List of works - Renata Riva

A highly convergent synthesis of tricyclic N-heterocycles coupling an Ugi reaction with a tandem S(N)2'-Heck double cyclization.

scientific article

A new class of cis-monobactam derivatives bearing a sulfamoyloxymethyl or an N-alkylsulfamoyloxymethyl group at position 4: synthesis and antibacterial activity

scientific article published on 01 March 1998

A new diversity oriented and metal-free approach to highly functionalized 3H-pyrimidin-4-ones

scientific article published on 02 February 2011

A novel highly selective chiral auxiliary for the asymmetric synthesis of L- and D-alpha-amino acid derivatives via a multicomponent Ugi reaction

scientific article published on 01 January 2005

A novel intramolecular Ugi reaction with 7-azabicyclo[2.2.1]heptane derivatives followed by post-condensation acylations: a new entry to azanorbornyl peptidomimetics.

scientific article

Application of tandem Ugi multi-component reaction/ring closing metathesis to the synthesis of a conformationally restricted cyclic pentapeptide

scientific article published on 23 November 2004

Asymmetrized tris(hydroxymethyl)methane as a precursor of N- and O-containing 6-membered heterocycles through ring-closing metathesis

scientific article published on 01 April 2005

Correction to "Diastereoselective Passerini Reaction of Biobased Chiral Aldehydes: Divergent Synthesis of Various Polyfunctionalized Heterocycles"

scientific article published on 08 June 2016

Development of a stereoselective Ugi reaction starting from an oxanorbornene β-amino acid derivative

scientific article published on 30 March 2012

Diastereoselective Passerini Reaction of Biobased Chiral Aldehydes: Divergent Synthesis of Various Polyfunctionalized Heterocycles

scientific article published on 17 March 2016

Diastereoselective Ugi reaction of chiral 1,3-aminoalcohols derived from an organocatalytic Mannich reaction.

scientific article published on 26 January 2016

Diversity oriented and chemoenzymatic synthesis of densely functionalized pyrrolidines through a highly diastereoselective Ugi multicomponent reaction

scientific article published on 04 January 2012

Diversity-oriented synthesis of dihydrobenzoxazepinones by coupling the Ugi multicomponent reaction with a Mitsunobu cyclization

scientific article published on 17 January 2014

Diversity-oriented synthesis of intensively blue emissive 3-hydroxyisoquinolines by sequential Ugi four-component reaction/reductive Heck cyclization

scientific article published on 4 November 2014

Enantio- and diastereoselective synthesis of highly substituted benzazepines by a multicomponent strategy coupled with organocatalytic and enzymatic procedures.

scientific article published on 18 December 2013

Enzymatically promoted release of organic molecules linked to magnetic nanoparticles.

scientific article published on 27 March 2018

Highly Convergent Synthesis of Intensively Blue Emissive Furo[2,3-c]isoquinolines by a Palladium-Catalyzed Cyclization Cascade of Unsaturated Ugi Products

scientific article published on 8 January 2016

Identification of lead compounds as antagonists of protein Bcl-xL with a diversity-oriented multidisciplinary approach

scientific article

Indole alkaloids. Enantioselective synthesis of (–)-alloyohimbane by a chemoenzymatic approach

Isocyanides and arylacetic acids: synthesis and reactivity of 3-aryl-2-acyloxyacrylamides, an example of serendipity-oriented synthesis.

scientific article published in September 2009

Ketene three-component reaction: a metal-free multicomponent approach to stereodefined captodative olefins

scientific article published on 09 January 2013

Long-range diastereoselectivity in Ugi reactions of 2-substituted dihydrobenzoxazepines.

