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List of works by Philippe Gautret

A Convenient Method for the Conversion of a Carboxy Group into a 4,6-Dimethoxy-1,3,5-triazine Group: Application to N-Benzylpyroglutamic Acids

A new synthesis of pyrrolo[3,2-b]quinolines by a tandem electrocyclization–oxidation process

An Improved Synthesis of Methyl 1,3-Dihydro-2H-pyrrolo[3,4-b]quinoline-2-carboxylate

An efficient one-pot reaction for the synthesis of pyrazolones bearing a phenothiazine unit

Antagonists of the P2X7 receptor: mechanism of enantioselective recognition using highly sulfated and sulfobutylether cyclodextrins by capillary electrokinetic chromatography

scientific article published on 18 July 2014

Antioxidant Activity of New Benzo[de]quinolines and Lactams: 2DQuantitative Structure-Activity Relationships

scientific article published on 01 September 2012

Corrigendum to “Evaluation and comparison of three different separation techniques for analysis of retroamide enantiomers and their biological evaluation against h -P2X7 receptor” [J. Chromatogr. B 986–987 (2015) 35–43]

scientific article published on 24 May 2016

Discovery of ferrocene-containing farnesyltransferase inhibitors. Investigation of bulky lipophilic groups for the A2 binding site of farnesyltransferase

Eaton's reagent-mediated domino π-cationic arylations of aromatic carboxylic acids to Iasi-red polymethoxylated polycyclic aromatic hydrocarbons: products with unprecedented biological activities as tubulin polymerization inhibitors.

scientific article

Enantioseparation of pyroglutamide derivatives on polysaccharide based chiral stationary phases by high-performance liquid chromatography and supercritical fluid chromatography: a comparative study

scientific article published on 4 July 2014

Evaluation and comparison of three different separation techniques for analysis of retroamide enantiomers and their biological evaluation against h-P2X7 receptor

scientific article published on 09 February 2015

Impact of Functional Groups on the Copper-Initiated N-Arylation of 5-Functionalized Pyrrolidin-2-ones and Their Vinylogues

ON the silylation of diarylcarbinols

On the structure of compounds obtained from the reaction of amines with 6,6-dimethyl-5,7-dioxaspiro[2.5]octane-4,8-dione

On the synthesis and biological properties of isocombretastatins: a case of ketone homologation during Wittig reaction attempts

scholarly article in RSC Advances, vol. 3 no. 11, 2013

Studies on Pyrrolidinones. A Silylated Approach to Fused Triazoles

Studies on Pyrrolidinones. An Improved One Pot Synthesis of 1,2,3,5,10,10a-Hexahydrobenz[f]indolizine-3,10-dione

Studies on Pyrrolidinones. An Improved Synthesis of Pyroglutamoyl Chloride

Studies on Pyrrolidinones: Chemistry of Dimethoxytriazines

Studies on indolizines. Evaluation of their biological properties as microtubule-interacting agents and as melanoma targeting compounds.

scientific article

Studies on pyrrolidinone. Synthesis of aza analogs of podophyllotoxin and related compounds

article published in 1999

Studies on pyrrolidinones. On the application of copper-catalyzed arylation of methyl pyroglutamate to obtain a new benzo[de]quinoline scaffold

Studies on pyrrolidinones. Reaction of pyroglutamic acid and vinylogues with aromatics in Eaton’s reagent

Studies on pyrrolidinones. Synthesis and reactivity of somen-protected pyroglutamic derivatives

Studies on pyrrolidinones. Synthesis ofN-benzhydrylpyroglutamic acids and esters

Synthesis and anticancer activity of analogues of phenstatin, with a phenothiazine A-ring, as a new class of microtubule-targeting agents

scientific article

Synthesis and biological evaluation of a new class of triazin–triazoles as potential inhibitors of human farnesyltransferase

Synthesis and biological evaluation of a new series of phenothiazine-containing protein farnesyltransferase inhibitors

scientific article published on 14 November 2012

Synthesis and biological evaluation of fluoro analogues of antimitotic phenstatin

scientific article published on 4 April 2013

Synthesis and biological evaluation of phenstatin metabolites

scientific article published on 27 August 2011

The revisited synthesis of tert-butyl pyroglutamate derivatives

Toward new camptothecins. Part 5: On the synthesis of precursors for the crucial Friedländer reaction

Toward new camptothecins. Part 6: Synthesis of crucial ketones and their use in Friedländer reaction

Toward new camptothecins. Part 7: Synthesis of thioluotonin and its 5-methoxycarbonyl derivative