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List of works by Nick Bushby

A modern approach to the synthesis of 2-(4-chlorophenyl)[2-(14)C]thiazol-4-ylacetic acid ([(14)C] fenclozic acid) and its acyl glucuronide metabolite.

scientific article published on 11 January 2013

Isotope labelling by reduction of nitriles: Application to the synthesis of isotopologues of tolmetin and celecoxib

scientific article

Minimal contribution of desmethyl-gefitinib, the major human plasma metabolite of gefitinib, to epidermal growth factor receptor (EGFR)-mediated tumour growth inhibition.

scientific article published on January 2006

Probe dependency in the determination of ligand binding kinetics at a prototypical G protein-coupled receptor.

scientific article published on 27 May 2019

Probing the mechanism of Prins cyclisations and application to the synthesis of 4-hydroxytetrahydropyrans

scientific article published on 16 June 2005

Route to Prolonged Residence Time at the Histamine H1 Receptor: Growing from Desloratadine to Rupatadine

scientific article published on 05 July 2019

Stereoselective synthesis of the tetrahydropyran core of polycarvernoside A

scientific article published on 01 June 2005

Synthesis of [(2)H6]ceftazidime as a stable isotopically labeled internal standard.

scientific article

Synthesis of [1,2-13C2, 15N]-L-homoserine and its incorporation by the PKS-NRPS system of Fusarium moniliforme into the mycotoxin fusarin C

scientific article published on 01 January 2007

[(14) C]-AZD1152 drug substance manufacture: challenges of an IV-infusion dosed human mass balance study in patients.

scientific article published in May 2016