-radiotracers for human use using Dragendorff reagent

scientific article published on 01 October 2020

An Updated Synthesis of N<sub>1</sub> '-([<sup>11</sup> C]Methyl)Naltrindole for Positron Emission Tomography Imaging of the Delta Opioid Receptor

scientific article published on 03 December 2020

An updated synthesis of [11 C]carfentanil for positron emission tomography (PET) imaging of the μ-opioid receptor.

scientific article published on 17 April 2017

Automated production of [11C]acetate and [11C]palmitate using a modified GE Tracerlab FXC-Pro ⬇️

scientific article published on January 8, 2011

Automated synthesis of PET radiotracers by copper-mediated 18 F-fluorination of organoborons: Importance of the order of addition and competing protodeborylation.

scientific article

Automated synthesis of [68Ga]oxine, improved preparation of 68Ga-labeled erythrocytes for blood-pool imaging, and preclinical evaluation in rodents

scientific article published on 01 February 2018

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6

scientific article published on 28 December 2019

C-H 18F-fluorination of 8-methylquinolines with Ag[18F]F

scientific article published on 01 March 2019

Carbon-11 labeled cathepsin K inhibitors: syntheses and preliminary in vivo evaluation

scientific article published on 18 February 2014

Classics in Neuroimaging: Development of PET Tracers for Imaging Monoamine Oxidases

scientific article published on 21 February 2019

Classics in Neuroimaging: Development of Positron Emission Tomography Tracers for Imaging the GABAergic Pathway

scientific article published on 24 June 2020

Classics in Neuroimaging: Shedding Light on Opioid Receptors with Positron Emission Tomography Imaging

scientific article published on 24 September 2020

Clinical Applications of Radiolabeled Peptides for PET

scientific article published on 07 June 2017

Clinical Applications of Small-molecule PET Radiotracers: Current Progress and Future Outlook.

scientific article published on 11 July 2017

Copper(II)-Mediated [C]Cyanation of Arylboronic Acids and Arylstannanes

scientific article published on 27 February 2018

Copper-Mediated Aminoquinoline-Directed Radiofluorination of Aromatic C−H Bonds with K18 F

scientific article published on 18 January 2019

Copper-Mediated Radiofluorination of Arylstannanes with [18F]KF.

scientific article published on 10 October 2016

Copper-catalyzed [18F]fluorination of (mesityl)(aryl)iodonium salts

scientific article published on 3 June 2014

Cu-Mediated C-H 18F-Fluorination of Electron-Rich (Hetero)arenes

scientific article published on 30 June 2017

Cyclotron-based production of 68Ga, [68Ga]GaCl3, and [68Ga]Ga-PSMA-11 from a liquid target

scientific article published on 12 November 2020

DARK Classics in Chemical Neuroscience: Cocaine

scientific article published on 24 April 2018

Determination of residual Kryptofix 2.2.2 levels in [18F]-labeled radiopharmaceuticals for human use.

scientific article published on 23 May 2007

Deuterium Kinetic Isotope Effect Studies of a Potential in Vivo Metabolic Trapping Agent for Monoamine Oxidase B

scientific article published on 17 August 2018

Development and implementation of ISAR, a new synthesis platform for radiopharmaceutical production

scientific article published on 18 September 2019

Development of Customized [18F]Fluoride Elution Techniques for the Enhancement of Copper-Mediated Late-Stage Radiofluorination.

scientific article published on 22 March 2017

Development of Positron Emission Tomography Radiotracers for the GABA Transporter 1

scientific article published on 24 May 2018

Enhanced radiosyntheses of [¹¹C]raclopride and [¹¹C]DASB using ethanolic loop chemistry.

scientific article

Ethanolic carbon-11 chemistry: the introduction of green radiochemistry

scientific article

Evaluating Cholinergic Receptor Expression in Guinea Pig Primary Auditory and Rostral Belt Cortices After Noise Damage Using [3H]Scopolamine and [18F]Flubatine Autoradiography.

scientific article published in January 2019

Evaluation of Enzyme Substrate Radiotracers as PET/MRS Hybrid Imaging Agents

scientific article published on 03 October 2018

Evaluation of [(11)C]N-Methyl Lansoprazole as a Radiopharmaceutical for PET Imaging of Tau Neurofibrillary Tangles.

scientific article

Evaluation of [18F]-N-Methyl lansoprazole as a Tau PET Imaging Agent in First-in-Human Studies

scientific article published on 15 January 2020

First-in-Human Brain Imaging of [18F]TRACK, a PET tracer for Tropomyosin Receptor Kinases

scientific article published on 29 April 2019

First-in-Human Studies of [18F] Fluorohydroxyphenethylguanidines

scientific article published on 01 December 2018

Fluorine-18 patents (2009-2015). Part 1: novel radiotracers

scientific article published on 16 December 2015

Fluorine-18 patents (2009-2015). Part 2: new radiochemistry.

scientific article published on September 2016

Fully automated preparation of [11C]choline and [18F]fluoromethylcholine using TracerLab synthesis modules and facilitated quality control using analytical HPLC

scientific article published on 13 October 2010

Fully automated radiosynthesis of [¹¹C]PBR28, a radiopharmaceutical for the translocator protein (TSPO) 18 kDa, using a GE TRACERlab FXC-Pro

scientific article published on 29 March 2012

Gallium-68: methodology and novel radiotracers for positron emission tomography (2012-2017)

scientific article published on 01 August 2018

Green approaches to late-stage fluorination: radiosyntheses of (18)F-labelled radiopharmaceuticals in ethanol and water.

