List of works - Vincent Lisowski

3D-QSAR and docking studies of selective GSK-3beta inhibitors. Comparison with a thieno[2,3-b]pyrrolizinone derivative, a new potential lead for GSK-3beta ligands.

scientific article published in May 2005

An efficient synthesis of pyrido-imidazodiazepinediones

Chemical optimization of new ligands of the low-density lipoprotein receptor as potential vectors for central nervous system targeting.

scientific article published on 14 February 2012

Chemistry of Ring-Fused Oxazine-2,4-diones

Cross-Claisen Condensation ofN-Fmoc-Amino Acids - A Short Route to Heterocyclic γ-Amino Acids

Cyclic Peptides with a Diversely Substituted Guanidine Bridge: Solid-Phase Synthesis and Structural Analysis

article

Design and characterization of a new cell-permeant inhibitor of the beta-secretase BACE1.

scientific article

Design, synthesis and antiproliferative activity of tripentones: a new series of antitubulin agents.

scientific article published in August 2001

Efficient one-pot microwave-assisted synthesis of 3-(thien-3-yl)imidazolidine-2,4-dione analogs

Efficient synthesis of novel 3-(Het)arylanthranilic acids via a suzuki cross-coupling reaction of 7-iodoisatin with (Het)arylboronic acids in water

scientific article published on 01 June 2000

Formulation of sustained release nanoparticles loaded with a tripentone, a new anticancer agent.

scientific article published on 24 May 2006

From Thienodiazepinediones to Thienopyridinones: Flexible Synthesis of Substituted Thieno[3,2-e][1,4]diazepinones and 6-Aminothieno[3,2-b]pyridinones

Further characterization of a putative serine protease contributing to the γ-secretase cleavage of β-amyloid precursor protein

scholarly article by Marine Peuchmaur published in February 2013

Helical Oligomers of Thiazole-Based γ-Amino Acids: Synthesis and Structural Studies

scientific article published on 25 April 2013

Imidazopyridine-fused [1,3]-diazepinones part 2: Structure-activity relationships and antiproliferative activity against melanoma cells.

scientific article published on 11 November 2016

Imidazopyridine-fused [1,3]-diazepinones: synthesis and antiproliferative activity.

scientific article published on 30 January 2014

Inhibitors of kallikrein-related peptidases: An overview.

scientific article

Pyrido-imidazodiazepinones as a new class of reversible inhibitors of human kallikrein 7.

scientific article

Reactivity Study of 1H-Thieno[3,2-d][1,3]oxazine-2,4-dione toward the Synthesis of Bicyclic 3,4-Dihydro-1H-thieno[3,2-e][1,4]diazepine-2,5-dione Analogues

Regio-Controlled Nucleophilic Attack of 3-Thiaisatoic Anhydride by α-Amino Acids: One-Pot Synthesis of 3-(2-Thienyl)imidazolidine-2,4-dione and 3,4-Substituted Thieno[2,3-e][1,4]diazepine-2,5-dione Analogues

Selective C-acylation of 2-aminoimidazo[1,2-a]pyridine: application to the synthesis of imidazopyridine-fused [1,3]diazepinones

scientific article

Solid phase synthesis of mono- or disubstituted arginine containing peptides from an isothiocitrulline precursor

Solid-Phase Synthesis of Isocoumarins: A Traceless Halocyclization Approach

Structure-Activity Relationships of JMV4463, a Vectorized Cathepsin D Inhibitor with Antiproliferative Properties: The Unique Role of the AMPA-Based Vector

scientific article published on 07 December 2015

Synthesis and biological evaluation as AChE inhibitors of new indanones and thiaindanones related to donepezil.

scientific article published on 30 August 2005

Synthesis and biological evaluation of novel pyrrolopyrrolizinones as anticancer agents

scientific article published on 29 September 2006

Synthesis and biological evaluation of thienopyrrolizines, a new family of CDK/GSK-3 inhibitors.

scientific article published in December 2004

Synthesis and initial results for MAO-B inhibition by new N-propargyl-3-pyrrol-1-ylindanamine derivatives, analogues of rasagiline

scientific article published in April 2003

Synthesis and reactivity of pyrrolo[3,2-d][1,3]oxazine-2,4-dione. Access to new pyrrolo[3,2-e][1,4]diazepine-2,5-diones

Synthesis of Thieno[3,2-e][1,4]diazepin-2-ones: Application of an Uncatalysed Pictet-Spengler Reaction

Synthesis of new 2-(aminomethyl)-4-phenylpyrrolo[1,2-a]-quinoxalines and their preliminary in-vivo central dopamine antagonist activity evaluation in mice

scientific article

Synthesis of new aromatic pyrrolo[2,1-c] [1,4]benzodiazepines and pyrrolo[1,2-a]thieno[3,2-e] [1,4]diazepines as anti-tumoral agents

scientific article published on December 2002

Synthetic therapeutic peptides: science and market

scientific article published on 30 October 2009

The HslV Protease from and Its Activation by C-terminal HslU Peptides ⬇️

scientific article published on 26 February 2019

Thiazole-Based γ-Building Blocks as Reverse-Turn Mimetic to Design a Gramicidin S Analogue: Conformational and Biological Evaluation

scientific article published on 25 March 2014

Thieno[3,2-e]diazepinediones and 3-thienylimidazolidinediones syntheses: regio-controlled ring opening of thiaisatoic anhydride by alpha-amino acids.

scientific article published in January 2009

Valuable Versatile Reactivity of Thiaisatoic Anhydrides: Expedient SolidPhase Synthesis of Thieno[1,4]diazepine-2,5-diones

[Onguent du Bec or king's drugs?].

scientific article

List of works by Vincent Lisowski

3D-QSAR and docking studies of selective GSK-3beta inhibitors. Comparison with a thieno[2,3-b]pyrrolizinone derivative, a new potential lead for GSK-3beta ligands.

