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List of works by Kenzo Yamatsugu

A method for the synthesis of an oseltamivir PET tracer.

scientific article published on 28 November 2007

A synthesis of Tamiflu by using a barium-catalyzed asymmetric Diels-Alder-type reaction.

scientific article published in January 2009

Antibody mimetic drug conjugate manufactured by high-yield Escherichia coli expression and non-covalent binding system

scientific article published in 2022

Enantioselective synthesis of SM-130686 based on the development of asymmetric Cu(I)F catalysis to access 2-oxindoles containing a tetrasubstituted carbon.

scientific article published in May 2009

Fidelity and Promiscuity of a Mycobacterial Glycosyltransferase

scientific article

Intracellular activation of acetyl-CoA by an artificial reaction promoter and its fluorescent detection

scientific article published on April 11, 2013

Kinetic analyses and structure-activity relationship studies of synthetic lysine acetylation catalysts

scientific article published on 07 July 2018

LC-MS/MS-based quantitative study of the acyl group- and site-selectivity of human sirtuins to acylated nucleosomes

scientific article published on 8 February 2018

Leading approaches in synthetic epigenetics for novel therapeutic strategies.

scientific article published on 6 April 2018

Limited brain distribution of [3R,4R,5S]-4-acetamido-5-amino-3-(1-ethylpropoxy)-1-cyclohexene-1-carboxylate phosphate (Ro 64-0802), a pharmacologically active form of oseltamivir, by active efflux across the blood-brain barrier mediated by organic a

scientific article published on 24 November 2008

P-glycoprotein restricts the penetration of oseltamivir across the blood-brain barrier.

scientific article published on 26 November 2007

Site-Selective Synthetic Acylation of a Target Protein in Living Cells Promoted by a Chemical Catalyst/Donor System

scientific article published on 24 May 2019

Sulfanylmethyldimethylaminopyridine as a Useful Thiol Additive for Ligation Chemistry in Peptide/Protein Synthesis

scientific article published on 12 May 2020

Supramolecular Ligands for Histone Tails by Employing a Multivalent Display of Trisulfonated Calix[4]arenes.

scientific article

Synthetic Posttranslational Modifications: Chemical Catalyst-Driven Regioselective Histone Acylation of Native Chromatin

scientific article published on 23 May 2017

Two approaches toward the formal total synthesis of oseltamivir phosphate (Tamiflu): catalytic enantioselective three-component reaction strategy and L-glutamic acid strategy.

scientific article published on 21 March 2013