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List of works by Robert Roskoski

A historical overview of protein kinases and their targeted small molecule inhibitors

scientific article published on 21 July 2015

Allosteric MEK1/2 inhibitors including cobimetanib and trametinib in the treatment of cutaneous melanomas

scientific article published on 9 December 2016

Anaplastic lymphoma kinase (ALK) inhibitors in the treatment of ALK-driven lung cancers

scientific article published on 8 January 2017

Anaplastic lymphoma kinase (ALK): Structure, oncogenic activation, and pharmacological inhibition

scientific article published on November 28, 2012

Classification of small molecule protein kinase inhibitors based upon the structures of their drug-enzyme complexes

scientific article published on 31 October 2015

Complex molecular regulation of tyrosine hydroxylase

scientific article published on 28 May 2014

Corrigendum to "Guidelines for preparing color figures for everyone including the colorblind" [Pharmacol. Res. 119 (2017) 240-241]

scientific article published on 29 September 2018

Cyclin-dependent protein kinase inhibitors including palbociclib as anticancer drugs

scientific article published on 16 March 2016

Cyclin-dependent protein serine/threonine kinase inhibitors as anticancer drugs

scientific article published on 30 November 2018

Dopamine, in the presence of tyrosinase, covalently modifies and inactivates tyrosine hydroxylase

scientific article published in December 1998

ERK1/2 MAP kinases: structure, function, and regulation

scientific article published on 27 April 2012

ErbB/HER protein-tyrosine kinases: Structures and small molecule inhibitors

scientific article

Guidelines for preparing color figures for everyone including the colorblind

scientific article published on 8 February 2017

Ibrutinib inhibition of Bruton protein-tyrosine kinase (BTK) in the treatment of B cell neoplasms

scientific article published on 15 September 2016

Janus kinase (JAK) inhibitors in the treatment of inflammatory and neoplastic diseases

scientific article

MEK1/2 dual-specificity protein kinases: Structure and regulation

scientific article published on 08 December 2011

Protein prenylation: a pivotal posttranslational process

scientific article

RAF protein-serine/threonine kinases: Structure and regulation

scientific article published on July 30, 2010

ROS1 protein-tyrosine kinase inhibitors in the treatment of ROS1 fusion protein-driven non-small cell lung cancers

scientific article published on 29 April 2017

Role of RET protein-tyrosine kinase inhibitors in the treatment RET-driven thyroid and lung cancers

scientific article

STI-571: an anticancer protein-tyrosine kinase inhibitor

scientific article

Signaling by Kit protein-tyrosine kinase--the stem cell factor receptor

scientific article

Small molecule inhibitors targeting the EGFR/ErbB family of protein-tyrosine kinases in human cancers

scientific article published on 27 November 2018

Src kinase regulation by phosphorylation and dephosphorylation

scientific article (publication date: 27 May 2005)

Src protein-tyrosine kinase structure and regulation

scientific article

Src protein-tyrosine kinase structure, mechanism, and small molecule inhibitors

scientific article published on 3 February 2015

Structure and regulation of Kit protein-tyrosine kinase--the stem cell factor receptor

scientific article

Sunitinib: a VEGF and PDGF receptor protein kinase and angiogenesis inhibitor

scientific article

Targeting oncogenic Raf protein-serine/threonine kinases in human cancers

scientific article published on 15 August 2018

The ErbB/HER family of protein-tyrosine kinases and cancer

scientific article

The ErbB/HER receptor protein-tyrosine kinases and cancer

scientific article

The biosynthesis of N-arachidonoyl dopamine (NADA), a putative endocannabinoid and endovanilloid, via conjugation of arachidonic acid with dopamine

scientific article published on 30 June 2009

The preclinical profile of crizotinib for the treatment of non-small-cell lung cancer and other neoplastic disorders

scientific article

The role of small molecule Kit protein-tyrosine kinase inhibitors in the treatment of neoplastic disorders.

scientific article

The role of small molecule platelet-derived growth factor receptor (PDGFR) inhibitors in the treatment of neoplastic disorders

scientific article published on 2 February 2018

VEGF receptor protein-tyrosine kinases: structure and regulation

scientific article published on 03 August 2008

Vascular endothelial growth factor (VEGF) and VEGF receptor inhibitors in the treatment of renal cell carcinomas

scientific article published on 18 March 2017

Vascular endothelial growth factor (VEGF) signaling in tumor progression

scientific article published on 26 February 2007