List of works - Antonella Di Pizio

A bioinspired in vitro bioelectronic tongue with human T2R38 receptor for high-specificity detection of N-C=S-containing compounds

scientific article published on 06 February 2019

Ac-tLeu-Asp-H is the minimal and highly effective human caspase-3 inhibitor: biological and in silico studies

scientific article

Allostery in Its Many Disguises: From Theory to Applications

scientific article published on 07 February 2019

Amino Acid derivatives as new zinc binding groups for the design of selective matrix metalloproteinase inhibitors.

scientific article

An integrated computational approach to rationalize the activity of non-zinc-binding MMP-2 inhibitors

scientific article

Astringent Gallic Acid in Red Wine Regulates Mechanisms of Gastric Acid Secretion via Activation of Bitter Taste Sensing Receptor TAS2R4

scientific article published in 2021

Beyond the Flavour: The Potential Druggability of Chemosensory G Protein-Coupled Receptors ⬇️

scientific article published on 20 March 2019

Bitter and sweet tasting molecules: It's complicated

scientific article published on 19 April 2018

BitterDB: taste ligands and receptors database in 2019

article

Bitterless Guaifenesin Prodrugs - Design, Synthesis, Characterization, In Vitro Kinetics and Bitterness Studies

scientific article published on 02 November 2018

Bone-Seeking Matrix Metalloproteinase Inhibitors for the Treatment of Skeletal Malignancy

scientific article published on 01 June 2020

Catechol-based matrix metalloproteinase inhibitors with additional antioxidative activity.

scientific article published on 24 August 2016

Comparing Class A GPCRs to bitter taste receptors: Structural motifs, ligand interactions and agonist-to-antagonist ratios.

scientific article

From Cell to Beak: In-Vitro and In-Vivo Characterization of Chicken Bitter Taste Thresholds.

scientific article

In Silico Investigation of Bitter Hop-Derived Compounds and Their Cognate Bitter Taste Receptors

scientific article published on 13 February 2020

In Silico Molecular Study of Tryptophan Bitterness

scientific article published on 11 October 2020

Independent Evolution of Strychnine Recognition by Bitter Taste Receptor Subtypes.

scientific article published on 2 March 2018

Insights into the Selectivity Mechanisms of Grapevine NIP Aquaporins

scientific article published on 13 September 2020

Ligand binding modes from low resolution GPCR models and mutagenesis: chicken bitter taste receptor as a test-case.

scientific article published on 15 August 2017

Malaria parasites both repress host CXCL10 and use it as a cue for growth acceleration

scientific article published on 11 August 2021

Molecular Features Underlying Selectivity in Chicken Bitter Taste Receptors

scientific article published on 31 January 2018

More than smell. COVID-19 is associated with severe impairment of smell, taste, and chemesthesis

scientific article published on 08 May 2020

Non-Zinc-Binding Inhibitors of MMP-13: GRID-Based Approaches to Rationalize the Binding Process.

scientific article published on 13 August 2015

Numerous Compounds Orchestrate Coffee’s Bitterness

scientific article published on 21 May 2020

Probing the Binding Pocket of the Broadly Tuned Human Bitter Taste Receptor TAS2R14 by Chemical Modification of Cognate Agonists

scientific article published on 17 February 2016

Probing the S1' site for the identification of non-zinc-binding MMP-2 inhibitors.

scientific article

Promiscuity and selectivity of bitter molecules and their receptors

scientific article published on 16 April 2015

RASA2 and NF1; two-negative regulators of Ras with complementary functions in melanoma

scientific article published on 26 November 2018

RGS7 is recurrently mutated in melanoma and promotes migration and invasion of human cancer cells

scientific article published on 12 January 2018

Rational design of agonists for bitter taste receptor TAS2R14: from modeling to bench and back

scientific article published on 24 June 2019

Recent smell loss is the best predictor of COVID-19: a preregistered, cross-sectional study

scientific article published on 26 July 2020

Recurrent inactivating RASA2 mutations in melanoma

scientific article published on 26 October 2015

Reengineering the ligand sensitivity of the broadly tuned human bitter taste receptor TAS2R14

scientific article published on 19 July 2018

List of works by Antonella Di Pizio

A bioinspired in vitro bioelectronic tongue with human T2R38 receptor for high-specificity detection of N-C=S-containing compounds

Ac-tLeu-Asp-H is the minimal and highly effective human caspase-3 inhibitor: biological and in silico studies

Allostery in Its Many Disguises: From Theory to Applications

Amino Acid derivatives as new zinc binding groups for the design of selective matrix metalloproteinase inhibitors.

An integrated computational approach to rationalize the activity of non-zinc-binding MMP-2 inhibitors

Astringent Gallic Acid in Red Wine Regulates Mechanisms of Gastric Acid Secretion via Activation of Bitter Taste Sensing Receptor TAS2R4

Beyond the Flavour: The Potential Druggability of Chemosensory G Protein-Coupled Receptors ⬇️

Bitter and sweet tasting molecules: It's complicated

BitterDB: taste ligands and receptors database in 2019

Bitterless Guaifenesin Prodrugs - Design, Synthesis, Characterization, In Vitro Kinetics and Bitterness Studies

Bone-Seeking Matrix Metalloproteinase Inhibitors for the Treatment of Skeletal Malignancy

Catechol-based matrix metalloproteinase inhibitors with additional antioxidative activity.

Comparing Class A GPCRs to bitter taste receptors: Structural motifs, ligand interactions and agonist-to-antagonist ratios.

From Cell to Beak: In-Vitro and In-Vivo Characterization of Chicken Bitter Taste Thresholds.

In Silico Investigation of Bitter Hop-Derived Compounds and Their Cognate Bitter Taste Receptors

In Silico Molecular Study of Tryptophan Bitterness

Independent Evolution of Strychnine Recognition by Bitter Taste Receptor Subtypes.

Insights into the Selectivity Mechanisms of Grapevine NIP Aquaporins

Ligand binding modes from low resolution GPCR models and mutagenesis: chicken bitter taste receptor as a test-case.

Malaria parasites both repress host CXCL10 and use it as a cue for growth acceleration

Molecular Features Underlying Selectivity in Chicken Bitter Taste Receptors

More than smell. COVID-19 is associated with severe impairment of smell, taste, and chemesthesis

Non-Zinc-Binding Inhibitors of MMP-13: GRID-Based Approaches to Rationalize the Binding Process.

Numerous Compounds Orchestrate Coffee’s Bitterness

Probing the Binding Pocket of the Broadly Tuned Human Bitter Taste Receptor TAS2R14 by Chemical Modification of Cognate Agonists

Probing the S1' site for the identification of non-zinc-binding MMP-2 inhibitors.

Promiscuity and selectivity of bitter molecules and their receptors

RASA2 and NF1; two-negative regulators of Ras with complementary functions in melanoma

RGS7 is recurrently mutated in melanoma and promotes migration and invasion of human cancer cells

Rational design of agonists for bitter taste receptor TAS2R14: from modeling to bench and back

Recent smell loss is the best predictor of COVID-19: a preregistered, cross-sectional study

Recurrent inactivating RASA2 mutations in melanoma

Reengineering the ligand sensitivity of the broadly tuned human bitter taste receptor TAS2R14