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List of works by Brendan Kelly

Allosteric modulation in monomers and oligomers of a G protein-coupled receptor

scientific article published on 06 May 2016

Correction to α2-Adrenoceptor Antagonists: Synthesis, Pharmacological Evaluation, and Molecular Modeling Investigation of Pyridinoguanidine, Pyridino-2-aminoimidazoline and Their Derivatives

scientific article published on 14 April 2015

Cryptic pocket formation underlies allosteric modulator selectivity at muscarinic GPCRs

scientific article published on 23 July 2019

Crystal Structure of a Full-Length Human Tetraspanin Reveals a Cholesterol-Binding Pocket

scientific article

Guanidinium-based derivatives: searching for new kinase inhibitors.

scientific article

Non-Covalent Interactions: Complexes of Guanidinium with DNA and RNA Nucleobases

scientific article published on 19 September 2013

Probing a 3,4'-bis-guanidinium diaryl derivative as an allosteric inhibitor of the Ras pathway.

scientific article published on 18 August 2015

Pyridin-2-yl Guanidine Derivatives: Conformational Control Induced by Intramolecular Hydrogen-Bonding Interactions

scientific article published on 17 October 2011

Single-Molecule Analysis of the Supramolecular Organization of the M2 Muscarinic Receptor and the Gαi1 Protein.

scientific article

Structure-activity relationships in non-ligand binding pocket (non-LBP) diarylhydrazide antiandrogens.

scientific article

Structure-inspired design of β-arrestin-biased ligands for aminergic GPCRs.

scientific article

Synthesis, biological evaluation and molecular modeling study of 5-trifluoromethyl-Δ2-pyrazoline and isomeric 5/3-trifluoromethylpyrazole derivatives as anti-inflammatory agents

scientific article published on 07 October 2013

Thiophene/thiazole-benzene replacement on guanidine derivatives targeting α2-Adrenoceptors.

scientific article

α2-adrenoceptor antagonists: synthesis, pharmacological evaluation, and molecular modeling investigation of pyridinoguanidine, pyridino-2-aminoimidazoline and their derivatives

scientific article published on 2 January 2015