scientific article published on 13 July 2011

Multicomponent synthesis of benzoxazinones via tandem Ugi/Mitsunobu reactions: an unexpected cine-substitution

scientific article published on 01 August 2008

Multicomponent synthesis of dihydrobenzoxazepinones by coupling Ugi and Mitsunobu reactions

scientific article published on 01 November 2006

Multicomponent synthesis of dihydrobenzoxazepinones, bearing four diversity points, as potential α-helix mimics

scientific article

Multicomponent, fragment-based synthesis of polyphenol-containing peptidomimetics and their inhibiting activity on beta-amyloid oligomerization

scientific article published on 31 October 2017

Novel application of α-azido aldehydes in multicomponent reactions: synthesis of triazolo-fused dihydrooxazinones via a Passerini reaction-dipolar cycloaddition strategy

scientific article published on 27 June 2011

OPHA (oxidation-Passerini-hydrolysis-alkylation) strategy: a four-step, one-pot improvement of the alkylative Passerini reaction.

scientific article published on 10 April 2014

Optimized synthesis of phosphatidylserine.

scientific article published on 9 February 2010

Passerini Reactions on Biocatalytically Derived Chiral Azetidines.

scientific article

Photocatalyzed synthesis of isochromanones and isobenzofuranones under batch and flow conditions

scientific article

Polyfunctionalized pyrrolidines by Ugi multicomponent reaction followed by palladium-mediated SN2' cyclizations

scientific article published on 15 January 2008

Rapid access to the highly oxygenated aspidosperma alkaloids vindoline, vindorosine, and cathovaline

Simplified dynemicin analogues: diastereoselective synthesis and evaluation of their activity against plasmid DNA.

scientific article

Synthesis and DNA-cleaving activity of lactenediynes conjugated with DNA-complexing moieties.

scientific article published on 13 February 2008

Synthesis and biological evaluation of new conformationally biased integrin ligands based on a tetrahydroazoninone scaffold.

scientific article published on 2 December 2006

Synthesis of 5-carboxamide-oxazolines with a Passerini-Zhu/Staudinger-Aza-Wittig two-step protocol

scientific article published on 01 September 2010

Synthesis of Vinyl Isocyanides and Development of a Convertible Isonitrile.

scientific article published on 16 March 2016

Synthesis of triazolo-fused benzoxazepines and benzoxazepinones via Passerini reactions followed by 1,3-dipolar cycloadditions

scientific article published on 04 June 2014

Three in the spotlight: Photoinduced stereoselective synthesis of (Z)-acyloxyacrylamides through a multicomponent approach

scientific article published on 08 April 2014

Ugi and Passerini reactions of biocatalytically derived chiral aldehydes: application to the synthesis of bicyclic pyrrolidines and of antiviral agent telaprevir

scientific article published on 24 March 2015

Ugi multicomponent reaction followed by an intramolecular nucleophilic substitution: convergent multicomponent synthesis of 1-sulfonyl 1,4-diazepan-5-ones and of their benzo-fused derivatives

scientific article published on 20 February 2007

List of works by Renata Riva

A highly convergent synthesis of tricyclic N-heterocycles coupling an Ugi reaction with a tandem S(N)2'-Heck double cyclization.

A new class of cis-monobactam derivatives bearing a sulfamoyloxymethyl or an N-alkylsulfamoyloxymethyl group at position 4: synthesis and antibacterial activity

A new diversity oriented and metal-free approach to highly functionalized 3H-pyrimidin-4-ones

A novel highly selective chiral auxiliary for the asymmetric synthesis of L- and D-alpha-amino acid derivatives via a multicomponent Ugi reaction

A novel intramolecular Ugi reaction with 7-azabicyclo[2.2.1]heptane derivatives followed by post-condensation acylations: a new entry to azanorbornyl peptidomimetics.

Application of tandem Ugi multi-component reaction/ring closing metathesis to the synthesis of a conformationally restricted cyclic pentapeptide

Asymmetrized tris(hydroxymethyl)methane as a precursor of N- and O-containing 6-membered heterocycles through ring-closing metathesis

Correction to "Diastereoselective Passerini Reaction of Biobased Chiral Aldehydes: Divergent Synthesis of Various Polyfunctionalized Heterocycles"

Development of a stereoselective Ugi reaction starting from an oxanorbornene β-amino acid derivative

Diastereoselective Passerini Reaction of Biobased Chiral Aldehydes: Divergent Synthesis of Various Polyfunctionalized Heterocycles

Diastereoselective Ugi reaction of chiral 1,3-aminoalcohols derived from an organocatalytic Mannich reaction.

