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List of works by František Trejtnar

3-Substituted N-Benzylpyrazine-2-carboxamide Derivatives: Synthesis, Antimycobacterial and Antibacterial Evaluation

scientific article published on 21 March 2017

99mTc demotate 1: biodistribution and elimination characteristics in rats

scientific article published on 01 June 2005

A comparison of in vitro methods for determining the membrane receptor expression in cell lines.

scientific article

A resurrection of 7-MEOTA: a comparison with tacrine.

scientific article published in October 2013

Analysis of accumulation of 99mTc-octreotide and 99mTc-EDDA/HYNIC-Tyr3-octreotide in the rat kidneys.

scientific article published in February 2004

Antibacterial Activity of Salicylanilide 4-(Trifluoromethyl)-benzoates

scientific article published on 25 March 2013

Antimicrobial activity of sulfonamides containing 5-chloro-2-hydroxybenzaldehyde and 5-chloro-2-hydroxybenzoic acid scaffold

scientific article published in April 2012

Azole antimycotics differentially affect rifampicin-induced pregnane X receptor-mediated CYP3A4 gene expression.

scientific article published on 12 November 2007

Biotransformation of anthelmintics and the activity of drug-metabolizing enzymes in the tapeworm Moniezia expansa

scientific article published on 6 November 2014

Bisamidate Prodrugs of 2-Substituted 9-[2-(Phosphonomethoxy)ethyl]adenine (PMEA, adefovir) as Selective Inhibitors of Adenylate Cyclase Toxin from Bordetella pertussis.

scientific article

Corrigendum to "Novel salicylanilides from 4,5-dihalogenated salicylic acids: Synthesis, antimicrobial activity and cytotoxicity" [Bioorg. Med. Chem. 25 (2017) 1524-1532].

scientific article published on 10 March 2017

Design, synthesis and anti-mycobacterial evaluation of some new N-phenylpyrazine-2-carboxamides

Determination of receptor protein binding site specificity and relative binding strength using a time-resolved competition assay.

scientific article published on 29 July 2014

Distribution, elimination, and renal handling of (99m)technetium-Demogastrin 1

scientific article published on 01 March 2012

Entecavir Interacts with Influx Transporters hOAT1, hCNT2, hCNT3, but Not with hOCT2: The Potential for Renal Transporter-Mediated Cytotoxicity and Drug-Drug Interactions

scientific article

Expression of organic cation transporter 1 (OCT1): unique patterns of indirect regulation by nuclear receptors and hepatospecific gene regulation

scientific article

Highly sensitive fast determination of entecavir in rat urine by means of hydrophilic interaction chromatography–ultra-high-performance liquid chromatography–tandem mass spectrometry

scientific article published on 01 April 2012

Honey flavonoids inhibit hOATP2B1 and hOATP1A2 transporters and hOATP-mediated rosuvastatin cell uptake in vitro

scientific article

How to address the sample preparation of hydrophilic compounds: Determination of entecavir in plasma and plasma ultrafiltrate with novel extraction sorbents

scientific article

In vitro comparison of renal handling and uptake of two somatostatin receptor-specific peptides labeled with indium-111.

scientific article published in December 2008

In vitro evaluation of concentration, labeling effectiveness and stability for 131 I-labeled radioimmunoassay ligand using real-time detection technology.

scientific article published on 13 December 2016

Interaction of soy isoflavones and their main metabolites with hOATP2B1 transporter

scientific article published on 22 June 2018

Interactions with selected drug renal transporters and transporter-mediated cytotoxicity in antiviral agents from the group of acyclic nucleoside phosphonates.

scientific article published on 13 July 2013

Iron reduction potentiates hydroxyl radical formation only in flavonols.

scientific article published on 14 July 2012

Modulatory effects of quercetin and rutin on the activity, expression and inducibility of CYP1A1 in intestinal HCT-8 cells.

scientific article

Novel derivatives of nitro-substituted salicylic acids: Synthesis, antimicrobial activity and cytotoxicity.

scientific article published on 24 October 2015

Novel salicylanilides from 4,5-dihalogenated salicylic acids: Synthesis, antimicrobial activity and cytotoxicity.

scientific article

Possible use of excretion of tubular epithelial cells for the study of the nephrotoxic effect of xenobiotics

scientific article published on 01 December 1996

Renal handling of amphotericin B and amphotericin B-deoxycholate and potential renal drug-drug interactions with selected antivirals.

scientific article

Salicylanilide diethyl phosphates: synthesis, antimicrobial activity and cytotoxicity.

scientific article published on 12 December 2013

Sex differences in stereospecificity of oracin reductases in ratin vitro andin vivo

scientific article published on 01 January 1999

Stereoselective pharmacokinetics and metabolism of flobufen in guinea pigs.

scientific article published in October 2003

Stereoselective pharmacokinetics of flobufen in rats

scientific article published on 01 January 1999

Steviol, an aglycone of steviol glycoside sweeteners, interacts with the pregnane X (PXR) and aryl hydrocarbon (AHR) receptors in detoxification regulation

scientific article published on 5 September 2017

Study of the biotransformation of a potential benzo[c]fluorene antineoplastic using high-performance liquid chromatography with high-speed-scanning ultraviolet detection

scientific article published on 01 May 1996

Sulfadiazine Salicylaldehyde-Based Schiff Bases: Synthesis, Antimicrobial Activity and Cytotoxicity.

scientific article

Synthesis and antimycobacterial evaluation of pyrazinamide derivatives with benzylamino substitution.

scientific article published on 27 November 2012

Synthesis and biological activity of new salicylanilide N,N-disubstituted carbamates and thiocarbamates.

scientific article published on 5 June 2014

Synthesis and in vitro antimycobacterial activity of 2-methoxybenzanilides and their thioxo analogues

scientific article published on 04 August 2012

Synthesis and in vitro antimycobacterial and isocitrate lyase inhibition properties of novel 2-methoxy-2′-hydroxybenzanilides, their thioxo analogues and benzoxazoles

scientific article published on 16 August 2012

Synthesis and in vitro evaluation of new derivatives of 2-substituted-6-fluorobenzo[d]thiazoles as cholinesterase inhibitors.

scientific article published on February 2013

Synthesis of readily available fluorophenylalanine derivatives and investigation of their biological activity

scientific article published on 21 February 2017

The effect of chelator type on in vitro receptor binding and stability in 177Lu-labeled cetuximab and panitumumab.

scientific article published on 29 May 2014

The in vivo disposition and in vitro transmembrane transport of two model radiometabolites of DOTA-conjugated receptor-specific peptides labelled with (177) Lu.

scientific article published on 3 November 2015

The involvement of selected membrane transport mechanisms in the cellular uptake of (177)Lu-labeled bombesin, somatostatin and gastrin analogues.

scientific article

The pregnane X receptor down-regulates organic cation transporter 1 (SLC22A1) in human hepatocytes by competing for ("squelching") SRC-1 coactivator

scientific article published on 27 February 2016

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