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List of works by Gabriel Navarrete-Vazquez

2-(2-Benzyl-oxyphen-yl)-1H-benzimid-azole.

scientific article published on 20 February 2008

2-(4-Acetamido-phen-oxy)-2-methyl-propanoic acid.

scientific article published on 28 February 2013

2-Methyl-2-(4-nitro-phen-oxy)propanoic acid

scientific article published on 8 November 2008

2-Methyl-2-(4-nitro-phenyl-sulfanyl)-propanoic acid

scientific article published on 6 December 2007

2-acylamino-5-nitro-1,3-thiazoles: preparation and in vitro bioevaluation against four neglected protozoan parasites

scientific article published on 31 January 2014

4-Meth-oxy-N-[6-methyl-2,3-dihydro-1,3-benzothia-zol-2-yl-idene]benzene-sulfonamide.

scientific article published on 6 December 2007

A comparative study of flavonoid analogues on streptozotocin-nicotinamide induced diabetic rats: quercetin as a potential antidiabetic agent acting via 11beta-hydroxysteroid dehydrogenase type 1 inhibition.

scientific article published in March 2010

Activity and property landscape modeling is at the interface of chemoinformatics and medicinal chemistry

scientific article published on July 2015

Antidiabetic activity of N-(6-substituted-1,3-benzothiazol-2-yl)benzenesulfonamides.

scientific article

Antidiabetic activity of some pentacyclic acid triterpenoids, role of PTP-1B: in vitro, in silico, and in vivo approaches

scientific article published on 30 March 2011

Antidiabetic and toxicological evaluations of naringenin in normoglycaemic and NIDDM rat models and its implications on extra-pancreatic glucose regulation.

scientific article

Antidiabetic effect of Achillea millefollium through multitarget interactions: α-glucosidases inhibition, insulin sensitization and insulin secretagogue activities.

scientific article published on 12 October 2017

Antidiabetic effect of Cordia morelosana, chemical and pharmacological studies

scientific article published on 07 January 2020

Antidiabetic, antihyperlipidemic and anti-inflammatory effects of tilianin in streptozotocin-nicotinamide diabetic rats.

scientific article published on 26 July 2016

Antihyperalgesic activity of a novel synthesized analogue of lidocaine in diabetic rats

scientific article published on 31 January 2013

Antihypertensive and vasorelaxant effects of dihydrospinochalcone-A isolated from Lonchocarpus xuul Lundell by NO production: computational and ex vivo approaches.

scientific article published on 20 July 2013

Antinociceptive effects of a new sigma-1 receptor antagonist (N-(2-morpholin-4-yl-ethyl)-2-(1-naphthyloxy)acetamide) in two types of nociception

scientific article published on 10 December 2015

Antiprotozoal Nitazoxanide Derivatives: Synthesis, Bioassays and QSAR Study Combined with Docking for Mechanistic Insight.

scientific article

Biopharmaceutic evaluation of novel anthelmintic (1H-benzimidazol-5(6)-yl)carboxamide derivatives

scientific article published on 16 May 2007

Biopharmaceutical Characterization and Bioavailability Study of a Tetrazole Analog of Clofibric Acid in Rat.

scientific article published on 14 February 2017

CB1 cannabinoid receptor expression is regulated by glucose and feeding in rat pancreatic islets.

scientific article published on 5 May 2010

Chemical constituents of the hemiparasitic plant Phoradendron brachystachyum DC Nutt (Viscaceae)

scientific article published on 23 February 2012

Complementary pharmacological and toxicological characterization data on the pharmacological profile of N-(2,6-dichlorophenyl)-2-(4-methyl-1-piperidinyl) acetamide.

scientific article

Complete NMR assignment of 3, 4-seco-lup-20(29)-en-3-oic acid from Decatropis bicolor

scientific article published on 5 March 2012

Crystal structure of 4-methyl-7-prop-oxy-2H-chromen-2-one

scientific article published on 31 October 2014

Depressant effects of Agastache mexicana methanol extract and one of major metabolites tilianin

scientific article published on 01 March 2015

Design and synthesis of N‑(benzylpiperidinyl)‑4‑fluorobenzamide: A haloperidol analog that reduces neuropathic nociception via σ1 receptor antagonism

scientific article published on 23 January 2020

Design, Synthesis and Biological Evaluation of 2-(2-Amino-5(6)-nitro-1H-benzimidazol-1-yl)-N-arylacetamides as Antiprotozoal Agents.

scientific article

Design, Synthesis and in Combo Antidiabetic Bioevaluation of Multitarget Phenylpropanoic Acids.

scientific article published on 6 February 2018

Design, microwave-assisted synthesis, and spasmolytic activity of 2-(alkyloxyaryl)-1H-benzimidazole derivatives as constrained stilbene bioisosteres

scientific article published on 19 June 2006

Design, synthesis and in vitro antiprotozoal activity of benzimidazole-pentamidine hybrids.

