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List of works by Yasuaki Anami

A mixed population of antagonist and agonist binding conformers in a single crystal explains partial agonism against vitamin D receptor: active vitamin D analogues with 22R-alkyl group

scientific article

Apo- and Antagonist-Binding Structures of Vitamin D Receptor Ligand-Binding Domain Revealed by Hybrid Approach Combining Small-Angle X-ray Scattering and Molecular Dynamics.

scientific article

Development of vitamin D analogs modulating the pocket structure of vitamin D receptor

scientific article published on January 2014

Disrupting LILRB4/APOE Interaction by an Efficacious Humanized Antibody Reverses T-cell Suppression and Blocks AML Development

scientific article published on 18 June 2019

Enzymatic conjugation using branched linkers for constructing homogeneous antibody-drug conjugates with high potency.

scientific article

Fine tuning of agonistic/antagonistic activity for vitamin D receptor by 22-alkyl chain length of ligands: 22S-Hexyl compound unexpectedly restored agonistic activity

scientific article

Glutamic acid-valine-citrulline linkers ensure stability and efficacy of antibody-drug conjugates in mice.

scientific article

Helix12-Stabilization Antagonist of Vitamin D Receptor

scientific article

Identification of the Histidine Residue in Vitamin D Receptor That Covalently Binds to Electrophilic Ligands

scientific article published on 11 July 2018

LILRB4-Targeting Antibody-Drug Conjugates for the Treatment of Acute Myeloid Leukemia

scientific article published on 02 September 2020

SRC2-3 binds to vitamin D receptor with high sensitivity and strong affinity

scientific article published on 14 November 2016

Total Synthesis of the Monomeric Unit of Lomaiviticin A

scientific article published on 13 November 2020

Transglutaminase-Mediated Conjugations

scientific article published on 01 January 2020

Truncated Autoinducing Peptide Conjugates Selectively Recognize and Kill Staphylococcus aureus.

scientific article published on 3 February 2017

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