List of works - Jarosław Sączewski

1-[(Imidazolidin-2-yl)imino]-1H-indoles as new hypotensive agents: synthesis and in vitro and in vivo biological studies

scientific article published on 27 August 2016

2-(4,5-Dihydro-1H-imidazol-2-yl)indazole (indazim) derivatives as selective I2 imidazoline receptor ligands ⬇️

scientific article published on October 1, 2003

2-Amino-4,5-dihydro-1H-imidazol-3-ium 7,8-dihydroimidazo[1,2-c][1,3,5]thiadiazine-2,4(6H)-dithione(1−) dimethylformamide disolvate

2-[(Arylmethoxy)imino]imidazolidines with potential biological activities

scientific article published in November 2009

Application of <i>Safirinium N</i>-Hydroxysuccinimide Esters to Derivatization of Peptides for High-Resolution Mass Spectrometry, Tandem Mass Spectrometry, and Fluorescent Labeling of Bacterial Cells

scientific article published on 17 December 2020

Carbon disulfide promoted reactions of 2-chloro-4,5-dihydro-imidazole with some N-nucleophiles

scientific article

Conjugate addition of nucleophiles to the vinyl function of 2-chloro-4-vinylpyrimidine derivatives

scientific article published on 19 March 2010

Copper(II)-assisted hydrolysis of cyclic ureas: Transformation of 1-(pyridin-2-yl)-2,3,7,8-tetrahydro-1 H -imidazo[2,1- b ][1,3,5]triazepin-5(6 H )-ones into N 1 -[1-(pyridin-2-yl)imidazolidin-2-ylidene]-ethane-1,2-diamine ligands

Experimental and theoretical studies on the tautomerism and reactivity of isoxazolo[3,4-b]quinolin-3(1H)-ones

First tandem nucleophilic addition–electrophilic amination reaction of Eschenmoser’s salts: synthesis of cyclic and spiro-fused hydrazonium salts

article

Hybrid Molecules Composed of 2,4-Diamino-1,3,5-triazines and 2-Imino-Coumarins and Coumarins. Synthesis and Cytotoxic Properties

scientific article published on 03 July 2018

Hydroxylamine-O-sulfonic Acid

Lipophilicity Determination of Antifungal Isoxazolo[3,4-b]pyridin-3(1H)-ones and Their N1-Substituted Derivatives with Chromatographic and Computational Methods

scientific article published on 26 November 2019

Lipophilicity Determination of Quaternary (Fluoro)Quinolones by Chromatographic and Theoretical Approaches

scientific article published on 24 October 2019

Modifications of quinolones and fluoroquinolones: hybrid compounds and dual-action molecules.

scientific article

N-(Imidazolidin-2-ylidene)-1-arylmethanamine Oxides: Synthesis, Structure and Pharmacological Evaluation

scientific article published on 14 November 2011

Synthesis and Antifungal Activity of Some 4,6-Dimethylisoxazolo[3,4- b]pyridin-3(1H)-one Derivatives.

scientific article published on 17 May 2016

Synthesis and Structure-Activity Relationship Analysis of 5-HT₇ Receptor Antagonists: Piperazin-1-yl Substituted Unfused Heterobiaryls.

scientific article published on 31 March 2016

Synthesis and biological evaluation of hybrid quinolone-based quaternary ammonium antibacterial agents

scientific article published on 27 June 2019

Synthesis and evaluation of dihydro-[1,2,4]triazolo[4,3-a]pyridin-2-ium carboxylates as fixed charge fluorescent derivatization reagents for MEKC and MS proteomic analyses

scientific article published in October 2020

Synthesis and in vitro anti-tumor activity of N-{1-[(3-thioxo-5,6-dihydroimidazo[2,1-c][1,2,4]thiadiazol-7-ylthio)thiocarbonyl]-2-imidazolidene}arylsulfonamides

scientific article published on 8 May 2006

Synthesis and molecular structure of (Z)-1H-purin-6-ylideneaminooxysulfonic acid: a possible secondary metabolite of adenine

Synthesis of 2,3-dihydroimidazo[1,2-a]pyrimidin-5(1H)-ones by the domino Michael addition retro-ene reaction of 2-alkoxyiminoimidazolidines and acetylene carboxylates

article

Synthesis of 4-substituted 2-(4-methylpiperazino)pyrimidines and quinazoline analogs as serotonin 5-HT 2A receptor ligands

scientific article published in November 2009

Synthesis of Heterocycles by Intramolecular Nucleophilic Substitution at an Electron-Deficient sp2 Nitrogen Atom

Synthesis of aza-aromatic hydroxylamine-O-sulfonates and their application to tandem nucleophilic addition–electrophilic 5-endo-trig cyclization

article

Synthesis of novel aryl(heteroaryl)sulfonyl ureas of possible biological interest

scientific article published on 26 February 2010

Synthesis, X-ray structure analysis and computational studies of novel bis(thiocarbamoyl) disulfides with non-covalent S⋯N and S⋯S interactions

Synthesis, crystal structure, 1H, 13C and 15N NMR studies, and biological evaluation of a new amidrazone-derived Au(III) complex

scientific article published in January 2019

Synthesis, molecular structure, and applications of 2-hydroxylamino-4,5-dihydroimidazolium-O-sulfonate to the synthesis of novel heterocyclic ring systems

scientific article

Synthesis, structural characterization and reactivity of new trisubstituted N1-acylamidrazones: solid state and solution studies

scientific article published in 2018

The Elusive Paal-Knorr Intermediates in the Trofimov Synthesis of Pyrroles: Experimental and Theoretical Studies

scientific article

The Tandem Mannich-Electrophilic Amination Reaction: a Versatile Platform for Fluorescent Probing and Labeling

scientific article published on 26 July 2013

List of works by Jarosław Sączewski

1-[(Imidazolidin-2-yl)imino]-1H-indoles as new hypotensive agents: synthesis and in vitro and in vivo biological studies