scientific article published on 4 May 2008

Design, synthesis, and in vitro antiprotozoal, antimycobacterial activities of N-{2-[(7-chloroquinolin-4-yl)amino]ethyl}ureas.

scientific article published on 30 July 2010

Design, synthesis, in vitro, in vivo and in silico pharmacological characterization of antidiabetic N-Boc-l-tyrosine-based compounds

scientific article published on 21 September 2018

Discovery of 2-(3,4-dichlorophenoxy)-N-(2-morpholin-4-ylethyl)acetamide: A selective σ1 receptor ligand with antinociceptive effect

scientific article published on 14 March 2016

Discovery of new dual PPARγ-GPR40 agonists with robust antidiabetic activity: Design, synthesis and in combo drug evaluation

scientific article published on 22 March 2017

Discovery of thiazolidine-2,4-dione/biphenylcarbonitrile hybrid as dual PPAR α/γ modulator with antidiabetic effect: in vitro, in silico and in vivo approaches.

scientific article published on 21 March 2013

Discovery, synthesis and in combo studies of a tetrazole analogue of clofibric acid as a potent hypoglycemic agent

scientific article published on 05 April 2013

Ethyl 2-{(2Z)-2-[(1-naphthyl-sulfon-yl)imino]-2,3-dihydro-1,3-thia-zol-4-yl}acetate monohydrate

scientific article published on 9 October 2010

Evaluation of the neuroprotective activity of stansin 6, a resin glycoside from Ipomoea stans.

scientific article published on 27 May 2014

Exploring the interplay of physicochemical properties, membrane permeability and giardicidal activity of some benzimidazole derivatives.

scientific article

Glycolipid ester-type heterodimers from Ipomoea tyrianthina and their pharmacological activity.

scientific article published on 25 June 2009

Hepta-, hexa-, penta-, tetra-, and trisaccharide resin glycosides from three species of Ipomoea and their antiproliferative activity on two glioma cell lines.

scientific article published on 2 July 2016

In vitro and in silico PTP-1B inhibition and in vivo antidiabetic activity of semisynthetic moronic acid derivatives

scientific article published on 03 March 2016

Metronidazole and Secnidazole Carbamates: Synthesis, Antiprotozoal Activity, and Molecular Dynamics Studies

scientific article published on 12 February 2020

Molecular Docking and Dynamics Simulation of Protein β-Tubulin and Antifungal Cyclic Lipopeptides

scientific article published on 18 September 2019

N-(2-morpholin-4-yl-ethyl)-2-(1naphthyloxy)acetamide inhibits the chronic constriction injury-generated hyperalgesia via the antagonism of sigma-1 receptors.

scientific article published on 23 June 2017

N-(4-Methoxy-2-nitrophenyl)hexadecanamide, a palmitoylethanolamide analogue, reduces formalin-induced nociception

scientific article published on 12 October 2012

Nitazoxanide, tizoxanide and a new analogue [4-nitro-N-(5-nitro-1,3-thiazol-2-yl)benzamide; NTB] inhibit the growth of kinetoplastid parasites (Trypanosoma cruzi and Leishmania mexicana) in vitro.

scientific article

Novel CB1 receptor antagonist BAR-1 modifies pancreatic islet function and clinical parameters in prediabetic and diabetic mice

scientific article published on 04 March 2020

Novel giardicidal compounds bearing proton pump inhibitor scaffold proceeding through triosephosphate isomerase inactivation

scientific article published on 10 August 2017

Novel inhibitors of human glucose-6-phosphate dehydrogenase (HsG6PD) affect the activity and stability of the protein

scientific article published on 18 December 2020

Palmitic acid analogues exhibiting antinociceptive activity in mice.

scientific article published in January 2007

Pharmacological characterization of the cardiovascular effect of Nibethione: ex vivo, in vivo and in silico studies

scientific article published on 04 June 2020

Pharmacological evaluation of metformin and N-benzylbiguanide, a novel analogue of metformin, on the vasopressor responses to adrenergic system stimulation in pithed rats with fructose-induced insulin resistance.

scientific article published in September 2017

Pharmacological profile of N-(2,6-dichlorophenyl)-2-(4-methyl-1-piperidinyl)acetamide, a novel analogue of lidocaine.

scientific article published on 12 May 2016

Proton pump inhibitors drastically modify triosephosphate isomerase from Giardia lamblia at functional and structural levels, providing molecular leads in the design of new antigiardiasic drugs

scientific article published on 28 October 2015

Relaxant activity of 2-(substituted phenyl)-1H-benzimidazoles on isolated rat aortic rings: design and synthesis of 5-nitro derivatives.

scientific article published on 17 February 2006

Relaxant effects of Artemisia ludoviciana on isolated rat smooth muscle tissues

article

Review of Theoretical Models to Study Natural Products with Antiprotozoal Activity.

scientific article published on 22 December 2016

Sedative, vasorelaxant, and cytotoxic effects of convolvulin from Ipomoea tyrianthina.

scientific article published on April 2011

Semisynthesis, ex vivo evaluation, and SAR studies of coumarin derivatives as potential antiasthmatic drugs.

