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List of works by Peter R Bernstein

A novel series of selective leukotriene antagonists: exploration and optimization of the acidic region in 1,6-disubstituted indoles and indazoles

scientific article published on 01 September 1990

Aerosolized leukotriene D4 converts monkeys that are negative aerosolized ascaris responders to positive airway responders

scientific article published on 01 March 1986

Azepines and piperidines with dual norepinephrine dopamine uptake inhibition and antidepressant activity

scientific article published on 12 November 2012

Calculation and application of activity discriminants in lead optimization.

scientific article published on 30 July 2010

Chemically stable homocinnamyl analogues of the leukotrienes: synthesis and preliminary biological evaluation

scientific article published on 01 December 1986

Comparative potency and pharmacology of isomers of leukotriene D4 on guinea-pig trachea: requirement for a 5(S)6(R) configuration

scientific article published on 01 April 1982

Correction to "Discovery of 6-Phenylhexanamide Derivatives as Potent Stereoselective Mitofusin Activators for the Treatment of Mitochondrial Diseases"

scientific article published on 21 August 2020

De novo design of a picomolar nonbasic 5-HT(1B) receptor antagonist

scientific article

Design of orally active, non-peptidic inhibitors of human leukocyte elastase

scientific article published on 01 April 1994

Design, synthesis, and SAR of tachykinin antagonists: modulation of balance in NK(1)/NK(2) receptor antagonist activity.

scientific article published in August 2002

Determination of SRS-A release from guinea-pig lungs by a radioimmunoassay

scientific article published on 01 December 1983

Discovery of a Potent and Selective PI3Kδ Inhibitor (<i>S</i>)-2,4-Diamino-6-((1-(7-fluoro-1-(4-fluorophenyl)-4-oxo-3-phenyl-4<i>H</i>-quinolizin-2-yl)ethyl)amino)pyrimidine-5-carbonitrile with Improved Pharmacokinetic Profile and Superior Efficacy

scientific article published on 01 December 2020

Discovery of spirofused piperazine and diazepane amides as selective histamine-3 antagonists with in vivo efficacy in a mouse model of cognition.

scientific article published on 27 January 2014

Effect of inhaled leukotriene D4 on human airways

scientific article published on 01 January 1988

Effect of trifluoromethyl ketone-based elastase inhibitors on neutrophil function in vitro ⬇️

scientific article published on September 1, 1998

Hydroxyacetophenone-derived antagonists of the peptidoleukotrienes.

scientific article

Mechanism of leukotriene D4-induced bronchoconstriction in normal subject.

scientific article published in September 1987

Naphtho[2,1-b][1,5] and [1,2-f][1,4]oxazocines as selective NK1 antagonists.

scientific article published on May 2004

Nonpeptidic inhibitors of human leukocyte elastase. 3. Design, synthesis, X-ray crystallographic analysis, and structure-activity relationships for a series of orally active 3-amino-6-phenylpyridin-2-one trifluoromethyl ketones

scientific article

Nonpeptidic inhibitors of human leukocyte elastase. 6. Design of a potent, intratracheally active, pyridone-based trifluoromethyl ketone

scientific article

Orally active trifluoromethyl ketone inhibitors of human leukocyte elastase

scientific article published on 01 September 1997

Pharmacophore-Based Design of Phenyl-[hydroxycyclohexyl] Cycloalkyl-Carboxamide Mitofusin Activators with Improved Neuronal Activity

scientific article published on 20 August 2021

Preclinical pharmacology and pharmacokinetics of AZD3783, a selective 5-hydroxytryptamine 1B receptor antagonist.

scientific article published on 8 August 2011

Structural analysis and optimization of NK(1) receptor antagonists through modulation of atropisomer interconversion properties.

scientific article published on January 2004

Synthesis, structure-activity relationships, and pharmacological evaluation of a series of fluorinated 3-benzyl-5-indolecarboxamides: identification of 4-[[5-[((2R)-2-methyl-4,4,4-trifluorobutyl)carbamoyl]-1-methyl indol- 3-yl]methyl]-3-methoxy-N-[(

scientific article published on 01 April 1994

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