List of works - Yuka Unno

Acinetobacter baumannii Lipopolysaccharide Influences Adipokine Expression in 3T3-L1 Adipocytes.

scientific article

Advanced glycation end products-modified proteins and oxidized LDL mediate down-regulation of leptin in mouse adipocytes via CD36.

scientific article published on December 2004

Design and synthesis of the stabilized analogs of belactosin A with the unnatural cis-cyclopropane structure.

scientific article published on 29 August 2013

Development of a new class of proteasome inhibitors with an epoxyketone warhead: Rational hybridization of non-peptidic belactosin derivatives and peptide epoxyketones

scientific article published on 24 April 2014

Glycolaldehyde-modified bovine serum albumin downregulates leptin expression in mouse adipocytes via a CD36-mediated pathway.

scientific article published on June 2005

Identification of a small-molecule inhibitor of the interaction between Survivin and Smac/DIABLO.

scientific article

Identification of novel kynurenine production-inhibiting benzenesulfonamide derivatives in cancer cells ⬇️

scientific article published on February 17, 2012

Investigation of the noncovalent binding mode of covalent proteasome inhibitors around the transition state by combined use of cyclopropylic strain-based conformational restriction and computational modeling.

scientific article published on 9 July 2013

Pathological roles of advanced glycation end product receptors SR-A and CD36.

scientific article published on June 2005

Peroxynitrite induces formation of N( epsilon )-(carboxymethyl) lysine by the cleavage of Amadori product and generation of glucosone and glyoxal from glucose: novel pathways for protein modification by peroxynitrite.

scientific article published in September 2002

Potent proteasome inhibitors derived from the unnatural cis-cyclopropane isomer of Belactosin A: synthesis, biological activity, and mode of action

scientific article

Rational hopping of a peptidic scaffold into non-peptidic scaffolds: structurally novel potent proteasome inhibitors derived from a natural product, belactosin A

scientific article published on 22 January 2014

Resolvin E1, but not resolvins E2 and E3, promotes fMLF-induced ROS generation in human neutrophils

scientific article published on 13 August 2018

S-benzylisothiourea derivatives as small-molecule inhibitors of indoleamine-2,3-dioxygenase.

scientific article published on 11 July 2010

Structurally novel highly potent proteasome inhibitors created by the structure-based hybridization of nonpeptidic belactosin derivatives and peptide boronates.

scientific article published on 25 February 2014

Synthesis of 2,3- and 3,4-methanoamino acid equivalents with stereochemical diversity and their conversion into the tripeptide proteasome inhibitor belactosin a and its highly potent cis-cyclopropane stereoisomer

scientific article published on 19 July 2008

Three-dimensional structure-activity relationship study of belactosin A and its stereo- and regioisomers: development of potent proteasome inhibitors by a stereochemical diversity-oriented strategy.

scientific article published on 12 March 2009

Virulence characteristics of Acinetobacter baumannii clinical isolates vary with the expression levels of omps.

scientific article

List of works by Yuka Unno

Acinetobacter baumannii Lipopolysaccharide Influences Adipokine Expression in 3T3-L1 Adipocytes.

Advanced glycation end products-modified proteins and oxidized LDL mediate down-regulation of leptin in mouse adipocytes via CD36.

Design and synthesis of the stabilized analogs of belactosin A with the unnatural cis-cyclopropane structure.

Development of a new class of proteasome inhibitors with an epoxyketone warhead: Rational hybridization of non-peptidic belactosin derivatives and peptide epoxyketones

Glycolaldehyde-modified bovine serum albumin downregulates leptin expression in mouse adipocytes via a CD36-mediated pathway.

Identification of a small-molecule inhibitor of the interaction between Survivin and Smac/DIABLO.

Identification of novel kynurenine production-inhibiting benzenesulfonamide derivatives in cancer cells ⬇️

Investigation of the noncovalent binding mode of covalent proteasome inhibitors around the transition state by combined use of cyclopropylic strain-based conformational restriction and computational modeling.

Pathological roles of advanced glycation end product receptors SR-A and CD36.

Peroxynitrite induces formation of N( epsilon )-(carboxymethyl) lysine by the cleavage of Amadori product and generation of glucosone and glyoxal from glucose: novel pathways for protein modification by peroxynitrite.

Potent proteasome inhibitors derived from the unnatural cis-cyclopropane isomer of Belactosin A: synthesis, biological activity, and mode of action

Rational hopping of a peptidic scaffold into non-peptidic scaffolds: structurally novel potent proteasome inhibitors derived from a natural product, belactosin A

Resolvin E1, but not resolvins E2 and E3, promotes fMLF-induced ROS generation in human neutrophils

S-benzylisothiourea derivatives as small-molecule inhibitors of indoleamine-2,3-dioxygenase.

Structurally novel highly potent proteasome inhibitors created by the structure-based hybridization of nonpeptidic belactosin derivatives and peptide boronates.

Synthesis of 2,3- and 3,4-methanoamino acid equivalents with stereochemical diversity and their conversion into the tripeptide proteasome inhibitor belactosin a and its highly potent cis-cyclopropane stereoisomer

Three-dimensional structure-activity relationship study of belactosin A and its stereo- and regioisomers: development of potent proteasome inhibitors by a stereochemical diversity-oriented strategy.

Virulence characteristics of Acinetobacter baumannii clinical isolates vary with the expression levels of omps.