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List of works by William P Katt

A tale of two glutaminases: homologous enzymes with distinct roles in tumorigenesis

scientific article published on 23 January 2017

A unique metabolic dependency for liver cancer stem cells

scientific article published on 20 December 2018

Amorphous Quantum Nanomaterials

scientific article published on 05 December 2018

An oxazole-based small-molecule Stat3 inhibitor modulates Stat3 stability and processing and induces antitumor cell effects

scientific article published on 01 December 2007

Characterization of the interactions of potent allosteric inhibitors with glutaminase C, a key enzyme in cancer cell glutamine metabolism.

scientific article published on 9 January 2018

Design and evaluation of novel glutaminase inhibitors

scientific article

Dibenzophenanthridines as inhibitors of glutaminase C and cancer cell proliferation.

scientific article published on 11 April 2012

Glutaminase regulation in cancer cells: a druggable chain of events.

scientific article published on 16 October 2013

Isoform selective inhibition of STAT1 or STAT3 homo-dimerization via peptidomimetic probes: structural recognition of STAT SH2 domains

scientific article

Less than the sum of its parts, a leinamycin precursor has superior properties

scientific article published on 23 June 2015

Mechanistic Basis of Glutaminase Activation: A KEY ENZYME THAT PROMOTES GLUTAMINE METABOLISM IN CANCER CELLS

scientific article

New developments in PEST shape/property hybrid descriptors.

scientific article published in February 2003

Opening up about Tissue Transglutaminase: When Conformation Matters More than Enzymatic Activity

article

Patents targeting the Warburg effect for cancer therapy: an interview with William P Katt

scientific article published on 01 January 2020

Potent, Plasmodium-selective farnesyltransferase inhibitors that arrest the growth of malaria parasites: structure-activity relationships of ethylenediamine-analogue scaffolds and homology model validation.

scientific article

Simultaneously targeting tissue transglutaminase and kidney type glutaminase sensitizes cancer cells to acid toxicity and offers new opportunities for therapeutic intervention

scientific article

Synthesis and biological evaluation of a 5-6-5 imidazole-phenyl-thiazole based alpha-helix mimetic

scientific article published on January 2009

Targeting Therapy Resistance: When Glutamine Catabolism Becomes Essential

scientific article published on 01 May 2018

Targeting amino acid metabolism for cancer therapy

scientific article published on 14 December 2016

Targeting protein-protein interactions: suppression of Stat3 dimerization with rationally designed small-molecule, nonpeptidic SH2 domain binders

scientific article

The diamond anniversary of tissue transglutaminase: a protein of many talents

scientific article published on 31 January 2018