List of works - Jon Våbenø

A minimalistic 3D pharmacophore model for cyclopentapeptide CXCR4 antagonists

scientific article published on 01 January 2006

Conformational restrictions in ligand binding to the human intestinal di-/tripeptide transporter: implications for design of hPEPT1 targeted prodrugs

scientific article published on 01 March 2005

Design, synthesis, and biological evaluation of scaffold-based tripeptidomimetic antagonists for CXC chemokine receptor 4 (CXCR4).

scientific article published on 14 July 2014

Determination of the binding mode for the cyclopentapeptide CXCR4 antagonist FC131 using a dual approach of ligand modifications and receptor mutagenesis

scientific article published on December 2014

Development of a QSAR Model for Binding of Tripeptides and Tripeptidomimetics to the Human Intestinal Di-/Tripeptide Transporter hPEPT1

article

Diastereoselective reduction of a chiral N-Boc-protected delta-amino-alpha,beta-unsaturated gamma-keto ester Phe-Gly dipeptidomimetic.

scientific article

Dipeptidomimetic ketomethylene isosteres as pro-moieties for drug transport via the human intestinal di-/tripeptide transporter hPEPT1: design, synthesis, stability, and biological investigations

scientific article published on 01 September 2004

Experimental determination of drug diffusion coefficients in unstirred aqueous environments by temporally resolved concentration measurements.

scientific article published on 20 February 2018

Influence of chain length on the activity of tripeptidomimetic antagonists for CXC chemokine receptor 4 (CXCR4).

scientific article published on 21 November 2016

Inhibition of HIV fusion by small molecule agonists through efficacy-engineering of CXCR4.

scientific article published on 20 February 2018

Phe-Gly dipeptidomimetics designed for the di-/tripeptide transporters PEPT1 and PEPT2: synthesis and biological investigations.

scientific article published on February 2004

Probing the Molecular Interactions between CXC Chemokine Receptor 4 (CXCR4) and an Arginine-Based Tripeptidomimetic Antagonist (KRH-1636)

scientific article published on 02 October 2015

Progress toward rationally designed small-molecule peptide and peptidomimetic CXCR4 antagonists

scientific article published on July 2015

Rational design of conformationally constrained cyclopentapeptide antagonists for C-x-C chemokine receptor 4 (CXCR4)

scientific article published on 22 October 2012

Structure-activity relationship for alkylating dipeptide nitrogen mustard derivatives.