An efficient synthesis of pyrido-imidazodiazepinediones

Chemical optimization of new ligands of the low-density lipoprotein receptor as potential vectors for central nervous system targeting.

Chemistry of Ring-Fused Oxazine-2,4-diones

Cross-Claisen Condensation ofN-Fmoc-Amino Acids - A Short Route to Heterocyclic γ-Amino Acids

Cyclic Peptides with a Diversely Substituted Guanidine Bridge: Solid-Phase Synthesis and Structural Analysis

Design and characterization of a new cell-permeant inhibitor of the beta-secretase BACE1.

Design, synthesis and antiproliferative activity of tripentones: a new series of antitubulin agents.

Efficient one-pot microwave-assisted synthesis of 3-(thien-3-yl)imidazolidine-2,4-dione analogs

Efficient synthesis of novel 3-(Het)arylanthranilic acids via a suzuki cross-coupling reaction of 7-iodoisatin with (Het)arylboronic acids in water

Formulation of sustained release nanoparticles loaded with a tripentone, a new anticancer agent.

From Thienodiazepinediones to Thienopyridinones: Flexible Synthesis of Substituted Thieno[3,2-e][1,4]diazepinones and 6-Aminothieno[3,2-b]pyridinones

Further characterization of a putative serine protease contributing to the γ-secretase cleavage of β-amyloid precursor protein

Helical Oligomers of Thiazole-Based γ-Amino Acids: Synthesis and Structural Studies

Imidazopyridine-fused [1,3]-diazepinones part 2: Structure-activity relationships and antiproliferative activity against melanoma cells.

Imidazopyridine-fused [1,3]-diazepinones: synthesis and antiproliferative activity.

Inhibitors of kallikrein-related peptidases: An overview.

Pyrido-imidazodiazepinones as a new class of reversible inhibitors of human kallikrein 7.

Reactivity Study of 1H-Thieno[3,2-d][1,3]oxazine-2,4-dione toward the Synthesis of Bicyclic 3,4-Dihydro-1H-thieno[3,2-e][1,4]diazepine-2,5-dione Analogues

Regio-Controlled Nucleophilic Attack of 3-Thiaisatoic Anhydride by α-Amino Acids: One-Pot Synthesis of 3-(2-Thienyl)imidazolidine-2,4-dione and 3,4-Substituted Thieno[2,3-e][1,4]diazepine-2,5-dione Analogues

Selective C-acylation of 2-aminoimidazo[1,2-a]pyridine: application to the synthesis of imidazopyridine-fused [1,3]diazepinones

Solid phase synthesis of mono- or disubstituted arginine containing peptides from an isothiocitrulline precursor

Solid-Phase Synthesis of Isocoumarins: A Traceless Halocyclization Approach

Structure-Activity Relationships of JMV4463, a Vectorized Cathepsin D Inhibitor with Antiproliferative Properties: The Unique Role of the AMPA-Based Vector

Synthesis and biological evaluation as AChE inhibitors of new indanones and thiaindanones related to donepezil.

Synthesis and biological evaluation of novel pyrrolopyrrolizinones as anticancer agents

Synthesis and biological evaluation of thienopyrrolizines, a new family of CDK/GSK-3 inhibitors.

Synthesis and initial results for MAO-B inhibition by new N-propargyl-3-pyrrol-1-ylindanamine derivatives, analogues of rasagiline

Synthesis and reactivity of pyrrolo[3,2-d][1,3]oxazine-2,4-dione. Access to new pyrrolo[3,2-e][1,4]diazepine-2,5-diones

Synthesis of Thieno[3,2-e][1,4]diazepin-2-ones: Application of an Uncatalysed Pictet-Spengler Reaction

Synthesis of new 2-(aminomethyl)-4-phenylpyrrolo[1,2-a]-quinoxalines and their preliminary in-vivo central dopamine antagonist activity evaluation in mice

Synthesis of new aromatic pyrrolo[2,1-c] [1,4]benzodiazepines and pyrrolo[1,2-a]thieno[3,2-e] [1,4]diazepines as anti-tumoral agents

Synthetic therapeutic peptides: science and market

The HslV Protease from and Its Activation by C-terminal HslU Peptides ⬇️

Thiazole-Based γ-Building Blocks as Reverse-Turn Mimetic to Design a Gramicidin S Analogue: Conformational and Biological Evaluation

Thieno[3,2-e]diazepinediones and 3-thienylimidazolidinediones syntheses: regio-controlled ring opening of thiaisatoic anhydride by alpha-amino acids.

Valuable Versatile Reactivity of Thiaisatoic Anhydrides: Expedient SolidPhase Synthesis of Thieno[1,4]diazepine-2,5-diones

[Onguent du Bec or king's drugs?].