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List of works by Bharat Shimpukade

Complex Pharmacology of Free Fatty Acid Receptors.

scientific article published on 14 June 2016

Concomitant action of structural elements and receptor phosphorylation determines arrestin-3 interaction with the free fatty acid receptor FFA4

scientific article published on 9 May 2014

Discovery of a Potent Free Fatty Acid 1 Receptor Agonist with Low Lipophilicity, Low Polar Surface Area, and Robust in Vivo Efficacy.

scientific article published on March 2016

Discovery of a potent and selective GPR120 agonist.

scientific article published on 2 May 2012

Epiminocyclohepta[b]indole analogs as 5-HT6 antagonists

scientific article published on 14 January 2012

Non-Acidic Free Fatty Acid Receptor 4 Agonists with Antidiabetic Activity

scientific article published on 29 August 2016

The GPR120 agonist TUG-891 promotes metabolic health by stimulating mitochondrial respiration in brown fat.

scientific article published on 17 January 2018

The molecular basis of ligand interaction at free fatty acid receptor 4 (FFA4/GPR120).

scientific article published on 24 May 2014

The pharmacology of TUG-891, a potent and selective agonist of the free fatty acid receptor 4 (FFA4/GPR120), demonstrates both potential opportunity and possible challenges to therapeutic agonism

scientific article published on 26 August 2013

Treatment with TUG891, a free fatty acid receptor 4 agonist, restores adipose tissue metabolic dysfunction following chronic sleep fragmentation in mice.

scientific article published on 16 March 2016