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List of works by Victoria Magrioti

2-Oxoamide inhibitors of cytosolic group IVA phospholipase A2 with reduced lipophilicity

scientific article published on 27 July 2016

2-Oxoamide inhibitors of phospholipase A2 activity and cellular arachidonate release based on dipeptides and pseudodipeptides

scientific article published on 03 May 2009

2-Oxoesters: A Novel Class of Potent and Selective Inhibitors of Cytosolic Group IVA Phospholipase A2.

scientific article published on August 2017

Autotaxin inhibitors: a patent review ⬇️

scientific article published on 06 May 2013

Cytosolic group IVA and calcium-independent group VIA phospholipase A2s act on distinct phospholipid pools in zymosan-stimulated mouse peritoneal macrophages

scientific article published on 13 December 2013

Differing roles for members of the phospholipase A2 superfamily in experimental autoimmune encephalomyelitis.

scientific article published on 13 February 2009

Inhibition of Ca2+-independent phospholipase A2β (iPLA2β) ameliorates islet infiltration and incidence of diabetes in NOD mice

scientific article

Inhibition of group IVA cytosolic phospholipase A2 by thiazolyl ketones in vitro, ex vivo, and in vivo

scientific article published on 3 September 2014

Inhibition of secreted phospholipases A₂ by 2-oxoamides based on α-amino acids: Synthesis, in vitro evaluation and molecular docking calculations.

scientific article

Inhibitors of secreted phospholipase A2 suppress the release of PGE2 in renal mesangial cells

scientific article published on 13 May 2016

New potent and selective polyfluoroalkyl ketone inhibitors of GVIA calcium-independent phospholipase A2.

scientific article published on 16 July 2013

Phospholipase A2 enzymes: physical structure, biological function, disease implication, chemical inhibition, and therapeutic intervention

scientific article

Phospholipase A2 inhibitors as potential therapeutic agents for the treatment of inflammatory diseases.

scientific article published on January 2010

Phospholipase A2 inhibitors for the treatment of inflammatory diseases: a patent review (2010--present).

scientific article published on 08 January 2013

Potent and selective fluoroketone inhibitors of group VIA calcium-independent phospholipase A2.

scientific article

Sterically hindered triacylglycerol analogues as potent inhibitors of human digestive lipases.

scientific article published in March 2004

Structure-activity relationship of 2-oxoamide inhibition of group IVA cytosolic phospholipase A2 and group V secreted phospholipase A2.

scientific article published on 2 August 2007

Structure-activity relationships of natural and non-natural amino acid-based amide and 2-oxoamide inhibitors of human phospholipase A(2) enzymes

scientific article

Synthesis and In vivo anti-inflammatory activity of long-chain 2-amino-alcohols.

scientific article

Synthesis and use of N, N-di-Boc-glutamate gamma-semialdehydes and related aldehydes.

scientific article

Synthesis of (S)-alpha-amino oleic acid.

scientific article published in February 2002

Synthesis of 2-oxoamides based on sulfonamide analogs of gamma-amino acids and their activity on phospholipase A2.

scientific article published on October 2008

Synthesis of Long-Chain β-Lactones and Their Antibacterial Activities against Pathogenic Mycobacteria

scientific article published on 17 January 2019

Synthesis of enantiopure non-natural alpha-amino acids using tert-butyl (2S)-2-[bis-(tert-butoxycarbonyl)amino]-5-oxopentanoate as key-intermediate:the first synthesis of(S)-2-amino-oleic acid.

scientific article

Synthesis of polyfluoro ketones for selective inhibition of human phospholipase A2 enzymes

scientific article published on December 2008

Triacylglycerols based on 2-(N-tert-butoxycarbonylamino)oleic acid are potent inhibitors of pancreatic lipase.

scientific article

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