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List of works by Nicolas Primas

2-Phenoxy-3-Trichloromethylquinoxalines Are Antiplasmodial Derivatives with Activity against the Apicoplast of

scientific article published on 26 July 2021

8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a]pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductases

scientific article published on 01 August 2018

A new synthetic route to original sulfonamide derivatives in 2-trichloromethylquinazoline series: a structure-activity relationship study of antiplasmodial activity.

scientific article

Cross-Coupling Synthesis of Methylallyl Alkenes: Scope Extension and Mechanistic Study

scientific article published on 21 December 2015

Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold.

scientific article published on 10 September 2016

Looking for new antiplasmodial quinazolines: DMAP-catalyzed synthesis of 4-benzyloxy- and 4-aryloxy-2-trichloromethylquinazolines and their in vitro evaluation toward Plasmodium falciparum

scientific article published on 28 April 2016

New series of monoamidoxime derivatives displaying versatile antiparasitic activity.

scientific article published on 30 September 2014

Nongenotoxic 3-Nitroimidazo[1,2-]pyridines Are NTR1 Substrates That Display Potent Antileishmanial Activity

scientific article published on 19 December 2018

Plasmodial Kinase Inhibitors Targeting Malaria: Recent Developments

scientific article published on 15 December 2020

Stability studies of five anti-infectious eye drops under exhaustive storage conditions.

scientific article published in December 2017

Synthesis and in vitro evaluation of 4-trichloromethylpyrrolo[1,2-a]quinoxalines as new antiplasmodial agents.

scientific article published on 10 June 2014