scientific article published on 24 August 2015

Guest Editorial

scientific article published on 29 June 2017

High affinity radiopharmaceuticals based upon lansoprazole for PET imaging of aggregated tau in Alzheimer's disease and progressive supranuclear palsy: synthesis, preclinical evaluation, and lead selection

scientific article (publication date: 20 August 2014)

High-Yielding Automated Convergent Synthesis of No-Carrier-Added [11C-Carbonyl]-Labeled Amino Acids Using the Strecker Reaction.

scientific article published on 7 November 2016

Highlighting the Versatility of the Tracerlab Synthesis Modules. Part 1: Fully Automated Production of [F]Labelled Radiopharmaceuticals using a Tracerlab FX(FN).

scientific article

Identification of AV-1451 as a Weak, Nonselective Inhibitor of Monoamine Oxidase

scientific article published on 05 August 2019

Identification of [18F]TRACK, a Fluorine-18-Labeled Tropomyosin Receptor Kinase (Trk) Inhibitor for PET Imaging

scientific article published on 19 December 2017

In Vivo Metabolic Trapping Radiotracers for Imaging Monoamine Oxidase-A and -B Enzymatic Activity.

scientific article published on 22 September 2015

Intranasal Opioid Administration in Rhesus Monkeys: PET Imaging and Antinociception.

scientific article published on 13 September 2016

Is logP truly dead?

scientific article

Issues in preclinical radiopharmaceutical research: Significance, relevance and reproducibility

scientific article published on 03 September 2018

Late-stage [(18)F]Fluorination: New Solutions to Old Problems

scientific article published on December 2014

Methods for the incorporation of carbon-11 to generate radiopharmaceuticals for PET imaging

scientific article published on 01 January 2009

Moving Metal-Mediated (18)F-Fluorination from Concept to Clinic.

scientific article published on 14 March 2016

NHC-Copper Mediated Ligand-Directed Radiofluorination of Aryl Halides

scientific article published on 10 April 2020

Novel fluorine-18 PET radiotracers based on flumazenil for GABAA imaging in the brain.

scientific article published on 23 July 2013

Novel strategies for fluorine-18 radiochemistry

scientific article published on 23 December 2011

One-pot synthesis of high molar activity 6-[18F]fluoro-l-DOPA by Cu-mediated fluorination of a BPin precursor

scientific article published on 19 September 2019

Preclinical Evaluation of 11C-Sarcosine as a Substrate of Proton-Coupled Amino Acid Transporters and First Human Application in Prostate Cancer.

scientific article published on 16 March 2017

Radiochemistry, PET Imaging, and the Internet of Chemical Things

scientific article

Radioligands for Tropomyosin Receptor Kinase (Trk) Positron Emission Tomography Imaging

scientific article published on 03 January 2019

Radionuclide Imaging for Neuroscience: Current Opinion and Future Directions

scientific article published on 01 January 2020

Radiosyntheses using fluorine-18: the art and science of late stage fluorination

scientific article

Radiosynthesis of [C]LY2795050 for Preclinical and Clinical PET Imaging Using Cu(II)-Mediated Cyanation

scientific article published on 13 November 2018

Ring opening of epoxides with [18F]FeF species to produce [18F]fluorohydrin PET imaging agents

scientific article published on 01 May 2019

Structural Basis for Achieving GSK-3β Inhibition with High Potency, Selectivity, and Brain Exposure for Positron Emission Tomography Imaging and Drug Discovery

scientific article published on 21 October 2019

Synthesis and Evaluation of [(18)F]RAGER: A First Generation Small-Molecule PET Radioligand Targeting the Receptor for Advanced Glycation Endproducts.

scientific article published on 15 January 2016

Synthesis and Initial In Vivo Evaluation of [C]AZ683-A Novel PET Radiotracer for Colony Stimulating Factor 1 Receptor (CSF1R)

scientific article published on 13 December 2018

Synthesis and Initial in Vivo Studies with [(11)C]SB-216763: The First Radiolabeled Brain Penetrative Inhibitor of GSK-3.

scientific article published on 10 March 2015

Synthesis and evaluation of [(11)C]PBD150, a radiolabeled glutaminyl cyclase inhibitor for the potential detection of Alzheimer's disease prior to amyloid β aggregation.

scientific article published on June 2015

Synthesis and evaluation of [(11)C]PyrATP-1, a novel radiotracer for PET imaging of glycogen synthase kinase-3β (GSK-3β)

scientific article

Synthesis and pre-clinical evaluation of a potential radiotracer for PET imaging of the dopamine D3 receptor.

scientific article

Synthesis of Diverse (11)C-Labeled PET Radiotracers via Direct Incorporation of [(11)C]CO2.

scientific article

Synthesis of [18F]Arenes via the Copper-Mediated [18F]Fluorination of Boronic Acids

scientific article published on 14 November 2015

Synthesis of high-molar-activity [18F]6-fluoro-L-DOPA suitable for human use via Cu-mediated fluorination of a BPin precursor

scientific article published on 08 April 2020

Targeted nanoparticles for multimodal imaging of the receptor for advanced glycation end-products

scientific article published on 01 December 2018

Targeting Metal-Aβ Aggregates with Bifunctional Radioligand [(11)C]L2-b and a Fluorine-18 Analogue [(18)F]FL2-b

scientific article

The Effects of Intramuscular Naloxone Dose on Mu Receptor Displacement of Carfentanil in Rhesus Monkeys

scientific article published on 17 March 2020

Use of 55 PET radiotracers under approval of a Radioactive Drug Research Committee (RDRC)

scientific article published on 11 November 2020

[(11)C]Ascorbic and [(11)C]dehydroascorbic acid, an endogenous redox pair for sensing reactive oxygen species using positron emission tomography

scientific article published on 10 March 2016

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