2-(4,5-Dihydro-1H-imidazol-2-yl)indazole (indazim) derivatives as selective I2 imidazoline receptor ligands ⬇️

2-Amino-4,5-dihydro-1H-imidazol-3-ium 7,8-dihydroimidazo[1,2-c][1,3,5]thiadiazine-2,4(6H)-dithione(1−) dimethylformamide disolvate

2-[(Arylmethoxy)imino]imidazolidines with potential biological activities

Application of <i>Safirinium N</i>-Hydroxysuccinimide Esters to Derivatization of Peptides for High-Resolution Mass Spectrometry, Tandem Mass Spectrometry, and Fluorescent Labeling of Bacterial Cells

Carbon disulfide promoted reactions of 2-chloro-4,5-dihydro-imidazole with some N-nucleophiles

Conjugate addition of nucleophiles to the vinyl function of 2-chloro-4-vinylpyrimidine derivatives

Copper(II)-assisted hydrolysis of cyclic ureas: Transformation of 1-(pyridin-2-yl)-2,3,7,8-tetrahydro-1 H -imidazo[2,1- b ][1,3,5]triazepin-5(6 H )-ones into N 1 -[1-(pyridin-2-yl)imidazolidin-2-ylidene]-ethane-1,2-diamine ligands

Experimental and theoretical studies on the tautomerism and reactivity of isoxazolo[3,4-b]quinolin-3(1H)-ones

First tandem nucleophilic addition–electrophilic amination reaction of Eschenmoser’s salts: synthesis of cyclic and spiro-fused hydrazonium salts

Hybrid Molecules Composed of 2,4-Diamino-1,3,5-triazines and 2-Imino-Coumarins and Coumarins. Synthesis and Cytotoxic Properties

Hydroxylamine-O-sulfonic Acid

Lipophilicity Determination of Antifungal Isoxazolo[3,4-b]pyridin-3(1H)-ones and Their N1-Substituted Derivatives with Chromatographic and Computational Methods

Lipophilicity Determination of Quaternary (Fluoro)Quinolones by Chromatographic and Theoretical Approaches

Modifications of quinolones and fluoroquinolones: hybrid compounds and dual-action molecules.

N-(Imidazolidin-2-ylidene)-1-arylmethanamine Oxides: Synthesis, Structure and Pharmacological Evaluation

Synthesis and Antifungal Activity of Some 4,6-Dimethylisoxazolo[3,4- b]pyridin-3(1H)-one Derivatives.

Synthesis and Structure-Activity Relationship Analysis of 5-HT₇ Receptor Antagonists: Piperazin-1-yl Substituted Unfused Heterobiaryls.

Synthesis and biological evaluation of hybrid quinolone-based quaternary ammonium antibacterial agents

Synthesis and evaluation of dihydro-[1,2,4]triazolo[4,3-a]pyridin-2-ium carboxylates as fixed charge fluorescent derivatization reagents for MEKC and MS proteomic analyses

Synthesis and in vitro anti-tumor activity of N-{1-[(3-thioxo-5,6-dihydroimidazo[2,1-c][1,2,4]thiadiazol-7-ylthio)thiocarbonyl]-2-imidazolidene}arylsulfonamides

Synthesis and molecular structure of (Z)-1H-purin-6-ylideneaminooxysulfonic acid: a possible secondary metabolite of adenine

Synthesis of 2,3-dihydroimidazo[1,2-a]pyrimidin-5(1H)-ones by the domino Michael addition retro-ene reaction of 2-alkoxyiminoimidazolidines and acetylene carboxylates

Synthesis of 4-substituted 2-(4-methylpiperazino)pyrimidines and quinazoline analogs as serotonin 5-HT 2A receptor ligands

Synthesis of Heterocycles by Intramolecular Nucleophilic Substitution at an Electron-Deficient sp2 Nitrogen Atom

Synthesis of aza-aromatic hydroxylamine-O-sulfonates and their application to tandem nucleophilic addition–electrophilic 5-endo-trig cyclization

Synthesis of novel aryl(heteroaryl)sulfonyl ureas of possible biological interest

Synthesis, X-ray structure analysis and computational studies of novel bis(thiocarbamoyl) disulfides with non-covalent S⋯N and S⋯S interactions

Synthesis, crystal structure, 1H, 13C and 15N NMR studies, and biological evaluation of a new amidrazone-derived Au(III) complex

Synthesis, molecular structure, and applications of 2-hydroxylamino-4,5-dihydroimidazolium-O-sulfonate to the synthesis of novel heterocyclic ring systems

Synthesis, structural characterization and reactivity of new trisubstituted N1-acylamidrazones: solid state and solution studies

The Elusive Paal-Knorr Intermediates in the Trofimov Synthesis of Pyrroles: Experimental and Theoretical Studies

The Tandem Mannich-Electrophilic Amination Reaction: a Versatile Platform for Fluorescent Probing and Labeling

The structure and theoretical study of 4-dimethylaminopyridinium N-(arylsulfonyl)carbamoylides