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List of works by Jiří Kuneš

2-(3-Methoxyphenyl)quinazoline Derivatives: A New Class of Direct Constitutive Androstane Receptor (CAR) Agonists.

scientific article published on 4 May 2016

3-Benzyl-2H-1,3-benzoxazine-2,4(3H)-diones, a new group of antimycobacterial compounds against potentially pathogenic strains.

scientific article published in November 2003

3-Substituted N-Benzylpyrazine-2-carboxamide Derivatives: Synthesis, Antimycobacterial and Antibacterial Evaluation

scientific article published on 21 March 2017

A New Insight into the Stereoelectronic Control of the Pd0 -Catalyzed Allylic Substitution: Application for the Synthesis of Multisubstituted Pyran-2-ones via an Unusual 1,3-Transposition

scientific article published on 09 May 2019

A note to the biological activity of benzoxazine derivatives containing the thioxo group.

scientific article published on 20 February 2010

Alkaloids from Zephyranthes robusta BAKER and their acetylcholinesterase- and butyrylcholinesterase-inhibitory activity.

scientific article published in June 2013

Alkylamino derivatives of pyrazinamide: synthesis and antimycobacterial evaluation

scientific article published on 19 December 2013

Analytical power of LLE-HPLC-PDA-MS/MS in drug metabolism studies: identification of new nabumetone metabolites.

scientific article published on 19 March 2013

Antifungal 3,5-disubstituted furanones: From 5-acyloxymethyl to 5-alkylidene derivatives.

scientific article

Antimycobacterial N-pyridinylsalicylamides, isosters of salicylamides.

scientific article

Antimycobacterial and antifungal isosters of salicylamides.

scientific article published in August 2003

Aromatic Esters of the Crinane Amaryllidaceae Alkaloid Ambelline as Selective Inhibitors of Butyrylcholinesterase

scientific article published on 20 April 2020

Azaphthalocyanines with fused triazolo rings: formation of sterically stressed constitutional isomers

scientific article published on 23 March 2012

Azole antimycotics differentially affect rifampicin-induced pregnane X receptor-mediated CYP3A4 gene expression.

scientific article published on 12 November 2007

Cholinesterase and Prolyl Oligopeptidase Inhibitory Activities of Alkaloids from Argemone platyceras (Papaveraceae).

scientific article published on 14 July 2017

Design, Synthesis, Antimycobacterial Evaluation, and In Silico Studies of 3-(Phenylcarbamoyl)-pyrazine-2-carboxylic Acids.

scientific article

Design, Synthesis, and Biological Evaluation of Isothiosemicarbazones with Antimycobacterial Activity

scientific article

Design, synthesis and anti-mycobacterial evaluation of some new N-phenylpyrazine-2-carboxamides

Design, synthesis and antimycobacterial activity of hybrid molecules combining pyrazinamide with a 4-phenylthiazol-2-amine scaffold

scientific article published on 22 February 2018

Determination of muscle relaxants pancuronium and vecuronium bromide by capillary electrophoresis with capacitively coupled contactless conductivity detection

scientific article published on 10 March 2011

Disposition study of a new potential antineoplastic agent dimefluron in rats using high-performance liquid chromatography with ultraviolet and mass spectrometric detection.

scientific article published in April 2005

Evaluation of natural antioxidants of Leuzea carthamoides as a result of a screening study of 88 plant extracts from the European Asteraceae and Cichoriaceae

scientific article published on 01 April 2008

Evaluation of natural substances from Evolvulus alsinoides L. with the purpose of determining their antioxidant potency

scientific article published on 01 August 2008

Fully substituted pyranones via quasi-heterogeneous genuinely ligand-free Migita-Stille coupling of iodoacrylates

scientific article published on 23 January 2015

Heterocyclic isosters of antimycobacterial salicylanilides.

scientific article

High-performance liquid chromatographic determination of tramadol and its O-desmethylated metabolite in blood plasma. Application to a bioequivalence study in humans

scientific article

Highly active antimycobacterial derivatives of benzoxazine.

scientific article published on 19 October 2010

Identification and characterization of thiosemicarbazones with antifungal and antitumor effects: cellular iron chelation mediating cytotoxic activity.

scientific article published on 13 August 2008

Isoquinoline Alkaloids from Fumaria officinalis L. and Their Biological Activities Related to Alzheimer's Disease.

scientific article

Metabolic profiling of a potential antifungal drug, 3-(4-bromophenyl)-5-acetoxymethyl-2,5-dihydrofuran-2-one, in mouse urine using high-performance liquid chromatography with UV photodiode-array and mass spectrometric detection.

scientific article

N-benzylsalicylthioamides: highly active potential antituberculotics.

