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List of works by Michal Bista

1,4-Thienodiazepine-2,5-diones via MCR (I): synthesis, virtual space and p53-Mdm2 activity.

scientific article published on 18 May 2010

Enabling large-scale design, synthesis and validation of small molecule protein-protein antagonists

scientific article

Enzymatic activity of the Staphylococcus aureus SplB serine protease is induced by substrates containing the sequence Trp-Glu-Leu-Gln

scientific article

Lifeact: a versatile marker to visualize F-actin

scientific article (publication date: July 2008)

MDMX contains an autoinhibitory sequence element

scientific article published on 14 October 2013

MTH1 Substrate Recognition--An Example of Specific Promiscuity

scientific article

Mapping the sugar dependency for rational generation of a DNA-RNA hybrid-guided Cas9 endonuclease.

scientific article published on 20 November 2017

On the mechanism of action of SJ-172550 in inhibiting the interaction of MDM4 and p53

scientific article

Positioning High-Throughput CETSA in Early Drug Discovery through Screening against B-Raf and PARP1

scientific article published on 13 December 2018

Potent and Selective Inhibitors of MTH1 Probe Its Role in Cancer Cell Survival

scientific article

Quantifying the relationship between inhibition of VEGFR-2, drug-induced blood pressure elevation and hypertension.

scientific article published on 21 November 2017

Robust NMR screening for lead compounds using tryptophan-containing proteins.

scientific article published in June 2009

Robust generation of lead compounds for protein-protein interactions by computational and MCR chemistry: p53/Hdm2 antagonists.

scientific article published on July 2010

Structural and functional characterization of SplA, an exclusively specific protease of Staphylococcus aureus

scientific article

Transient Protein States in Designing Inhibitors of the MDM2-p53 Interaction

scientific article

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