List of works - Andrzej Orzeszko

Benzimidazole inhibitors of protein kinase CK2 potently inhibit the activity of atypical protein kinase Rio1

scientific article published on December 2016

CK2α and CK2α' subunits differ in their sensitivity to 4,5,6,7-tetrabromo- and 4,5,6,7-tetraiodo-1H-benzimidazole derivatives

scientific article published on 13 November 2011

Cell-permeable dual inhibitors of protein kinases CK2 and PIM-1: structural features and pharmacological potential

scientific article

Deoxynucleosides with benzimidazoles as aglycone moiety are potent anticancer agents.

scientific article

Exploiting the repertoire of CK2 inhibitors to target DYRK and PIM kinases.

scientific article

In Search of the Antimicrobial Potential of Benzimidazole Derivatives.

scientific article published in August 2016

Modified tetrahalogenated benzimidazoles with CK2 inhibitory activity are active against human prostate cancer cells LNCaP in vitro ⬇️

scientific article published on May 24, 2012

Novel adamantylated pyrimidines and their preliminary biological evaluations.

scientific article

Quantum-chemical insight into structure-reactivity relationship in 4,5,6,7-tetrahalogeno-1H-benzimidazoles: a combined X-ray, DSC, DFT/QTAIM, Hirshfeld surface-based, and molecular docking approach.

scientific article published on 5 March 2014

Structural study of selected polyhalogenated benzimidazoles (protein kinase CK2 inhibitors) by nuclear quadrupole double resonance, X-ray, and density functional theory

scientific article published in January 2010

Synthesis and anti-HIV studies of 2- and 3-adamantyl-substituted thiazolidin-4-ones

scientific article published on 10 March 2008

Synthesis and anti-HIV studies of 2-adamantyl-substituted thiazolidin-4-ones

scientific article published on 20 January 2007

Synthesis and antibacterial activity of 5-adamantan-1-yl-methyl analogues of trimethoprim

scientific article published on 01 September 2006

Synthesis and antibacterial activity of adamantyl substituted pyrimidines

scientific article published in November 2004

Synthesis and antimicrobial activity of new adamantane derivatives III.

scientific article published in August 2002

Synthesis and antimycobacterial activity of selected nitrobenzyloxylated benzotriazoles.

scientific article published in July 2008

Synthesis and antiviral activity of some 5'-N-phthaloyl-3'-azido-2',3'-dideoxythymidine analogues

scientific article published in May 2003

Synthesis and proapoptotic properties of new casein kinase II inhibitors

scientific article published on November 1, 2010

Synthesis of new analogs of benzotriazole, benzimidazole and phthalimide--potential inhibitors of human protein kinase CK2.

scientific article published on 7 January 2009

Tetraiodobenzimidazoles are potent inhibitors of protein kinase CK2.

scientific article published on 27 August 2009

The Electrochemical Behavior of Bunte Salts

The selectivity of inhibitors of protein kinase CK2: an update

scientific article

Tumor necrosis factor-alpha production-regulating activity of phthalimide derivatives in genetically modified murine melanoma cells B78H1.

scientific article published in May 2003

List of works by Andrzej Orzeszko

Benzimidazole inhibitors of protein kinase CK2 potently inhibit the activity of atypical protein kinase Rio1

CK2α and CK2α' subunits differ in their sensitivity to 4,5,6,7-tetrabromo- and 4,5,6,7-tetraiodo-1H-benzimidazole derivatives

Cell-permeable dual inhibitors of protein kinases CK2 and PIM-1: structural features and pharmacological potential

Deoxynucleosides with benzimidazoles as aglycone moiety are potent anticancer agents.

Exploiting the repertoire of CK2 inhibitors to target DYRK and PIM kinases.

In Search of the Antimicrobial Potential of Benzimidazole Derivatives.

Modified tetrahalogenated benzimidazoles with CK2 inhibitory activity are active against human prostate cancer cells LNCaP in vitro ⬇️

Novel adamantylated pyrimidines and their preliminary biological evaluations.

Quantum-chemical insight into structure-reactivity relationship in 4,5,6,7-tetrahalogeno-1H-benzimidazoles: a combined X-ray, DSC, DFT/QTAIM, Hirshfeld surface-based, and molecular docking approach.

Structural study of selected polyhalogenated benzimidazoles (protein kinase CK2 inhibitors) by nuclear quadrupole double resonance, X-ray, and density functional theory

Synthesis and anti-HIV studies of 2- and 3-adamantyl-substituted thiazolidin-4-ones

Synthesis and anti-HIV studies of 2-adamantyl-substituted thiazolidin-4-ones

Synthesis and antibacterial activity of 5-adamantan-1-yl-methyl analogues of trimethoprim

Synthesis and antibacterial activity of adamantyl substituted pyrimidines

Synthesis and antimicrobial activity of new adamantane derivatives III.

Synthesis and antimycobacterial activity of selected nitrobenzyloxylated benzotriazoles.

Synthesis and antiviral activity of some 5'-N-phthaloyl-3'-azido-2',3'-dideoxythymidine analogues

Synthesis and proapoptotic properties of new casein kinase II inhibitors

Synthesis of new analogs of benzotriazole, benzimidazole and phthalimide--potential inhibitors of human protein kinase CK2.

Tetraiodobenzimidazoles are potent inhibitors of protein kinase CK2.

The Electrochemical Behavior of Bunte Salts

The selectivity of inhibitors of protein kinase CK2: an update

Tumor necrosis factor-alpha production-regulating activity of phthalimide derivatives in genetically modified murine melanoma cells B78H1.