List of works - Ryo Yazaki

Amino Acid Schiff Base Bearing Benzophenone Imine As a Platform for Highly Congested Unnatural α-Amino Acid Synthesis

scientific article published on 22 April 2020

An Expeditious Route to trans-Configured Tetrahydrothiophenes Enabled by Fe(OTf)3 -Catalyzed [3+2] Cycloaddition of Donor-Acceptor Cyclopropanes with Thionoesters

scientific article published on 25 March 2018

Asymmetric synthesis of isothiazoles through Cu catalysis: direct catalytic asymmetric conjugate addition of allyl cyanide to α,β-unsaturated thioamides

scientific article published on 05 July 2011

Catalytic Aerobic Chemoselective α-Oxidation of Acylpyrazoles en Route to α-Hydroxy Acid Derivatives.

scientific article published on 30 May 2017

Catalytic Aerobic Cross-Dehydrogenative Coupling of Azlactones en Route to α,α-Disubstituted α-Amino Acids

scientific article published on 12 May 2020

Catalytic Chemoselective Conjugate Addition of Amino Alcohols to α,β-Unsaturated Ester: Hydroxy Group over Amino Group and Conjugate Addition over Transesterification

scientific article published on 01 January 2017

Chemo- and Regioselective Direct Functional Group Installation through Catalytic Hydroxy Group Selective Conjugate Addition of Amino Alcohols to α,β-Unsaturated Sulfonyl Compounds

scientific article published on 30 June 2016

Chemoselective Catalytic α-Oxidation of Carboxylic Acids: Iron/Alkali Metal Cooperative Redox Active Catalysis

scientific article published on 24 February 2020

Chemoselective catalytic conjugate addition of alcohols over amines

scientific article published on 22 January 2014

Concise enantioselective synthesis of duloxetine via direct catalytic asymmetric aldol reaction of thioamide.

scientific article published on 24 April 2012

Cooperative activation of alkyne and thioamide functionalities; direct catalytic asymmetric conjugate addition of terminal alkynes to α,β-unsaturated thioamides.

scientific article

Direct Catalytic Chemoselective α-Amination of Acylpyrazoles: A Concise Route to Unnatural α-Amino Acid Derivatives

scientific article published on 18 February 2016

Direct catalytic asymmetric Mannich-type reaction of thioamides.

scientific article published in January 2009

Direct catalytic asymmetric addition of allyl cyanide to ketones.

scientific article published in March 2009

Direct catalytic asymmetric addition of allylic cyanides to ketoimines.

scientific article

Direct catalytic asymmetric aldol reactions of thioamides: toward a stereocontrolled synthesis of 1,3-polyols.

scientific article published in December 2009

Direct catalytic asymmetric alkynylation of ketoimines

scientific article published on 18 January 2013

Direct catalytic asymmetric conjugate addition of terminal alkynes to alpha,beta-unsaturated thioamides.

scientific article published on August 2010

Direct catalytic asymmetric intramolecular conjugate addition of thioamide to α,β-unsaturated esters

scientific article published on 20 September 2011

Direct catalytic enantio- and diastereoselective aldol reaction of thioamides

scientific article published on 18 March 2011

Enantioselective synthesis of a GPR40 agonist AMG 837 via catalytic asymmetric conjugate addition of terminal alkyne to α,β-unsaturated thioamide

scientific article published on 03 February 2011

Growth Suppression of Human Colorectal Cancer Cells with Mutated KRAS by 3-Deaza-cytarabine in 3D Floating Culture

scientific article published on 01 July 2018

Intermediate as catalyst: catalytic asymmetric conjugate addition of nitroalkanes to α,β-unsaturated thioamides

scientific article published on 23 November 2011

Oxetanyl peptides: novel peptidomimetic modules for medicinal chemistry

scientific article

Strategy for Catalytic Chemoselective Cross-Enolate Coupling Reaction via a Transient Homocoupling Dimer

scientific article published on 31 May 2018

Toward the total synthesis of onchidin, a cytotoxic cyclic depsipeptide from a mollusc

scientific article published on 01 January 2007

μ-Oxo-Dinuclear-Iron(III)-Catalyzed O-Selective Acylation of Aliphatic and Aromatic Amino Alcohols and Transesterification of Tertiary Alcohols.

scientific article

List of works by Ryo Yazaki

Amino Acid Schiff Base Bearing Benzophenone Imine As a Platform for Highly Congested Unnatural α-Amino Acid Synthesis

An Expeditious Route to trans-Configured Tetrahydrothiophenes Enabled by Fe(OTf)3 -Catalyzed [3+2] Cycloaddition of Donor-Acceptor Cyclopropanes with Thionoesters

Asymmetric synthesis of isothiazoles through Cu catalysis: direct catalytic asymmetric conjugate addition of allyl cyanide to α,β-unsaturated thioamides

Catalytic Aerobic Chemoselective α-Oxidation of Acylpyrazoles en Route to α-Hydroxy Acid Derivatives.

Catalytic Aerobic Cross-Dehydrogenative Coupling of Azlactones en Route to α,α-Disubstituted α-Amino Acids

Catalytic Chemoselective Conjugate Addition of Amino Alcohols to α,β-Unsaturated Ester: Hydroxy Group over Amino Group and Conjugate Addition over Transesterification

Chemo- and Regioselective Direct Functional Group Installation through Catalytic Hydroxy Group Selective Conjugate Addition of Amino Alcohols to α,β-Unsaturated Sulfonyl Compounds

Chemoselective Catalytic α-Oxidation of Carboxylic Acids: Iron/Alkali Metal Cooperative Redox Active Catalysis

Chemoselective catalytic conjugate addition of alcohols over amines

Concise enantioselective synthesis of duloxetine via direct catalytic asymmetric aldol reaction of thioamide.

Cooperative activation of alkyne and thioamide functionalities; direct catalytic asymmetric conjugate addition of terminal alkynes to α,β-unsaturated thioamides.

Direct Catalytic Chemoselective α-Amination of Acylpyrazoles: A Concise Route to Unnatural α-Amino Acid Derivatives

Direct catalytic asymmetric Mannich-type reaction of thioamides.

Direct catalytic asymmetric addition of allyl cyanide to ketones.

Direct catalytic asymmetric addition of allylic cyanides to ketoimines.

Direct catalytic asymmetric aldol reactions of thioamides: toward a stereocontrolled synthesis of 1,3-polyols.

Direct catalytic asymmetric alkynylation of ketoimines

Direct catalytic asymmetric conjugate addition of terminal alkynes to alpha,beta-unsaturated thioamides.

Direct catalytic asymmetric intramolecular conjugate addition of thioamide to α,β-unsaturated esters

Direct catalytic enantio- and diastereoselective aldol reaction of thioamides

Enantioselective synthesis of a GPR40 agonist AMG 837 via catalytic asymmetric conjugate addition of terminal alkyne to α,β-unsaturated thioamide

Growth Suppression of Human Colorectal Cancer Cells with Mutated KRAS by 3-Deaza-cytarabine in 3D Floating Culture

Intermediate as catalyst: catalytic asymmetric conjugate addition of nitroalkanes to α,β-unsaturated thioamides

Oxetanyl peptides: novel peptidomimetic modules for medicinal chemistry

Strategy for Catalytic Chemoselective Cross-Enolate Coupling Reaction via a Transient Homocoupling Dimer

Toward the total synthesis of onchidin, a cytotoxic cyclic depsipeptide from a mollusc

μ-Oxo-Dinuclear-Iron(III)-Catalyzed O-Selective Acylation of Aliphatic and Aromatic Amino Alcohols and Transesterification of Tertiary Alcohols.