scientific article

N-substituted 5-amino-6-methylpyrazine-2,3-dicarbonitriles: microwave-assisted synthesis and biological properties.

scientific article

Neighboring group effect in Pd-catalyzed carbonylation terminated by lactonization: a need for a protective group and/or DMF.

scientific article published in October 2004

New antioxidant flavonoid isolated from Leuzea carthamoides.

scientific article published in February 2010

New potentially active pyrazinamide derivatives synthesized under microwave conditions.

scientific article published on 3 July 2014

Novel Halogenated Pyrazine-Based Chalcones as Potential Antimicrobial Drugs

scientific article published on 27 October 2016

Novel bronchodilatory quinazolines and quinoxalines: synthesis and biological evaluation.

scientific article published on 2 January 2014

Novel pyrazine analogs of chalcones: synthesis and evaluation of their antifungal and antimycobacterial activity.

scientific article published on 12 January 2015

On the relationship between the substitution pattern of thiobenzanilides and their antimycobacterial activity.

scientific article published in September 2002

Quinaldine derivatives: preparation and biological activity

scientific article published on 01 November 2005

Quinazoline derivatives with antitubercular activity

scientific article

Scalable Synthesis of Human Ultralong Chain Ceramides

scientific article published on 19 October 2015

Substituted 5-aroylpyrazine-2-carboxylic acid derivatives: synthesis and biological activity.

scientific article published in November 2003

Synthesis and Antifungal Screening of 2-{[1-(5-Alkyl/arylalkylpyrazin-2-yl)ethylidene]hydrazono}-1,3-thiazolidin-4-ones.

scientific article published on 23 November 2016

Synthesis and Antimicrobial Evaluation of 6-Alkylamino-N-phenylpyrazine-2-carboxamides

scientific article

Synthesis and Biological Activity of Quaternary Ammonium Salt-Type Agents Containing Cholesterol and Terpenes

scientific article published on 24 March 2014

Synthesis and Biological Evaluation of N-Alkyl-3-(alkylamino)-pyrazine-2-carboxamides.

scientific article published on 14 May 2015

Synthesis and antimicrobial evaluation of new 2-substituted 5,7-di-tert-butylbenzoxazoles.

scientific article published on 19 June 2006

Synthesis and antimycobacterial evaluation of N-substituted 3-aminopyrazine-2,5-dicarbonitriles.

scientific article

Synthesis and antimycobacterial evaluation of N-substituted 5-chloropyrazine-2-carboxamides

scientific article published on 21 April 2013

Synthesis and antimycobacterial evaluation of pyrazinamide derivatives with benzylamino substitution.

scientific article published on 27 November 2012

Synthesis and antimycobacterial evaluation of substituted pyrazinecarboxamides

scientific article published in May 2008

Synthesis and antimycobacterial properties of N-substituted 6-amino-5-cyanopyrazine-2-carboxamides.

scientific article published on January 2011

Synthesis and biological activity of desmethoxy analogues of coruscanone A.

scientific article

Synthesis and characterization of (Z)-5-arylmethylidene-rhodanines with photosynthesis-inhibiting properties.

scientific article published on 22 June 2011

Synthesis and in vitro antifungal activity of 4-substituted phenylguanidinium salts.

scientific article

Synthesis and structure-antifungal activity relationships of 3-aryl-5-alkyl-2,5-dihydrofuran-2-ones and their carbanalogues: further refinement of tentative pharmacophore group.

scientific article

Synthesis of (2E)-2-methyl-3-(4-([4-(quinolin-2-ylmethoxy)phenyl]sulfanyl)phenyl)prop-2-enoic acid (VUFB 20609) and 2-methyl-3-(4-([4-(quinolin-2-ylmethoxy)phenyl]sulfanyl)phenyl)propanoic acid (VUFB 20584) as potential antileukotrienic agents.

scientific article published on June 2004

Synthesis, antimycobacterial activity and in vitro cytotoxicity of 5-chloro-N-phenylpyrazine-2-carboxamides.

scientific article published on 2 December 2013

Synthesis, antimycobacterial, antifungal and photosynthesis-inhibiting activity of chlorinated N-phenylpyrazine-2-carboxamides.

scientific article published on 26 November 2010

TFP as a ligand in Au(i)-catalyzed dihydropyran synthesis. Unprecedented rearrangement of dihydropyrans into cyclopentenones ⬇️

scientific article published on July 18, 2011

The oriented development of antituberculotics (Part II): halogenated 3-(4-alkylphenyl)-1,3-benzoxazine-2,4-(3H)-diones

scientific article published on 01 May 2007

The oriented development of antituberculotics: salicylanilides

scientific article published on 01 November 2006

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