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List of works by Matjaz Brvar

Design, Synthesis, and Evaluation of Novel Tyrosine-Based DNA Gyrase B Inhibitors.

scientific article published on 16 June 2017

Discovery of 4,5,6,7-Tetrahydrobenzo[1,2-d]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site

scientific article published on 8 July 2015

Discovery of mono- and disubstituted 1H-pyrazolo[3,4]pyrimidines and 9H-purines as catalytic inhibitors of human DNA topoisomerase IIα.

scientific article published on 17 December 2014

Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors.

scientific article published on 22 February 2017

Discovery of the first inhibitors of bacterial enzyme D-aspartate ligase from Enterococcus faecium (Aslfm).

scientific article

In silico discovery and biophysical evaluation of novel 5-(2-hydroxybenzylidene) rhodanine inhibitors of DNA gyrase B

scientific article published on 03 March 2012

In silico discovery of 2-amino-4-(2,4-dihydroxyphenyl)thiazoles as novel inhibitors of DNA gyrase B.

scientific article published on 22 December 2009

Linker-switch approach towards new ATP binding site inhibitors of DNA gyrase B.

scientific article

Molecular Mechanism of Action for Allosteric Modulators and Agonists in CC-chemokine Receptor 5 (CCR5).

scientific article published on 10 November 2016

Monocyclic 4-amino-6-(phenylamino)-1,3,5-triazines as inhibitors of human DNA topoisomerase IIα

scientific article published on 22 October 2014

N-Phenyl-4,5-dibromopyrrolamides and N-Phenylindolamides as ATP Competitive DNA Gyrase B Inhibitors: Design, Synthesis, and Evaluation

scientific article

New N-phenyl-4,5-dibromopyrrolamides and N-Phenylindolamides as ATPase inhibitors of DNA gyrase.

scientific article

Receptor structure-based discovery of non-metabolite agonists for the succinate receptor GPR91.

scientific article published on 30 September 2017

Structure-Activity Investigations and Optimisations of Non-metabolite Agonists for the Succinate Receptor 1.

scientific article published on 3 July 2018

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