List of works - Frédéric Rodriguez

Asymmetric Synthesis and Binding Study of New Long-Chain HPA-12 Analogues as Potent Ligands of the Ceramide Transfer Protein CERT.

scientific article published on 31 March 2016

Chemical synthesis and biological evaluation of triazole derivatives as inhibitors of InhA and antituberculosis agents.

scientific article published on 23 March 2012

Design of granulatimide and isogranulatimide analogues as potential Chk1 inhibitors: Study of amino-platforms for their synthesis.

scientific article

Design, chemical synthesis of 3-(9H-fluoren-9-yl)pyrrolidine-2,5-dione derivatives and biological activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis

scientific article published on 2 October 2013

Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growth.

scientific article published on 20 June 2015

Electrooptics studies of Escherichia coli electropulsation: orientation, permeabilization, and gene transfer.

scientific article published on November 1998

Iminosugar-based ceramide mimicry for the design of new CERT START domain ligands.

scientific article published on 14 February 2017

Irreversible inhibition of aldolase by a phosphorylated alpha-dicarbonyl compound

scientific article published on 01 February 2008

Modification of endothelial nitric oxide synthase by 4-oxo-2(E)-nonenal(ONE) in preeclamptic placentas

scientific article published on 16 July 2019

New potent bisubstrate inhibitors of histone acetyltransferase p300: design, synthesis and biological evaluation

scientific article published on 30 November 2010

Pyrrolidinone and pyrrolidine derivatives: Evaluation as inhibitors of InhA and Mycobacterium tuberculosis.

scientific article published on 16 July 2016

Selective Targeting of the Interconversion between Glucosylceramide and Ceramide by Scaffold Tailoring of Iminosugar Inhibitors

scientific article published on 19 January 2019

Self-association processes involving anthracene labeled phosphatidylcholines in model membrane.

scientific article published in February 1995

Synthesis and biological activities of triazole derivatives as inhibitors of InhA and antituberculosis agents

scientific article published on 16 September 2011

Synthesis and evaluation of α-ketotriazoles and α,β-diketotriazoles as inhibitors of Mycobacterium tuberculosis.

scientific article published on 8 July 2013

Synthesis and in vitro antiproliferative activity of amido and amino analogues of the marine alkaloid isogranulatimide.

scientific article

Synthesis of 3-heteryl substituted pyrrolidine-2,5-diones via catalytic Michael reaction and evaluation of their inhibitory activity against InhA and Mycobacterium tuberculosis

scientific article published on 04 November 2013

The CERT antagonist HPA-12: first practical synthesis and individual binding evaluation of the four stereoisomers.

scientific article

Watson-Crick base-pairing properties of nucleic acid analogues with stereocontrolled alpha and beta torsion angles (alpha,beta-D-CNAs)

scientific article published on 01 May 2006

List of works by Frédéric Rodriguez

Asymmetric Synthesis and Binding Study of New Long-Chain HPA-12 Analogues as Potent Ligands of the Ceramide Transfer Protein CERT.

Chemical synthesis and biological evaluation of triazole derivatives as inhibitors of InhA and antituberculosis agents.

Design of granulatimide and isogranulatimide analogues as potential Chk1 inhibitors: Study of amino-platforms for their synthesis.

Design, chemical synthesis of 3-(9H-fluoren-9-yl)pyrrolidine-2,5-dione derivatives and biological activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis

Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growth.

Electrooptics studies of Escherichia coli electropulsation: orientation, permeabilization, and gene transfer.

Iminosugar-based ceramide mimicry for the design of new CERT START domain ligands.

Irreversible inhibition of aldolase by a phosphorylated alpha-dicarbonyl compound

Modification of endothelial nitric oxide synthase by 4-oxo-2(E)-nonenal(ONE) in preeclamptic placentas

New potent bisubstrate inhibitors of histone acetyltransferase p300: design, synthesis and biological evaluation

Pyrrolidinone and pyrrolidine derivatives: Evaluation as inhibitors of InhA and Mycobacterium tuberculosis.

Selective Targeting of the Interconversion between Glucosylceramide and Ceramide by Scaffold Tailoring of Iminosugar Inhibitors

Self-association processes involving anthracene labeled phosphatidylcholines in model membrane.

Synthesis and biological activities of triazole derivatives as inhibitors of InhA and antituberculosis agents

Synthesis and evaluation of α-ketotriazoles and α,β-diketotriazoles as inhibitors of Mycobacterium tuberculosis.

Synthesis and in vitro antiproliferative activity of amido and amino analogues of the marine alkaloid isogranulatimide.

Synthesis of 3-heteryl substituted pyrrolidine-2,5-diones via catalytic Michael reaction and evaluation of their inhibitory activity against InhA and Mycobacterium tuberculosis

The CERT antagonist HPA-12: first practical synthesis and individual binding evaluation of the four stereoisomers.

Watson-Crick base-pairing properties of nucleic acid analogues with stereocontrolled alpha and beta torsion angles (alpha,beta-D-CNAs)