List of works - Jean-François Brière

A Unique (3+2) Annulation Reaction between Meldrum's Acid and Nitrones: Mechanistic Insight by ESI-IMS-MS and DFT Studies.

scientific article published on 3 January 2018

A diastereoselective and concise synthesis of functionalised vinyl epoxides with a Morita-Baylis-Hillman backbone

scientific article published on 10 July 2006

A stereodivergent synthesis of beta-hydroxy-alpha-methylene lactones via vinyl epoxides.

scientific article published on 9 April 2008

Base-Assisted Intramolecular C–N Coupling Reaction from NH2-Bound Cyclopalladated l-Phenylalanine to Indoline-2-carboxylic Acid

scientific article

Concise synthesis of an enantiopure bicyclic pyrazinone as constrained peptidomimetic building block

scientific article published on 03 February 2012

Design of sulfides with a locked conformation as promoters of catalytic and asymmetric sulfonium ylide epoxidation.

scientific article published in May 2005

Developments in Meyers' lactamization methodology: en route to bi(hetero)aryl structures with defined axial chirality

scientific article published on 07 August 2013

Domino Aza-Michael-ih-Diels-Alder Reaction to Various 3-Vinyl-1,2,4-triazines: Access to Polysubstituted Tetrahydro-1,6-naphthyridines.

scientific article

Enantioselective Phase-Transfer Catalyzed α-Sulfanylation of Isoxazolidin-5-ones: An Entry to β(2,2) -Amino Acid Derivatives

scientific article published on 14 September 2016

Enantioselective catalytic synthesis of α-aryl-α-SCF3-β2,2-amino acids

scientific article published on 01 January 2020

Enantioselective phase-transfer catalysis: synthesis of pyrazolines

scientific article published on 01 September 2010

Enantioselective synthesis of bio-relevant 3,5-diaryl pyrazolines

scientific article published on 11 April 2012

Heterogeneous-phase Sonogashira cross-coupling reaction on COC surface for the grafting of biomolecules - Application to isatin

scientific article published on 03 June 2019

Highly regio- and diastereoselective anionic [3 + 2] cycloaddition under phase transfer catalytic conditions

scientific article published on 28 April 2011

Intramolecular photochemical dioxenone-alkene [2 + 2] cycloadditions as an approach to the bicyclo[2.1.1]hexane moiety of solanoeclepin A.

scientific article

Organocatalysed decarboxylative protonation process from Meldrum's acid: enantioselective synthesis of isoxazolidinones.

scientific article

Organocatalysed multicomponent synthesis of pyrazolidinones: Meldrum's acid approach

scientific article published on 01 September 2014

Organocatalysed synthesis of isoxazolines initiated by a chemoselective oxa-Michael reaction of N-BocNHOH

scientific article published on 01 February 2014

Organocatalytic Multicomponent Synthesis of α/β-Dipeptide Derivatives

scientific article published on 11 March 2020

Organocatalytic aza-Michael Reaction to 3-Vinyl-1,2,4-triazines as a Valuable Bifunctional Platform

scientific article published on 01 March 2019

Organocatalyzed Multicomponent Synthesis of Isoxazolidin-5-ones

scientific article published on 21 October 2015

Recent advances in cooperative ion pairing in asymmetric organocatalysis.

scientific article

Scaffold hopping strategy toward original pyrazolines as selective CB2 receptor ligands

scientific article published on 26 October 2012

Second generation N-heterocyclic carbene-Pt(0) complexes as efficient catalysts for the hydrosilylation of alkenes

scientific article published on 21 June 2005

Sequential Michael Addition and Enamine-Promoted Inverse Electron Demanding Diels-Alder Reaction upon 3-Vinyl-1,2,4-triazine Platforms

scientific article published on 11 June 2015

Stereocontrolled lithiation/trapping of chiral 2-alkylideneaziridines: investigation into the role of the aziridine nitrogen stereodynamics

scientific article published on 01 November 2014

Straightforward stereoselective synthesis of spiro-epoxyoxindoles

scientific article published on 30 March 2007

TBD-organocatalysed synthesis of pyrazolines.

scientific article published on 17 July 2009

The Catalytic Regio- and Stereoselective Synthesis of 1,6-Diazabicyclo[4.3.0]nonane-2,7-diones

scientific article

List of works by Jean-François Brière

A Unique (3+2) Annulation Reaction between Meldrum's Acid and Nitrones: Mechanistic Insight by ESI-IMS-MS and DFT Studies.

A diastereoselective and concise synthesis of functionalised vinyl epoxides with a Morita-Baylis-Hillman backbone

A stereodivergent synthesis of beta-hydroxy-alpha-methylene lactones via vinyl epoxides.

Base-Assisted Intramolecular C–N Coupling Reaction from NH2-Bound Cyclopalladated l-Phenylalanine to Indoline-2-carboxylic Acid

Concise synthesis of an enantiopure bicyclic pyrazinone as constrained peptidomimetic building block

Design of sulfides with a locked conformation as promoters of catalytic and asymmetric sulfonium ylide epoxidation.

Developments in Meyers' lactamization methodology: en route to bi(hetero)aryl structures with defined axial chirality

Domino Aza-Michael-ih-Diels-Alder Reaction to Various 3-Vinyl-1,2,4-triazines: Access to Polysubstituted Tetrahydro-1,6-naphthyridines.

Enantioselective Phase-Transfer Catalyzed α-Sulfanylation of Isoxazolidin-5-ones: An Entry to β(2,2) -Amino Acid Derivatives

Enantioselective catalytic synthesis of α-aryl-α-SCF3-β2,2-amino acids

Enantioselective phase-transfer catalysis: synthesis of pyrazolines

Enantioselective synthesis of bio-relevant 3,5-diaryl pyrazolines

Heterogeneous-phase Sonogashira cross-coupling reaction on COC surface for the grafting of biomolecules - Application to isatin

Highly regio- and diastereoselective anionic [3 + 2] cycloaddition under phase transfer catalytic conditions

Intramolecular photochemical dioxenone-alkene [2 + 2] cycloadditions as an approach to the bicyclo[2.1.1]hexane moiety of solanoeclepin A.

Organocatalysed decarboxylative protonation process from Meldrum's acid: enantioselective synthesis of isoxazolidinones.

Organocatalysed multicomponent synthesis of pyrazolidinones: Meldrum's acid approach

Organocatalysed synthesis of isoxazolines initiated by a chemoselective oxa-Michael reaction of N-BocNHOH

Organocatalytic Multicomponent Synthesis of α/β-Dipeptide Derivatives

Organocatalytic aza-Michael Reaction to 3-Vinyl-1,2,4-triazines as a Valuable Bifunctional Platform

Organocatalyzed Multicomponent Synthesis of Isoxazolidin-5-ones

Recent advances in cooperative ion pairing in asymmetric organocatalysis.

Scaffold hopping strategy toward original pyrazolines as selective CB2 receptor ligands

Second generation N-heterocyclic carbene-Pt(0) complexes as efficient catalysts for the hydrosilylation of alkenes

Sequential Michael Addition and Enamine-Promoted Inverse Electron Demanding Diels-Alder Reaction upon 3-Vinyl-1,2,4-triazine Platforms

Stereocontrolled lithiation/trapping of chiral 2-alkylideneaziridines: investigation into the role of the aziridine nitrogen stereodynamics

Straightforward stereoselective synthesis of spiro-epoxyoxindoles

TBD-organocatalysed synthesis of pyrazolines.

The Catalytic Regio- and Stereoselective Synthesis of 1,6-Diazabicyclo[4.3.0]nonane-2,7-diones