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List of works by Gilles H Goetz

'Upenamide: An unprecedented macrocyclic alkaloid from the Indonesian sponge Echinochalina sp

scientific article published on 01 December 2000

A Fast Chromatographic Method for Estimating Lipophilicity and Ionization in Nonpolar Membrane-Like Environment

article

A new depsipeptide from the sacoglossan mollusk Elysia ornata and the green alga Bryopsis species

scientific article published on 01 January 2000

Chemical and biological integrity in natural products screening

scientific article published on 01 September 2005

Chiral Sulfoxide-Induced Single Turn Peptide α-Helicity.

scientific article published on 9 December 2016

Comparative pharmacokinetic profile of cyclosporine (CsA) with a decapeptide and a linear analogue

scientific article published on 07 March 2017

Desorption electrospray ionization (DESI) with atmospheric pressure ion mobility spectrometry for drug detection

scientific article

Determining molecular properties with differential mobility spectrometry and machine learning

scientific article published in Nature Communications

Discovery of Potent and Orally Bioavailable Macrocyclic Peptide-Peptoid Hybrid CXCR7 Modulators.

scientific article published on 18 October 2017

Discovery of a novel class of exquisitely selective mesenchymal-epithelial transition factor (c-MET) protein kinase inhibitors and identification of the clinical candidate 2-(4-(1-(quinolin-6-ylmethyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)-1H-pyraz

scientific article

EPSA: A Novel Supercritical Fluid Chromatography Technique Enabling the Design of Permeable Cyclic Peptides.

scientific article published on 4 August 2014

High throughput method for the indirect detection of intramolecular hydrogen bonding

scientific article published on 31 March 2014

Integrating Intramolecular Hydrogen Bonding (IMHB) Considerations in Drug Discovery Using ΔlogP As a Tool

scientific article published on 12 June 2013

Kulokekahilide-1, a cytotoxic depsipeptide from the cephalaspidean mollusk Philinopsis speciosa.

scientific article published in March 2002

On-column solvent exchange for purified preparative fractions

scientific article published on 14 May 2010

Peptide to Peptoid Substitutions Increase Cell Permeability in Cyclic Hexapeptides.

scientific article published on 5 June 2015

Relationship between Passive Permeability and Molecular Polarity Using Block Relevance Analysis.

scientific article published on 30 December 2016

Synthesis of a water-soluble analog of 6-methyl-3-N-alkyl catechol labeled with carbon 13: NMR approach to the reactivity of poison ivy/oak sensitizers toward proteins.

scientific article

Systematic N-methylation of oxytocin: Impact on pharmacology and intramolecular hydrogen bonding network.

scientific article published on 31 May 2016

Terpenes and flavonoids from an Egyptian collection of Cleome droserifolia.

scientific article published in April 2010

The cyanobacterial origin of potent anticancer agents originally isolated from sea hares.

scientific article

The discovery of potent nonstructural protein 5A (NS5A) inhibitors with a unique resistance profile-Part 2.

scientific article published on 11 April 2014

Ugibohlin: a new dibromo-seco-isophakellin from Axinella carteri

scientific article published on 01 December 2001

Use of 3D properties to characterize beyond rule-of-5 property space for passive permeation

scientific article published on 20 March 2012