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List of works by Richard M van Rijn

A FLIPR assay for evaluating agonists and antagonists of GPCR heterodimers.

scientific article

A Review of the Therapeutic Potential of Recently Developed G Protein-Biased Kappa Agonists

article

A critical evaluation of TRPA1-mediated locomotor behavior in zebrafish as a screening tool for novel anti-nociceptive drug discovery

scientific article published on 20 February 2019

A non-convulsant delta-opioid receptor agonist, KNT-127, reduces cortical spreading depression and nitroglycerin-induced allodynia

scientific article published on 16 December 2020

Adolescent intake of caffeinated energy drinks does not affect adult alcohol consumption in C57BL/6 and BALB/c mice

scientific article published on 24 May 2016

An integrated perspective on diabetic, alcoholic, and drug-induced neuropathy, etiology, and treatment in the US.

scientific article

Anti-analgesic effect of the mu/delta opioid receptor heteromer revealed by ligand-biased antagonism

scientific article

Arrestin recruitment and signaling by G protein-coupled receptor heteromers

scientific article published on 09 November 2018

Behavioral Characterization of β-Arrestin 1 Knockout Mice in Anxiety-Like and Alcohol Behaviors.

scientific article

Commonly Used Anesthesia/Euthanasia Methods for Brain Collection Differentially Impact MAPK Activity in Male and Female C57BL/6 Mice

scientific article published on 28 March 2019

Critical Role for Gi/o-Protein Activity in the Dorsal Striatum in the Reduction of Voluntary Alcohol Intake in C57Bl/6 Mice.

scientific article published on 5 April 2018

Delta Opioid Pharmacology in Relation to Alcohol Behaviors.

scientific article

Discovery of naturally occurring splice variants of the rat histamine H3 receptor that act as dominant-negative isoforms

scientific article

Drug screening with zebrafish visual behavior identifies carvedilol as a potential treatment for an autosomal dominant form of retinitis pigmentosa

scientific article published on 01 June 2021

Emergence of functional spinal delta opioid receptors after chronic ethanol exposure

scientific article

Functional histamine H3 and adenosine A2A receptor heteromers in recombinant cells and rat striatum.

scientific article published on 4 December 2017

G protein-biased kratom-alkaloids and synthetic carfentanil-amide opioids as potential treatments for alcohol use disorder

scientific article published on 24 January 2020

Identification of a selective small-molecule inhibitor of type 1 adenylyl cyclase activity with analgesic properties.

scientific article published on 21 February 2017

Involvement of delta opioid receptors in alcohol withdrawal-induced mechanical allodynia in male C57BL/6 mice.

scientific article published on 21 August 2016

Isolation and Pharmacological Characterization of Six Opioidergic Picralima nitida Alkaloids

scientific article published on 16 December 2020

Isolation of acetylcholinesterase inhibitory alkaloids from Nerine bowdenii.

scientific article published in February 2010

Methadone antinociception is dependent on peripheral opioid receptors

scientific article

Oligomerization of recombinant and endogenously expressed human histamine H(4) receptors

scientific article published on 27 April 2006

Optimization of a 1,3,4-oxadiazole series for inhibition of Ca2+/calmodulin-stimulated activity of adenylyl cyclases 1 and 8 for the treatment of chronic pain

scientific article published on 16 November 2018

Pharmacological traits of delta opioid receptors: pitfalls or opportunities?

scientific article published on 07 May 2013

Repeated Use of the Psychoactive Substance Ethylphenidate Impacts Neurochemistry and Reward Learning in Adolescent Male and Female Mice

scientific article published on 19 February 2019

Rubiscolins are naturally occurring G protein-biased delta opioid receptor peptides

scientific article published on 24 December 2018

Selection of DNA-Encoded Libraries to Protein Targets within and on Living Cells

scientific article published on 22 October 2019

Synthesis and structure-activity relationships of indole and benzimidazole piperazines as histamine H(4) receptor antagonists.

scientific article published on November 2004

The Meta-Position of Phe4 in Leu-Enkephalin Regulates Potency, Selectivity, Functional Activity, and Signaling Bias at the Delta and Mu Opioid Receptors

scientific article published on 12 December 2019

The delta(1) opioid receptor is a heterodimer that opposes the actions of the delta(2) receptor on alcohol intake

scientific article published on 03 July 2009

The only way is up: preventing opioid tolerance by promoting cell surface expression of MOR-DOR heterodimers?

scientific article

Unique Behavioral and Neurochemical Effects Induced by Repeated Adolescent Consumption of Caffeine-Mixed Alcohol in C57BL/6 Mice

scientific article (publication date: 2016)

β-Arrestin 2 dependence of δ opioid receptor agonists is correlated with alcohol intake

scientific article published on 27 October 2015

β-Arrestin-Dependent Dopaminergic Regulation of Calcium Channel Activity in the Axon Initial Segment.

scientific article

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