Search filters

List of works by Steven Verhelst

4-Bromophenacyl bromide specifically inhibits rhoptry secretion during Toxoplasma invasion

scientific article

A General Solid Phase Method for the Preparation of Diverse Azapeptide Probes Directed Against Cysteine Proteases

scientific article published on 01 December 2005

A Mild Chemically Cleavable Linker System for Functional Proteomic Applications

scientific article published on 01 January 2007

A Substrate-Inspired Probe Monitors Translocation, Activation, and Subcellular Targeting of Bacterial Type III Effector Protease AvrPphB

scientific article published on 01 February 2013

A selective activity-based probe for the papain family cysteine protease dipeptidyl peptidase I/cathepsin C.

scientific article published on May 2006

A simple and effective cleavable linker for chemical proteomics applications

scientific article published on October 2012

A stereoselective route towards highly functionalized 4,6-diaminocyclohexene derivatives

ATP13A3 is a major component of the enigmatic mammalian polyamine transport system

scientific article published on 11 December 2020

Activity-Based Protein Profiling of Rhomboid Proteases in Liposomes

scientific article published on 19 June 2015

Activity-Based Protein Profiling of Serine Proteases in Immune Cells

scientific article published on 19 August 2020

Activity-based probes for rhomboid proteases discovered in a mass spectrometry-based assay

scientific article

Activity-based probes for the study of proteases: recent advances and developments.

scientific article published on 19 March 2012

Alkyne derivatives of isocoumarins as clickable activity-based probes for serine proteases.

scientific article

Bioorthogonal Reactions in Activity-Based Protein Profiling

scientific article published on 18 December 2020

Chemical Tools for the Study of Intramembrane Proteases

scientific article published on 16 October 2015

Cleavable trifunctional biotin reagents for protein labelling, capture and release.

scientific article published in June 2013

Clickable polyamine derivatives as chemical probes for the polyamine transport system

scientific article published on 16 February 2018

Comparative analysis of click chemistry mediated activity-based protein profiling in cell lysates.

scientific article published on 11 October 2013

Design and synthesis of a protein:Farnesyltransferase inhibitor based on sugar amino acids

article by Herman S Overkleeft et al published May 1999 in Tetrahedron Letters

Detection of protease activity in cells and animals.

scientific article published on 07 May 2015

Development of calpain-specific inactivators by screening of positional scanning epoxide libraries

scientific article

Discovery of Cellular Roles of Intramembrane Proteases

scientific article published on 24 July 2019

Inhibitor Fingerprinting of Rhomboid Proteases by Activity-Based Protein Profiling Reveals Inhibitor Selectivity and Rhomboid Autoprocessing

scientific article published on 28 July 2015

Inhibitors of rhomboid proteases

scientific article published on 10 July 2015

Kinase Photoaffinity Labeling Reveals Low Selectivity Profile of the IRE1 Targeting Imidazopyrazine-Based KIRA6 Inhibitor

scientific article published on 08 December 2020

Minitags for small molecules: detecting targets of reactive small molecules in living plant tissues using 'click chemistry'.

scientific article

Mixed alkyl aryl phosphonate esters as quenched fluorescent activity-based probes for serine proteases

scientific article published in February 2015

Probing Functional Tyrosines ⬇️

scientific article published on April 18, 2013

Protease Specificity Profiling in a Pipet Tip Using "Charge-Synchronized" Proteome-Derived Peptide Libraries.

scientific article published on 17 April 2018

Role for cathepsin F in invariant chain processing and major histocompatibility complex class II peptide loading by macrophages

scientific article

Short Peptides with Uncleavable Peptide Bond Mimetics as Photoactivatable Caspase-3 Inhibitors

scientific article published on 08 January 2019

Solid-phase methods for the preparation of epoxysuccinate-based inhibitors of cysteine proteases.

scientific article published in November 2006

Solid-phase synthesis of double-headed epoxysuccinyl activity-based probes for selective targeting of papain family cysteine proteases.

scientific article

Specificity of aza-peptide electrophile activity-based probes of caspases

scientific article published on 15 December 2006

Stress-induced inflammation evoked by immunogenic cell death is blunted by the IRE1α kinase inhibitor KIRA6 through HSP60 targeting

scientific article published on 27 August 2021

Surface plasmon resonance evaluation of various aminoglycoside-RNA hairpin interactions reveals low degree of selectivity.

scientific article published in July 2004

Synthesis of orthogonally protected 2-deoxystreptamine stereoisomers

Tagging and detection strategies for activity-based proteomics.

scientific article published on 13 December 2006

Target profiling of 4-hydroxyderricin in S. aureus reveals seryl-tRNA synthetase binding and inhibition by covalent modification.

scientific article published on 8 January 2013

The structural basis for catalysis and substrate specificity of a rhomboid protease

scientific article

Tuning activity-based probe selectivity for serine proteases by on-resin 'click' construction of peptide diphenyl phosphonates.

scientific article

Tuning probe selectivity for chemical proteomics applications ⬇️

scientific article published on December 28, 2012

Paulina is supported by:

About Paulina

Help