List of works - Ajiroghene Thomas

1,2,4-triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A₃ receptor antagonists. Synthesis, structure-affinity relationships and molecular modeling studies.

scientific article published on 27 November 2014

8-(2-Furyl)adenine derivatives as A₂A adenosine receptor ligands.

scientific article published on 17 October 2013

A Novel Class of Dopamine D4 Receptor Ligands Bearing an Imidazoline Nucleus

scientific article published on 15 March 2016

Antiproliferative evaluation of isofuranodiene on breast and prostate cancer cell lines.

scientific article published on 22 May 2014

Different efficacy of adenosine and NECA derivatives at the human A3 adenosine receptor: insight into the receptor activation switch.

scientific article

Evaluation of adenine as scaffold for the development of novel P2X3 receptor antagonists.

scientific article published on 24 April 2013

Evidence for the existence of a specific g protein-coupled receptor activated by guanosine

scientific article published on 15 April 2011

Exploring the 7-oxo-thiazolo[5,4-d]pyrimidine core for the design of new human adenosine A3 receptor antagonists. Synthesis, molecular modeling studies and pharmacological evaluation

scientific article published on 04 April 2015

Innovative functional cAMP assay for studying G protein-coupled receptors: application to the pharmacological characterization of GPR17.

scientific article

Medicinal chemistry of P2X receptors: agonists and orthosteric antagonists.

scientific article

Molecular modeling study on potent and selective adenosine A(3) receptor agonists.

scientific article published on 22 September 2010

Neuropeptide S receptor: recent updates on nonpeptide antagonist discovery.

scientific article published on 30 March 2011

Purinergic P2X receptors: structural models and analysis of ligand-target interaction.

scientific article published on 25 October 2014

Simulation and Comparative Analysis of Different Binding Modes of Non-nucleoside Agonists at the A2A Adenosine Receptor.

scientific article published on 28 June 2016

Simulation and comparative analysis of binding modes of nucleoside and non-nucleoside agonists at the A2B adenosine receptor

scientific article published on 20 December 2013

The Length and Flexibility of the 2-Substituent of 9-Ethyladenine Derivatives Modulate Affinity and Selectivity for the Human A2A Adenosine Receptor

scientific article published on April 2016

List of works by Ajiroghene Thomas

1,2,4-triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A₃ receptor antagonists. Synthesis, structure-affinity relationships and molecular modeling studies.

8-(2-Furyl)adenine derivatives as A₂A adenosine receptor ligands.

A Novel Class of Dopamine D4 Receptor Ligands Bearing an Imidazoline Nucleus

Antiproliferative evaluation of isofuranodiene on breast and prostate cancer cell lines.

Different efficacy of adenosine and NECA derivatives at the human A3 adenosine receptor: insight into the receptor activation switch.

Evaluation of adenine as scaffold for the development of novel P2X3 receptor antagonists.

Evidence for the existence of a specific g protein-coupled receptor activated by guanosine

Exploring the 7-oxo-thiazolo[5,4-d]pyrimidine core for the design of new human adenosine A3 receptor antagonists. Synthesis, molecular modeling studies and pharmacological evaluation

Innovative functional cAMP assay for studying G protein-coupled receptors: application to the pharmacological characterization of GPR17.

Medicinal chemistry of P2X receptors: agonists and orthosteric antagonists.

Molecular modeling study on potent and selective adenosine A(3) receptor agonists.

Neuropeptide S receptor: recent updates on nonpeptide antagonist discovery.

Purinergic P2X receptors: structural models and analysis of ligand-target interaction.

Simulation and Comparative Analysis of Different Binding Modes of Non-nucleoside Agonists at the A2A Adenosine Receptor.

Simulation and comparative analysis of binding modes of nucleoside and non-nucleoside agonists at the A2B adenosine receptor

The Length and Flexibility of the 2-Substituent of 9-Ethyladenine Derivatives Modulate Affinity and Selectivity for the Human A2A Adenosine Receptor