Diversity oriented and chemoenzymatic synthesis of densely functionalized pyrrolidines through a highly diastereoselective Ugi multicomponent reaction

Diversity-oriented synthesis of dihydrobenzoxazepinones by coupling the Ugi multicomponent reaction with a Mitsunobu cyclization

Diversity-oriented synthesis of intensively blue emissive 3-hydroxyisoquinolines by sequential Ugi four-component reaction/reductive Heck cyclization

Enantio- and diastereoselective synthesis of highly substituted benzazepines by a multicomponent strategy coupled with organocatalytic and enzymatic procedures.

Enzymatically promoted release of organic molecules linked to magnetic nanoparticles.

Highly Convergent Synthesis of Intensively Blue Emissive Furo[2,3-c]isoquinolines by a Palladium-Catalyzed Cyclization Cascade of Unsaturated Ugi Products

Identification of lead compounds as antagonists of protein Bcl-xL with a diversity-oriented multidisciplinary approach

Indole alkaloids. Enantioselective synthesis of (–)-alloyohimbane by a chemoenzymatic approach

Isocyanides and arylacetic acids: synthesis and reactivity of 3-aryl-2-acyloxyacrylamides, an example of serendipity-oriented synthesis.

Ketene three-component reaction: a metal-free multicomponent approach to stereodefined captodative olefins

Long-range diastereoselectivity in Ugi reactions of 2-substituted dihydrobenzoxazepines.

Multicomponent synthesis of benzoxazinones via tandem Ugi/Mitsunobu reactions: an unexpected cine-substitution

Multicomponent synthesis of dihydrobenzoxazepinones by coupling Ugi and Mitsunobu reactions

Multicomponent synthesis of dihydrobenzoxazepinones, bearing four diversity points, as potential α-helix mimics

Multicomponent, fragment-based synthesis of polyphenol-containing peptidomimetics and their inhibiting activity on beta-amyloid oligomerization

Novel application of α-azido aldehydes in multicomponent reactions: synthesis of triazolo-fused dihydrooxazinones via a Passerini reaction-dipolar cycloaddition strategy

OPHA (oxidation-Passerini-hydrolysis-alkylation) strategy: a four-step, one-pot improvement of the alkylative Passerini reaction.

Optimized synthesis of phosphatidylserine.

Passerini Reactions on Biocatalytically Derived Chiral Azetidines.

Photocatalyzed synthesis of isochromanones and isobenzofuranones under batch and flow conditions

Polyfunctionalized pyrrolidines by Ugi multicomponent reaction followed by palladium-mediated SN2' cyclizations

Rapid access to the highly oxygenated aspidosperma alkaloids vindoline, vindorosine, and cathovaline

Simplified dynemicin analogues: diastereoselective synthesis and evaluation of their activity against plasmid DNA.

Synthesis and DNA-cleaving activity of lactenediynes conjugated with DNA-complexing moieties.

Synthesis and biological evaluation of new conformationally biased integrin ligands based on a tetrahydroazoninone scaffold.

Synthesis of 5-carboxamide-oxazolines with a Passerini-Zhu/Staudinger-Aza-Wittig two-step protocol

Synthesis of Vinyl Isocyanides and Development of a Convertible Isonitrile.

Synthesis of triazolo-fused benzoxazepines and benzoxazepinones via Passerini reactions followed by 1,3-dipolar cycloadditions

Three in the spotlight: Photoinduced stereoselective synthesis of (Z)-acyloxyacrylamides through a multicomponent approach

Ugi and Passerini reactions of biocatalytically derived chiral aldehydes: application to the synthesis of bicyclic pyrrolidines and of antiviral agent telaprevir

Ugi multicomponent reaction followed by an intramolecular nucleophilic substitution: convergent multicomponent synthesis of 1-sulfonyl 1,4-diazepan-5-ones and of their benzo-fused derivatives