List of works - Ayumu Niida

A Short-Length Peptide YY Analogue with Anorectic Effect in Mice.

scientific article published on 18 May 2017

A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres

scientific article published on 28 September 2006

Antiobesity Effect of a Short-Length Peptide YY Analogue after Continuous Administration in Mice.

scientific article published in May 2017

Antiobesity and emetic effects of a short-length peptide YY analog and its PEGylated and alkylated derivatives

scientific article published on 8 December 2017

Crystal Structure of a Human K-Ras G12D Mutant in Complex with GDP and the Cyclic Inhibitory Peptide KRpep-2d.

scientific article published on 10 May 2017

Design and synthesis of downsized metastin (45-54) analogs with maintenance of high GPR54 agonistic activity

scientific article published on 18 October 2005

Diastereoselective Synthesis of ψ[(E)-CHCMe]- and ψ[(Z)-CHCMe]-Type Dipeptide Isosteres by Organocopper-Mediatedanti-SN2‘ Reaction

scientific article published on 01 April 2002

Diastereoselective Synthesis ofψ[(E)-CMeCH]- andψ[(E)-CMeCMe]- Type Dipeptide Isosteres Based on Organocopper-Mediatedanti-SN2‘ Reaction

scientific article published on 01 April 2002

Diastereoselective synthesis of new psi[(E)-CH=CMe]- and psi[(Z)-CH=CMe]-type alkene dipeptide isosteres by organocopper reagents and application to conformationally restricted cyclic RGD peptidomimetics.

scientific article published in August 2002

Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres

scientific article published on 01 January 2007

Highly potent antiobesity effect of a short-length peptide YY analog in mice

scientific article published in September 2017

Investigation of the structural requirements of K-Ras(G12D) selective inhibitory peptide KRpep-2d using alanine scans and cysteine bridging.

scientific article

K-Ras(G12D)-selective inhibitory peptides generated by random peptide T7 phage display technology.

scientific article

Metastin and its variant forms suppress migration of pancreatic cancer cells

scientific article published on February 2004

Potent antiobesity effect of a short-length peptide YY-analogue continuously administered in mice

scientific article

Stereoselective Synthesis of 3,6-Disubstituted-3,6-dihydropyridin-2-ones as Potential Diketopiperazine Mimetics Using Organocopper-Mediatedanti-SN2‘ Reactions and Their Use in the Preparation of Low-Molecule CXCR4 Antagonists

scientific article published on 01 May 2006

Stereoselective synthesis of (Z)-alkene-containing proline dipeptide mimetics

scientific article published on 01 June 2006

Structure-activity relationship study on small peptidic GPR54 agonists.

scientific article published in August 2006

Synthesis of (Z)-Alkene and (E)-Fluoroalkene-Containing Diketopiperazine Mimetics Utilizing Organocopper-Mediated Reduction−Alkylation and Diastereoselectivity Examination Using DFT Calculations

scientific article published on 01 May 2006

Unequivocal Synthesis of (Z)-Alkene and (E)-Fluoroalkene Dipeptide Isosteres To Probe Structural Requirements of the Peptide Transporter PEPT1

scientific article published on 01 February 2006

List of works by Ayumu Niida

A Short-Length Peptide YY Analogue with Anorectic Effect in Mice.

A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres

Antiobesity Effect of a Short-Length Peptide YY Analogue after Continuous Administration in Mice.

Antiobesity and emetic effects of a short-length peptide YY analog and its PEGylated and alkylated derivatives

Crystal Structure of a Human K-Ras G12D Mutant in Complex with GDP and the Cyclic Inhibitory Peptide KRpep-2d.

Design and synthesis of downsized metastin (45-54) analogs with maintenance of high GPR54 agonistic activity

Diastereoselective Synthesis of ψ[(E)-CHCMe]- and ψ[(Z)-CHCMe]-Type Dipeptide Isosteres by Organocopper-Mediatedanti-SN2‘ Reaction

Diastereoselective Synthesis ofψ[(E)-CMeCH]- andψ[(E)-CMeCMe]- Type Dipeptide Isosteres Based on Organocopper-Mediatedanti-SN2‘ Reaction

Diastereoselective synthesis of new psi[(E)-CH=CMe]- and psi[(Z)-CH=CMe]-type alkene dipeptide isosteres by organocopper reagents and application to conformationally restricted cyclic RGD peptidomimetics.

Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres

Highly potent antiobesity effect of a short-length peptide YY analog in mice

Investigation of the structural requirements of K-Ras(G12D) selective inhibitory peptide KRpep-2d using alanine scans and cysteine bridging.

K-Ras(G12D)-selective inhibitory peptides generated by random peptide T7 phage display technology.

Metastin and its variant forms suppress migration of pancreatic cancer cells

Potent antiobesity effect of a short-length peptide YY-analogue continuously administered in mice

Stereoselective Synthesis of 3,6-Disubstituted-3,6-dihydropyridin-2-ones as Potential Diketopiperazine Mimetics Using Organocopper-Mediatedanti-SN2‘ Reactions and Their Use in the Preparation of Low-Molecule CXCR4 Antagonists

Stereoselective synthesis of (Z)-alkene-containing proline dipeptide mimetics

Structure-activity relationship study on small peptidic GPR54 agonists.

Synthesis of (Z)-Alkene and (E)-Fluoroalkene-Containing Diketopiperazine Mimetics Utilizing Organocopper-Mediated Reduction−Alkylation and Diastereoselectivity Examination Using DFT Calculations

Unequivocal Synthesis of (Z)-Alkene and (E)-Fluoroalkene Dipeptide Isosteres To Probe Structural Requirements of the Peptide Transporter PEPT1