scientific article published on 12 March 2014

Spasmolytic action of Lepechinia caulescens is through calcium channel blockade and NO release.

scientific article published on 19 August 2007

Synthesis and antimycobacterial activity of 4-(5-substituted-1,3,4-oxadiazol-2-yl)pyridines

scientific article published on 25 May 2007

Synthesis and antinociceptive evaluation of bioisosteres and hybrids of naproxen, ibuprofen and paracetamol.

scientific article published on 4 March 2018

Synthesis and antiparasitic activity of 1H-benzimidazole derivatives.

scientific article

Synthesis and antiparasitic activity of albendazole and mebendazole analogues.

scientific article published in October 2003

Synthesis and antiprotozoal activity of some 2-(trifluoromethyl)-1H-benzimidazole bioisosteres

scientific article published on 2 November 2005

Synthesis and biological activity of 2-(trifluoromethyl)-1H-benzimidazole derivatives against some protozoa and Trichinella spiralis

scientific article published on 7 April 2010

Synthesis and evaluation of thiazolidine-2,4-dione/benzazole derivatives as inhibitors of protein tyrosine phosphatase 1B (PTP-1B): Antihyperglycemic activity with molecular docking study

scientific article published on 29 August 2018

Synthesis and in vitro trichomonicidal, giardicidal and amebicidal activity of N-acetamide(sulfonamide)-2-methyl-4-nitro-1H-imidazoles

scientific article

Synthesis and preliminary evaluation of selected 2-aryl-5(6)-nitro- 1H-benzimidazole derivatives as potential anticancer agents

scientific article published on February 2011

Synthesis of 2-{2-[(α/β-naphthalen-1-ylsulfonyl)amino]-1,3-thiazol-4-yl} acetamides with 11β-hydroxysteroid dehydrogenase inhibition and in combo antidiabetic activities

scientific article published on 08 January 2014

Synthesis of benzologues of Nitazoxanide and Tizoxanide: a comparative study of their in vitro broad-spectrum antiprotozoal activity.

scientific article

Synthesis of nitro(benzo)thiazole acetamides and in vitro antiprotozoal effect against amitochondriate parasites Giardia intestinalis and Trichomonas vaginalis

scientific article published on 10 March 2015

Synthesis of oleanolic acid derivatives: In vitro, in vivo and in silico studies for PTP-1B inhibition

scientific article published on 16 September 2014

Synthesis, Screening and in silico Simulations of Anti-Parasitic Propamidine/Benzimidazole Derivatives.

scientific article published on 11 August 2016

Synthesis, in vitro and computational studies of protein tyrosine phosphatase 1B inhibition of a small library of 2-arylsulfonylaminobenzothiazoles with antihyperglycemic activity.

scientific article

Synthesis, in vitro and in silico screening of ethyl 2-(6-substituted benzo[d]thiazol-2-ylamino)-2-oxoacetates as protein-tyrosine phosphatase 1B inhibitors

scientific article published on 26 April 2012

Synthesis, in vitro and in silico studies of a PPARγ and GLUT-4 modulator with hypoglycemic effect

scientific article published on 01 August 2014

Synthesis, in vitro and in vivo giardicidal activity of nitrothiazole-NSAID chimeras displaying broad antiprotozoal spectrum

scientific article published on 24 May 2017

Synthesis, vasorelaxant activity and antihypertensive effect of benzo[d]imidazole derivatives

scientific article published on 14 April 2010

Therapeutic efficacy of liposomes containing 4-(5-pentadecyl-1,3,4-oxadiazol-2-yl)pyridine in a murine model of progressive pulmonary tuberculosis.

scientific article published on 2 April 2015

Toxicological Screening of Four Bioactive Citroflavonoids: In Vitro, In Vivo, and In Silico Approaches

scientific article published on 16 December 2020

Tracheal relaxation through calcium channel blockade of Achillea millefolium hexanic extract and its main bioactive compounds

scientific article published on 05 February 2020

Triterpenoids from Hibiscus sabdariffa L. with PPARδ/γ Dual Agonist Action: In Vivo, In Vitro and In Silico Studies

scientific article published on 16 January 2019

Tyrianthinic acids from Ipomoea tyrianthina and their antimycobacterial activity, cytotoxicity, and effects on the central nervous system

scientific article published on October 2008

Ursolic acid derivatives as potential antidiabetic agents: In vitro, in vivo, and in silico studies.

scientific article

Ursolic acid mediates the vasorelaxant activity of Lepechinia caulescens via NO release in isolated rat thoracic aorta

scientific article published on 21 April 2006

Vasorelaxant activity of some structurally related triterpenic acids from Phoradendron reichenbachianum (Viscaceae) mainly by NO production: ex vivo and in silico studies

scientific article published on 29 May 2012

Vasorelaxant effect of flavonoids through calmodulin inhibition: Ex vivo, in vitro, and in silico approaches

scientific article published on 04 November 2010

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