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List of works by Xavier Ligneau

4-(omega-(alkyloxy)alkyl)-1H-imidazole derivatives as histamine H(3) receptor antagonists/agonists

scientific article published on May 2004

Acidic elements in histamine H(3) receptor antagonists

scientific article published on 21 January 2010

An inverse agonist of the histamine H(3) receptor improves wakefulness in narcolepsy: studies in orexin-/- mice and patients

scientific article

Brain histamine and schizophrenia: potential therapeutic applications of H3-receptor inverse agonists studied with BF2.649.

scientific article

Ether derivatives of 3-piperidinopropan-1-ol as non-imidazole histamine H3 receptor antagonists

scientific article published on 8 February 2006

First metal-containing histamine H3 receptor ligands

scientific article published in June 2010

High constitutive activity of native H3 receptors regulates histamine neurons in brain.

scientific article

Influence of bulky substituents on histamine h(3) receptor agonist/antagonist properties

scientific article published in August 2002

Meta-substituted aryl(thio)ethers as potent partial agonists (or antagonists) for the histamine H3 receptor lacking a nitrogen atom in the side chain

scientific article

Nonclinical cardiovascular safety of pitolisant: comparing International Conference on Harmonization S7B and Comprehensive in vitro Pro-arrhythmia Assay initiative studies.

scientific article published on 23 September 2017

Novel nonimidazole histamine H3 receptor antagonists: 1-(4-(phenoxymethyl)benzyl)piperidines and related compounds

scientific article published in April 2003

Piperidino-hydrocarbon compounds as novel non-imidazole histamine H(3)-receptor antagonists

scientific article

Preclinical evaluation of the abuse potential of Pitolisant, a histamine H₃ receptor inverse agonist/antagonist compared with Modafinil

scientific article published on June 2013

Progress in the proxifan class: heterocyclic congeners as novel potent and selective histamine H(3)-receptor antagonists

scientific article published in May 2002

Protean agonism at histamine H3 receptors in vitro and in vivo

scientific article

Search for histamine H(3) receptor ligands with combined inhibitory potency at histamine N-methyltransferase: omega-piperidinoalkanamine derivatives

scientific article published in October 2004

Structural variations of 1-(4-(phenoxymethyl)benzyl)piperidines as nonimidazole histamine H3 receptor antagonists

scientific article published in May 2004

Synthesis and evaluation of a 2-benzothiazolylphenylmethyl ether class of histamine H4 receptor antagonists

scientific article published on 19 September 2016

Therapeutic implications of constitutive activity of receptors: the example of the histamine H3 receptor.

scientific article

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